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Items: 1 to 20 of 11418

1.

Analysis of GABAA receptor activation by combinations of agonists acting at the same or distinct binding sites.

Shin DJ, Germann AL, Covey DF, Steinbach JH, Akk G.

Mol Pharmacol. 2018 Oct 18. pii: mol.118.113464. doi: 10.1124/mol.118.113464. [Epub ahead of print]

PMID:
30337372
2.

APPLYING THE MONOD-WYMAN-CHANGEUX ALLOSTERIC ACTIVATION MODEL TO PSEUDO-STEADY-STATE RESPONSES FROM GABAA RECEPTORS.

Steinbach JH, Akk G.

Mol Pharmacol. 2018 Oct 17. pii: mol.118.113787. doi: 10.1124/mol.118.113787. [Epub ahead of print]

PMID:
30333132
3.

Involvement of 5-HT1A and 5-HT2A receptors but not α2-adrenoceptors in the acute electrophysiological effects of cariprazine in the rat brain in vivo.

Herman A, El Mansari M, Adham N, Kiss B, Farkas B, Blier P.

Mol Pharmacol. 2018 Oct 15. pii: mol.118.113290. doi: 10.1124/mol.118.113290. [Epub ahead of print]

4.

Pyrimidinyl Biphenylureas Act as Allosteric Modulators to activate Cannabinoid Receptor 1 and initiate β-Arrestin-dependent Responses.

Jagla CAD, Scott CE, Tang Y, Qiao C, Mateo-Semidey GE, Yudowski GA, Lu D, Kendall DA.

Mol Pharmacol. 2018 Oct 15. pii: mol.118.112854. doi: 10.1124/mol.118.112854. [Epub ahead of print]

5.
6.

Physicochemical solubility of and biological sensitivity to long-chain alcohols determine the cutoff chain length in biological activity.

Matsumoto A, Uesono Y.

Mol Pharmacol. 2018 Oct 5. pii: mol.118.112656. doi: 10.1124/mol.118.112656. [Epub ahead of print]

7.

Activated CaMKIIα binds to the mGlu5 metabotropic glutamate receptor and modulates calcium mobilization.

Marks CR, Shonesy BC, Wang X, Stephenson JR, Niswender C, Colbran RJ.

Mol Pharmacol. 2018 Oct 3. pii: mol.118.113142. doi: 10.1124/mol.118.113142. [Epub ahead of print]

8.

Reduced Activity of GGPPS Mutant is Involved in Bisphosphonates-Induced Atypical Fractures.

Lisnyansky M, Kapelushnik N, Ben-Bassat A, Marom M, Loewenstein A, Khananshvili D, Giladi M, Haitin Y.

Mol Pharmacol. 2018 Oct 1. pii: mol.118.113670. doi: 10.1124/mol.118.113670. [Epub ahead of print]

9.

Differential effects of integrin αv knockdown and cilengitide on sensitisation of triple-negative breast cancer and melanoma cells to microtubule poisons.

Stojanovic N, Dekanic A, Paradzik M, Majhen D, Ferencak K, Ruscic J, Bardak I, Supina C, Tomicic MT, Christmann M, Osmak M, Ambriovic-Ristov A.

Mol Pharmacol. 2018 Sep 27. pii: mol.118.113027. doi: 10.1124/mol.118.113027. [Epub ahead of print]

10.

Functional Expression of Organic Anion Transporting Polypeptide 1a4 (Oatp1a4) is Regulated by Transforming Growth Factor-/Activin Receptor-like Kinase 1 (TGF-/ALK1) Signaling at the Blood-Brain Barrier.

Abdullahi W, Brzica H, Hirsch NA, Reilly BG, Ronaldson PT.

Mol Pharmacol. 2018 Sep 27. pii: mol.118.112912. doi: 10.1124/mol.118.112912. [Epub ahead of print]

11.

Modeling and mutational analysis of the binding mode for the multimodal antidepressant drug vortioxetine to the human 5-HT3A receptor.

Ladefoged LK, Munro L, Pedersen AJ, Balle T, Bang-Andersen B, Lummis SCR, Schiott B, Kristensen AS.

Mol Pharmacol. 2018 Sep 26. pii: mol.118.113530. doi: 10.1124/mol.118.113530. [Epub ahead of print]

12.

Homogeneous, real-time NanoBRET binding assays for the histamine H3 and H4 receptor on living cells.

Mocking TAM, Verweij EWE, Vischer HF, Leurs R.

Mol Pharmacol. 2018 Sep 24. pii: mol.118.113373. doi: 10.1124/mol.118.113373. [Epub ahead of print]

13.

Betacellulin (BTC) Biases the EGFR to Dimerize with ErbB3.

Rush JS, Peterson JL, Ceresa BP.

Mol Pharmacol. 2018 Sep 24. pii: mol.118.113399. doi: 10.1124/mol.118.113399. [Epub ahead of print]

14.

Utility of an "Allosteric Site-Impaired" M2 Muscarinic Acetylcholine Receptor as a Novel Construct for Validating Mechanisms of Action of Synthetic and Putative Endogenous Allosteric Modulators.

Von Moo E, Sexton PM, Christopoulos A, Valant C.

Mol Pharmacol. 2018 Nov;94(5):1298-1309. doi: 10.1124/mol.118.112490. Epub 2018 Sep 13.

PMID:
30213802
15.

Effects of HCN Channels in the Rostral Ventrolateral Medulla Contribute to the Cardiovascular Effects of Propofol.

Hu Z, Wu Z, Gao J, Jia Q, Li N, Ouyang Y, Yao S, Chen X.

Mol Pharmacol. 2018 Nov;94(5):1280-1288. doi: 10.1124/mol.118.111898. Epub 2018 Sep 7.

PMID:
30194107
16.

Molecular Characterization of Binding Loop E in the Nematode Cys-Loop GABA Receptor.

Kwaka A, Hassan Khatami M, Foster J, Cochrane E, Habibi SA, de Haan HW, Forrester SG.

Mol Pharmacol. 2018 Nov;94(5):1289-1297. doi: 10.1124/mol.118.112821. Epub 2018 Sep 7.

PMID:
30194106
17.

Activation of Caenorhabditis elegans Levamisole-Sensitive and Mammalian Nicotinic Receptors by the Antiparasitic Bephenium.

Turani O, Hernando G, Corradi J, Bouzat C.

Mol Pharmacol. 2018 Nov;94(5):1270-1279. doi: 10.1124/mol.118.113357. Epub 2018 Sep 6.

PMID:
30190363
18.

Chemoproteomic Discovery of a Ritanserin-Targeted Kinase Network Mediating Apoptotic Cell Death of Lung Tumor Cells.

Campbell ST, Franks CE, Borne AL, Shin M, Zhang L, Hsu KL.

Mol Pharmacol. 2018 Nov;94(5):1246-1255. doi: 10.1124/mol.118.113001. Epub 2018 Aug 29.

PMID:
30158316
19.

Correction to "Identification of AICP as a GluN2C-Selective N-Methyl-D-Aspartate Receptor Superagonist at the GluN1 Glycine Site".

[No authors listed]

Mol Pharmacol. 2018 Oct;94(4):1101-1102. doi: 10.1124/mol.117.108944err. No abstract available.

20.

The Novel Activity of Carbamazepine as an Activation Modulator Extends from NaV1.7 Mutations to the NaV1.8-S242T Mutant Channel from a Patient with Painful Diabetic Neuropathy.

Han C, Themistocleous AC, Estacion M, Dib-Hajj FB, Blesneac I, Macala L, Fratter C, Bennett DL, Waxman SG, Dib-Hajj SD.

Mol Pharmacol. 2018 Nov;94(5):1256-1269. doi: 10.1124/mol.118.113076. Epub 2018 Aug 22.

PMID:
30135145

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