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Items: 18

1.

Rapid approach to complex boronic acids.

Neochoritis CG, Shaabani S, Ahmadianmoghaddam M, Zarganes-Tzitzikas T, Gao L, Novotná M, Mitríková T, Romero AR, Irianti MI, Xu R, Olechno J, Ellson R, Helan V, Kossenjans M, Groves MR, Dömling A.

Sci Adv. 2019 Jul 5;5(7):eaaw4607. doi: 10.1126/sciadv.aaw4607. eCollection 2019 Jul.

2.

MCR Scaffolds Get Hotter with 18F-Labeling.

Zarganes-Tzitzikas T, Clemente GS, Elsinga PH, Dömling A.

Molecules. 2019 Apr 4;24(7). pii: E1327. doi: 10.3390/molecules24071327.

3.

Atorvastatin (Lipitor) by MCR.

Zarganes-Tzitzikas T, Neochoritis CG, Dömling A.

ACS Med Chem Lett. 2019 Feb 7;10(3):389-392. doi: 10.1021/acsmedchemlett.8b00579. eCollection 2019 Mar 14.

4.

Design of indole- and MCR-based macrocycles as p53-MDM2 antagonists.

Neochoritis CG, Kazemi Miraki M, Abdelraheem EMM, Surmiak E, Zarganes-Tzitzikas T, Łabuzek B, Holak TA, Dömling A.

Beilstein J Org Chem. 2019 Feb 20;15:513-520. doi: 10.3762/bjoc.15.45. eCollection 2019.

5.

Application of Silver Nanoparticles in the Multicomponent Reaction Domain: A Combined Catalytic Reduction Methodology to Efficiently Access Potential Hypertension or Inflammation Inhibitors.

Iordanidou D, Zarganes-Tzitzikas T, Neochoritis CG, Dömling A, Lykakis IN.

ACS Omega. 2018 Nov 30;3(11):16005-16013. doi: 10.1021/acsomega.8b02749. Epub 2018 Nov 27.

6.

Synthesis of Highly Substituted Imidazole Uracil Containing Molecules via Ugi-4CR and Passerini-3CR.

Madhavachary R, Zarganes-Tzitzikas T, Patil P, Kurpiewska K, Kalinowska-Tłuścik J, Dömling A.

ACS Comb Sci. 2018 Apr 9;20(4):192-196. doi: 10.1021/acscombsci.7b00145. Epub 2018 Feb 26.

7.

Discovery of chromenes as inhibitors of macrophage migration inhibitory factor.

Kok T, Wapenaar H, Wang K, Neochoritis CG, Zarganes-Tzitzikas T, Proietti G, Eleftheriadis N, Kurpiewska K, Kalinowska-Tłuścik J, Cool RH, Poelarends GJ, Dömling A, Dekker FJ.

Bioorg Med Chem. 2018 Mar 1;26(5):999-1005. doi: 10.1016/j.bmc.2017.12.032. Epub 2017 Dec 24.

8.

Immune Checkpoint PD-1/PD-L1: Is There Life Beyond Antibodies?

Konstantinidou M, Zarganes-Tzitzikas T, Magiera-Mularz K, Holak TA, Dömling A.

Angew Chem Int Ed Engl. 2018 Apr 23;57(18):4840-4848. doi: 10.1002/anie.201710407. Epub 2018 Feb 23. Review.

9.

Bioactive Macrocyclic Inhibitors of the PD-1/PD-L1 Immune Checkpoint.

Magiera-Mularz K, Skalniak L, Zak KM, Musielak B, Rudzinska-Szostak E, Berlicki Ł, Kocik J, Grudnik P, Sala D, Zarganes-Tzitzikas T, Shaabani S, Dömling A, Dubin G, Holak TA.

Angew Chem Int Ed Engl. 2017 Oct 23;56(44):13732-13735. doi: 10.1002/anie.201707707. Epub 2017 Sep 26.

10.

Inhibitors of programmed cell death 1 (PD-1): a patent review (2010-2015).

Zarganes-Tzitzikas T, Konstantinidou M, Gao Y, Krzemien D, Zak K, Dubin G, Holak TA, Dömling A.

Expert Opin Ther Pat. 2016 Sep;26(9):973-7. doi: 10.1080/13543776.2016.1206527. Epub 2016 Jul 6. No abstract available.

11.

Multicomponent Reactions, Union of MCRs and Beyond.

Zarganes-Tzitzikas T, Chandgude AL, Dömling A.

Chem Rec. 2015 Oct;15(5):981-96. doi: 10.1002/tcr.201500201. Epub 2015 Sep 11. Review.

PMID:
26455350
12.

Leuckart-Wallach Route Toward Isocyanides and Some Applications.

Neochoritis CG, Zarganes-Tzitzikas T, Stotani S, Dömling A, Herdtweck E, Khoury K, Dömling A.

ACS Comb Sci. 2015 Sep 14;17(9):493-9. doi: 10.1021/acscombsci.5b00066. Epub 2015 Aug 10.

PMID:
26226194
13.

Concise Synthesis of Tetrazole-keto-piperazines by Two Consecutive Ugi Reactions.

Zarganes-Tzitzikas T, Patil P, Khoury K, Herdtweck E, Dömling A.

European J Org Chem. 2015 Jan;2015(1):51-55. Epub 2014 Nov 17. No abstract available.

14.

Modern Multicomponent Reactions for better Drug Syntheses**

Zarganes-Tzitzikas T, Dömling A.

Org Chem Front. 2014 Sep 1;1(7):834-837.

15.

One-pot five-component synthesis of spirocyclopenta[b]chromene derivatives and their acid-catalyzed rearrangement.

Terzidis MA, Zarganes-Tzitzikas T, Tsimenidis C, Stephanidou-Stephanatou J, Tsoleridis CA, Kostakis GE.

J Org Chem. 2012 Oct 19;77(20):9018-28. doi: 10.1021/jo3014947. Epub 2012 Sep 28.

PMID:
22978377
16.

One-pot synthesis of functionalized spirobenzofuranones via MCR involving 3-cyanochromones.

Zarganes-Tzitzikas T, Terzidis MA, Stephanidou-Stephanatou J, Tsoleridis CA, Kostakis GE.

J Org Chem. 2011 Nov 4;76(21):9008-14. doi: 10.1021/jo201732g. Epub 2011 Oct 12.

PMID:
21992417
17.

Synthesis of 2-keto-imidazoles utilizing N-arylamino-substituted N-heterocyclic carbenes.

Zarganes-Tzitzikas T, Neochoritis CG, Stephanidou-Stephanatou J, Tsoleridis CA.

J Org Chem. 2011 Mar 4;76(5):1468-71. doi: 10.1021/jo102244x. Epub 2011 Jan 20.

PMID:
21250708
18.

One-pot microwave assisted synthesis under green chemistry conditions, antioxidant screening, and cytotoxicity assessments of benzimidazole Schiff bases and pyrimido[1,2-a]benzimidazol-3(4H)-ones.

Neochoritis CG, Zarganes-Tzitzikas T, Tsoleridis CA, Stephanidou-Stephanatou J, Kontogiorgis CA, Hadjipavlou-Litina DJ, Choli-Papadopoulou T.

Eur J Med Chem. 2011 Jan;46(1):297-306. doi: 10.1016/j.ejmech.2010.11.018. Epub 2010 Nov 19.

PMID:
21146903

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