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Items: 30

1.

Saturation limits the contribution of acceleration feedback to balancing against reaction delay.

Zhang L, Stepan G, Insperger T.

J R Soc Interface. 2018 Jan;15(138). pii: 20170771. doi: 10.1098/rsif.2017.0771.

PMID:
29386400
2.

On the analysis of the double Hopf bifurcation in machining processes via centre manifold reduction.

Molnar TG, Dombovari Z, Insperger T, Stepan G.

Proc Math Phys Eng Sci. 2017 Nov;473(2207):20170502. doi: 10.1098/rspa.2017.0502. Epub 2017 Nov 15.

PMID:
29225502
3.

Quantization improves stabilization of dynamical systems with delayed feedback.

Stepan G, Milton JG, Insperger T.

Chaos. 2017 Nov;27(11):114306. doi: 10.1063/1.5006777.

PMID:
29195339
4.

Antiviral Activity of Bictegravir (GS-9883), a Novel Potent HIV-1 Integrase Strand Transfer Inhibitor with an Improved Resistance Profile.

Tsiang M, Jones GS, Goldsmith J, Mulato A, Hansen D, Kan E, Tsai L, Bam RA, Stepan G, Stray KM, Niedziela-Majka A, Yant SR, Yu H, Kukolj G, Cihlar T, Lazerwith SE, White KL, Jin H.

Antimicrob Agents Chemother. 2016 Nov 21;60(12):7086-7097. Print 2016 Dec.

5.

Stabilizing skateboard speed-wobble with reflex delay.

Varszegi B, Takacs D, Stepan G, Hogan SJ.

J R Soc Interface. 2016 Aug;13(121). pii: 20160345. doi: 10.1098/rsif.2016.0345.

6.

Novel (2,6-difluorophenyl)(2-(phenylamino)pyrimidin-4-yl)methanones with restricted conformation as potent non-nucleoside reverse transcriptase inhibitors against HIV-1.

Šimon P, Baszczyňski O, Šaman D, Stepan G, Hu E, Lansdon EB, Jansa P, Janeba Z.

Eur J Med Chem. 2016 Oct 21;122:185-195. doi: 10.1016/j.ejmech.2016.06.026. Epub 2016 Jun 17.

PMID:
27371922
7.

Rapid In Vitro Evaluation of Antiretroviral Barrier to Resistance at Therapeutic Drug Levels.

Mulato A, Hansen D, Thielen A, Porter D, Stepan G, White K, Daeumer M, Cihlar T, Yant SR.

AIDS Res Hum Retroviruses. 2016 Dec;32(12):1237-1247. Epub 2016 Jul 25.

PMID:
27356854
8.

Role of Mitochondrial RNA Polymerase in the Toxicity of Nucleotide Inhibitors of Hepatitis C Virus.

Feng JY, Xu Y, Barauskas O, Perry JK, Ahmadyar S, Stepan G, Yu H, Babusis D, Park Y, McCutcheon K, Perron M, Schultz BE, Sakowicz R, Ray AS.

Antimicrob Agents Chemother. 2015 Nov 23;60(2):806-17. doi: 10.1128/AAC.01922-15. Print 2016 Feb.

9.

On the bistable zone of milling processes.

Dombovari Z, Stepan G.

Philos Trans A Math Phys Eng Sci. 2015 Sep 28;373(2051). pii: 20140409. doi: 10.1098/rsta.2014.0409.

10.

In Vitro Virology Profile of Tenofovir Alafenamide, a Novel Oral Prodrug of Tenofovir with Improved Antiviral Activity Compared to That of Tenofovir Disoproxil Fumarate.

Callebaut C, Stepan G, Tian Y, Miller MD.

Antimicrob Agents Chemother. 2015 Oct;59(10):5909-16. doi: 10.1128/AAC.01152-15. Epub 2015 Jul 6.

11.

Abyssomicin 2 reactivates latent HIV-1 by a PKC- and HDAC-independent mechanism.

León B, Navarro G, Dickey BJ, Stepan G, Tsai A, Jones GS, Morales ME, Barnes T, Ahmadyar S, Tsiang M, Geleziunas R, Cihlar T, Pagratis N, Tian Y, Yu H, Linington RG.

Org Lett. 2015 Jan 16;17(2):262-5. doi: 10.1021/ol503349y. Epub 2015 Jan 5.

12.

Histone deacetylase inhibitor romidepsin induces HIV expression in CD4 T cells from patients on suppressive antiretroviral therapy at concentrations achieved by clinical dosing.

Wei DG, Chiang V, Fyne E, Balakrishnan M, Barnes T, Graupe M, Hesselgesser J, Irrinki A, Murry JP, Stepan G, Stray KM, Tsai A, Yu H, Spindler J, Kearney M, Spina CA, McMahon D, Lalezari J, Sloan D, Mellors J, Geleziunas R, Cihlar T.

PLoS Pathog. 2014 Apr 10;10(4):e1004071. doi: 10.1371/journal.ppat.1004071. eCollection 2014 Apr.

13.

Study of marine natural products including resorcyclic acid lactones from Humicola fuscoatra that reactivate latent HIV-1 expression in an in vitro model of central memory CD4+ T cells.

Mejia EJ, Loveridge ST, Stepan G, Tsai A, Jones GS, Barnes T, White KN, Drašković M, Tenney K, Tsiang M, Geleziunas R, Cihlar T, Pagratis N, Tian Y, Yu H, Crews P.

J Nat Prod. 2014 Mar 28;77(3):618-24. doi: 10.1021/np400889x. Epub 2014 Feb 4.

14.

Inhibition of hepatitis C virus replication by GS-6620, a potent C-nucleoside monophosphate prodrug.

Feng JY, Cheng G, Perry J, Barauskas O, Xu Y, Fenaux M, Eng S, Tirunagari N, Peng B, Yu M, Tian Y, Lee YJ, Stepan G, Lagpacan LL, Jin D, Hung M, Ku KS, Han B, Kitrinos K, Perron M, Birkus G, Wong KA, Zhong W, Kim CU, Carey A, Cho A, Ray AS.

Antimicrob Agents Chemother. 2014;58(4):1930-42. doi: 10.1128/AAC.02351-13. Epub 2014 Jan 13.

15.

Contact patch memory of tyres leading to lateral vibrations of four-wheeled vehicles.

Takács D, Stépán G.

Philos Trans A Math Phys Eng Sci. 2013 May 20;371(1993):20120427. doi: 10.1098/rsta.2012.0427. Print 2013 Jun 28.

16.

9-[2-(R)-(Phosphonomethoxy)propyl]-2,6-diaminopurine (R)-PMPDAP and its prodrugs: optimized preparation, including identification of by-products formed, and antiviral evaluation in vitro.

Krečmerová M, Jansa P, Dračínský M, Sázelová P, Kašička V, Neyts J, Auwerx J, Kiss E, Goris N, Stepan G, Janeba Z.

Bioorg Med Chem. 2013 Mar 1;21(5):1199-208. doi: 10.1016/j.bmc.2012.12.044. Epub 2013 Jan 9.

PMID:
23375089
17.

Acceleration feedback improves balancing against reflex delay.

Insperger T, Milton J, Stépán G.

J R Soc Interface. 2013 Feb;10(79):20120763. doi: 10.1098/rsif.2012.0763.

18.

A novel and efficient one-pot synthesis of symmetrical diamide (bis-amidate) prodrugs of acyclic nucleoside phosphonates and evaluation of their biological activities.

Jansa P, Baszczyňski O, Dračínský M, Votruba I, Zídek Z, Bahador G, Stepan G, Cihlar T, Mackman R, Holý A, Janeba Z.

Eur J Med Chem. 2011 Sep;46(9):3748-54. doi: 10.1016/j.ejmech.2011.05.040. Epub 2011 May 23.

PMID:
21664011
19.

Traffic jams: dynamics and control.

Orosz G, Wilson RE, Stépán G.

Philos Trans A Math Phys Eng Sci. 2010 Oct 13;368(1928):4455-79. doi: 10.1098/rsta.2010.0205.

20.

Delayed feedback of sampled higher derivatives.

Insperger T, Stepan G, Turi J.

Philos Trans A Math Phys Eng Sci. 2010 Jan 28;368(1911):469-82. doi: 10.1098/rsta.2009.0246.

21.

Exciting traffic jams: nonlinear phenomena behind traffic jam formation on highways.

Orosz G, Wilson RE, Szalai R, Stépán G.

Phys Rev E Stat Nonlin Soft Matter Phys. 2009 Oct;80(4 Pt 2):046205. Epub 2009 Oct 6.

PMID:
19905413
22.

Delay effects in the human sensory system during balancing.

Stepan G.

Philos Trans A Math Phys Eng Sci. 2009 Mar 28;367(1891):1195-212. doi: 10.1098/rsta.2008.0278.

23.

Delay effects in brain dynamics. Introduction.

Stepan G.

Philos Trans A Math Phys Eng Sci. 2009 Mar 28;367(1891):1059-62. doi: 10.1098/rsta.2008.0279.

24.

Identification of a 5-HT4 receptor antagonist clinical candidate through side-chain modification.

Clark RD, Jahangir A, Alam M, Rocha C, Lin L, Bjorner B, Nguyen K, Grady C, Williams TJ, Stepan G, Tang HM, Ford AP.

Bioorg Med Chem Lett. 2005 Mar 15;15(6):1697-700.

PMID:
15745824
25.

Global dynamics of low immersion high-speed milling.

Szalai R, Stépán G, Hogan SJ.

Chaos. 2004 Dec;14(4):1069-77.

PMID:
15568921
26.

Effect of YM-44781, YM-44778 and YM-49598, novel tachykinin antagonists, in a drug-induced bladder contraction model.

Choppin A, Groke G, Bringas A, Stepan G, Dillon MP.

Pharmacology. 2002 May;65(2):96-102.

PMID:
11937780
27.

Characterization of the muscarinic receptor in isolated uterus of sham operated and ovariectomized rats.

Choppin A, Stepan GJ, Loury DN, Watson N, Eglen RM.

Br J Pharmacol. 1999 Aug;127(7):1551-8.

28.

Human cloned alpha1A-adrenoceptor isoforms display alpha1L-adrenoceptor pharmacology in functional studies.

Daniels DV, Gever JR, Jasper JR, Kava MS, Lesnick JD, Meloy TD, Stepan G, Williams TJ, Clarke DE, Chang DJ, Ford AP.

Eur J Pharmacol. 1999 Apr 16;370(3):337-43.

PMID:
10334511
29.

Inhibition of interleukin 1 (IL-1) binding and bioactivity in vitro and modulation of acute inflammation in vivo by IL-1 receptor antagonist and anti-IL-1 receptor monoclonal antibody.

McIntyre KW, Stepan GJ, Kolinsky KD, Benjamin WR, Plocinski JM, Kaffka KL, Campen CA, Chizzonite RA, Kilian PL.

J Exp Med. 1991 Apr 1;173(4):931-9.

30.

Effect of aminophylline on cisplatin nephrotoxicity in the rat.

Heidemann HT, Müller S, Mertins L, Stepan G, Hoffmann K, Ohnhaus EE.

Br J Pharmacol. 1989 Jun;97(2):313-8.

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