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Items: 29

1.

Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells.

Zwergel C, Schnekenburger M, Sarno F, Battistelli C, Manara MC, Stazi G, Mazzone R, Fioravanti R, Gros C, Ausseil F, Florean C, Nebbioso A, Strippoli R, Ushijima T, Scotlandi K, Tripodi M, Arimondo PB, Altucci L, Diederich M, Mai A, Valente S.

Clin Epigenetics. 2019 May 6;11(1):68. doi: 10.1186/s13148-019-0663-8.

2.

Histone deacetylases as an epigenetic pillar for the development of hybrid inhibitors in cancer.

Stazi G, Fioravanti R, Mai A, Mattevi A, Valente S.

Curr Opin Chem Biol. 2019 Jun;50:89-100. doi: 10.1016/j.cbpa.2019.03.002. Epub 2019 Apr 12. Review.

PMID:
30986654
3.

Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells.

Stazi G, Battistelli C, Piano V, Mazzone R, Marrocco B, Marchese S, Louie SM, Zwergel C, Antonini L, Patsilinakos A, Ragno R, Viviano M, Sbardella G, Ciogli A, Fabrizi G, Cirilli R, Strippoli R, Marchetti A, Tripodi M, Nomura DK, Mattevi A, Mai A, Valente S.

Eur J Med Chem. 2019 Feb 1;163:722-735. doi: 10.1016/j.ejmech.2018.11.050. Epub 2018 Nov 28.

PMID:
30576903
4.

Application of Small Epigenetic Modulators in Pediatric Medulloblastoma.

Zwergel C, Romanelli A, Stazi G, Besharat ZM, Catanzaro G, Tafani M, Valente S, Mai A.

Front Pediatr. 2018 Dec 3;6:370. doi: 10.3389/fped.2018.00370. eCollection 2018. Review.

5.

Six Years (2012-2018) of Researches on Catalytic EZH2 Inhibitors: The Boom of the 2-Pyridone Compounds.

Fioravanti R, Stazi G, Zwergel C, Valente S, Mai A.

Chem Rec. 2018 Dec;18(12):1818-1832. doi: 10.1002/tcr.201800091. Epub 2018 Oct 19. Review.

PMID:
30338896
6.

Correction to 'Pyrazole-based inhibitors of enhancer of zeste homologue 2 induce apoptosis and autophagy in cancer cells'.

Mellini P, Marrocco B, Borovika D, Polletta L, Carnevale I, Saladini S, Stazi G, Zwergel C, Trapencieris P, Ferretti E, Tafani M, Valente S, Mai A.

Philos Trans R Soc Lond B Biol Sci. 2018 Sep 19;373(1755). pii: 20180305. doi: 10.1098/rstb.2018.0305. No abstract available.

7.

A Quinoline-Based DNA Methyltransferase Inhibitor as a Possible Adjuvant in Osteosarcoma Therapy.

Manara MC, Valente S, Cristalli C, Nicoletti G, Landuzzi L, Zwergel C, Mazzone R, Stazi G, Arimondo PB, Pasello M, Guerzoni C, Picci P, Nanni P, Lollini PL, Mai A, Scotlandi K.

Mol Cancer Ther. 2018 Sep;17(9):1881-1892. doi: 10.1158/1535-7163.MCT-17-0818. Epub 2018 Jun 29.

8.

Trends of LSD1 inhibitors in viral infections.

Zwergel C, Stazi G, Mai A, Valente S.

Future Med Chem. 2018 May 1;10(10):1133-1136. doi: 10.4155/fmc-2018-0065. Epub 2018 May 22. No abstract available.

9.

BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability.

Jennings LE, Schiedel M, Hewings DS, Picaud S, Laurin CMC, Bruno PA, Bluck JP, Scorah AR, See L, Reynolds JK, Moroglu M, Mistry IN, Hicks A, Guzanov P, Clayton J, Evans CNG, Stazi G, Biggin PC, Mapp AK, Hammond EM, Humphreys PG, Filippakopoulos P, Conway SJ.

Bioorg Med Chem. 2018 Jul 15;26(11):2937-2957. doi: 10.1016/j.bmc.2018.05.003. Epub 2018 May 15.

10.

Pyrazole-based inhibitors of enhancer of zeste homologue 2 induce apoptosis and autophagy in cancer cells.

Mellini P, Marrocco B, Borovika D, Polletta L, Carnevale I, Saladini S, Stazi G, Zwergel C, Trapencieris P, Ferretti E, Tafani M, Valente S, Mai A.

Philos Trans R Soc Lond B Biol Sci. 2018 Jun 5;373(1748). pii: 20170150. doi: 10.1098/rstb.2017.0150. Erratum in: Philos Trans R Soc Lond B Biol Sci. 2018 Sep 19;373(1755):.

11.

The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells.

Miele E, Valente S, Alfano V, Silvano M, Mellini P, Borovika D, Marrocco B, Po A, Besharat ZM, Catanzaro G, Battaglia G, Abballe L, Zwergel C, Stazi G, Milite C, Castellano S, Tafani M, Trapencieris P, Mai A, Ferretti E.

Oncotarget. 2017 Aug 2;8(40):68557-68570. doi: 10.18632/oncotarget.19782. eCollection 2017 Sep 15.

12.

Novel coumarin- and quinolinone-based polycycles as cell division cycle 25-A and -C phosphatases inhibitors induce proliferation arrest and apoptosis in cancer cells.

Zwergel C, Czepukojc B, Evain-Bana E, Xu Z, Stazi G, Mori M, Patsilinakos A, Mai A, Botta B, Ragno R, Bagrel D, Kirsch G, Meiser P, Jacob C, Montenarh M, Valente S.

Eur J Med Chem. 2017 Jul 7;134:316-333. doi: 10.1016/j.ejmech.2017.04.012. Epub 2017 Apr 10.

PMID:
28431339
13.

EZH2 inhibitors: a patent review (2014-2016).

Stazi G, Zwergel C, Mai A, Valente S.

Expert Opin Ther Pat. 2017 Jul;27(7):797-813. doi: 10.1080/13543776.2017.1316976. Epub 2017 Apr 20. Review.

PMID:
28394193
14.

LSD1 inhibitors: a patent review (2010-2015).

Stazi G, Zwergel C, Valente S, Mai A.

Expert Opin Ther Pat. 2016 May;26(5):565-80. doi: 10.1517/13543776.2016.1165209. Epub 2016 Mar 28. Review.

PMID:
27019002
15.

Discovery of a Novel Inhibitor of Histone Lysine-Specific Demethylase 1A (KDM1A/LSD1) as Orally Active Antitumor Agent.

Vianello P, Botrugno OA, Cappa A, Dal Zuffo R, Dessanti P, Mai A, Marrocco B, Mattevi A, Meroni G, Minucci S, Stazi G, Thaler F, Trifir├│ P, Valente S, Villa M, Varasi M, Mercurio C.

J Med Chem. 2016 Feb 25;59(4):1501-17. doi: 10.1021/acs.jmedchem.5b01209. Epub 2016 Jan 7.

PMID:
26702542
16.

Daptomycin efficacy in the central nervous system of a patient with disseminated methicillin-resistant Staphylococcus aureus infection: a case report.

Taglietti F, Campanile F, Capone A, Di Caro A, Grilli E, Stazi G, Bertuccio T, Petrosillo N, Stefani S.

J Med Case Rep. 2012 Aug 31;6:264. doi: 10.1186/1752-1947-6-264.

17.

Efficacy of levosimendan in Takotsubo-related cardiogenic shock.

Antonini M, Stazi GV, Cirasa MT, Garotto G, Frustaci A.

Acta Anaesthesiol Scand. 2010 Jan;54(1):119-20. doi: 10.1111/j.1399-6576.2009.02105.x. No abstract available.

PMID:
19961441
18.

Fenoldopam in newborn patients undergoing cardiopulmonary bypass: controlled clinical trial.

Ricci Z, Stazi GV, Di Chiara L, Morelli S, Vitale V, Giorni C, Ronco C, Picardo S.

Interact Cardiovasc Thorac Surg. 2008 Dec;7(6):1049-53. doi: 10.1510/icvts.2008.185025. Epub 2008 Sep 9.

PMID:
18782787
19.

Role of vasopressin in the treatment of anaphylactic shock in a child undergoing surgery for congenital heart disease: a case report.

Di Chiara L, Stazi GV, Ricci Z, Polito A, Morelli S, Giorni C, La Salvia O, Vitale V, Rossi E, Picardo S.

J Med Case Rep. 2008 Feb 5;2:36. doi: 10.1186/1752-1947-2-36.

20.

Inotropic support and peritoneal dialysis adequacy in neonates after cardiac surgery.

Ricci Z, Morelli S, Ronco C, Polito A, Stazi GV, Giorni C, Di Chiara L, Picardo S.

Interact Cardiovasc Thorac Surg. 2008 Feb;7(1):116-20. Epub 2007 Nov 30.

PMID:
18055480
21.

Renal replacement therapy in neonates with congenital heart disease.

Morelli S, Ricci Z, Di Chiara L, Stazi GV, Polito A, Vitale V, Giorni C, Iacoella C, Picardo S.

Contrib Nephrol. 2007;156:428-33.

PMID:
17464154
22.

Non-invasive pressure support ventilation in patients with acute respiratory failure after bilateral lung transplantation.

Rocco M, Conti G, Antonelli M, Bufi M, Costa MG, Alampi D, Ruberto F, Stazi GV, Pietropaoli P.

Intensive Care Med. 2001 Oct;27(10):1622-6.

PMID:
11685303
23.

Internal carotid artery dissection in a patient with Beh├žet's syndrome.

Pannone A, Lucchetti G, Stazi G, Corvi F, Ferguson TL, Massucci M, Zaccaria A.

Ann Vasc Surg. 1998 Sep;12(5):463-7.

PMID:
9732425
24.

[Creatine phosphate: an additive to cardioplegic solutions. Clinical study].

D'Alessandro LC, Cini R, Stazi G, Pucci A, De Benedictis F, Rabitti G, Benhar M, Giacopino F, Pezza E, Cioli G.

Cardiologia. 1987 Mar;32(3):307-13. Italian. No abstract available.

PMID:
3607801
25.

[Paradoxical motion of the interventricular septum in echocardiography during right ventricular volume overload: a new pathogenetic conception].

Pezza V, Stazi GC, Giacopino F, Cini R, Carbone C, Danini M, Iacobellis GF.

Cardiologia. 1984 Dec;29(12):687-705. Italian. No abstract available.

PMID:
6534517
26.

[Indirect ECG signs of inferior infarct].

Puletti M, Borgia C, Jacobellis G, Gradi P, Stazi GC, Curione M.

Boll Soc Ital Cardiol. 1981;26(10):1255-7. Italian. No abstract available.

PMID:
7349151
27.

[The incidence of mitral prolapse in congenital idiopathic scoliosis].

Jacobellis GF, Matteoli S, Stazi GC.

Boll Soc Ital Cardiol. 1981;26(9):815-7. Review. Italian. No abstract available.

PMID:
7052102
28.

[Anaphylatic shock due to sodium dehydrocholate].

Stazi GC, Matteoli S, Righetti G, Puletti M.

Minerva Cardioangiol. 1979 Jun;27(6):407-10. Italian. No abstract available.

PMID:
471265
29.

[Mitral valve prolapse during the acute phase of myocardial infarct].

Jacobellis GF, Matteoli S, Polizzi CA, Ferranti E, Stazi GC, Puletti M.

Boll Soc Ital Cardiol. 1979;24(8):849-54. Review. Italian. No abstract available.

PMID:
399440

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