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Items: 1 to 50 of 58

2.

Further comparison of primary hit identification by different assay technologies and effects of assay measurement variability.

Wu X, Sills MA, Zhang JH.

J Biomol Screen. 2005 Sep;10(6):581-9. Epub 2005 Aug 15.

PMID:
16103421
3.
4.

Comparison of assay technologies for a tyrosine kinase assay generates different results in high throughput screening.

Sills MA, Weiss D, Pham Q, Schweitzer R, Wu X, Wu JJ.

J Biomol Screen. 2002 Jun;7(3):191-214.

PMID:
12097183
5.

The discovery and characterization of an interleukin 6 cytokine family antagonist protein from a marine sponge, Callyspongia sp.

Peppard JV, Loo P, Sills MA, Wennogle L, Wright A, Pomponi S, Cueto M.

Adv Exp Med Biol. 2001;484:77-87. No abstract available.

PMID:
11419009
6.

Microxine, a new cdc2 kinase inhibitor from the Australian marine sponge Microxina species.

Killday KB, Yarwood D, Sills MA, Murphy PT, Hooper JN, Wright AE.

J Nat Prod. 2001 Apr;64(4):525-6.

PMID:
11325241
8.

Digital Imaging as a Detection Method for a Fluorescent Protease Assay in 96-Well and Miniaturized Assay Plate Formats.

Abriola L, Chin M, Fuerst P, Schweitzer R, Sills MA.

J Biomol Screen. 1999;4(3):121-127.

PMID:
10838420
9.

Measurement of cdk4 kinase activity using an affinity peptide-tagging technology.

Wu JJ, Yarwood DR, Sills MA, Chaudhuri B, Muller L, Zurini M, Sills MA.

Comb Chem High Throughput Screen. 2000 Feb;3(1):27-36.

PMID:
10702611
10.

In vitro and in vivo evaluation of an endothelin inhibitor reveals novel K+ channel opening activity.

Webb RL, Hu S, Sills MA, Bazil MK, Cioffi CL, Shetty SS, Lappe RW, Rigel DF.

Biochem Biophys Res Commun. 1996 Oct 3;227(1):176-81.

PMID:
8858121
11.

Measurement of the protein tyrosine kinase activity of c-src using time-resolved fluorometry of europium chelates.

Braunwalder AF, Yarwood DR, Sills MA, Lipson KE.

Anal Biochem. 1996 Jul 1;238(2):159-64.

PMID:
8660605
12.

Characterization of an interleukin 6 cytokine family antagonist protein from a marine sponge, Callyspongia sp.

Peppard JV, Loo P, Sills MA, Munster D, Pomponi SA, Wright AE.

J Biol Chem. 1996 Mar 29;271(13):7281-4.

13.

A solid-phase assay for the determination of protein tyrosine kinase activity of c-src using scintillating microtitration plates.

Braunwaler AF, Yarwood DR, Hall T, Missbach M, Lipson KE, Sills MA.

Anal Biochem. 1996 Feb 1;234(1):23-6.

PMID:
8742077
14.

The unusual binding properties of the endothelin receptor antagonist CGS 27830 distinguishes receptor/agonist interactions.

Chin MH, Cioffi CL, Garay M, Neale RF, Shetty SS, DelGrande D, Mugrage B, Sills MA, Lipson KE.

J Pharmacol Exp Ther. 1996 Jan;276(1):74-83.

PMID:
8558459
16.

Aplysillin A, a thrombin receptor antagonist from the marine sponge Aplysina fistularis fulva.

Gulavita NK, Pomponi SA, Wright AE, Garay M, Sills MA.

J Nat Prod. 1995 Jun;58(6):954-7.

PMID:
7673943
17.

Identification of a receptor-binding region in the core segment of the human anaphylatoxin C5a.

Vlattas I, Sytwu II, Dellureficio J, Stanton J, Braunwalder AF, Galakatos N, Kramer R, Seligmann B, Sills MA, Wasvary J.

J Med Chem. 1994 Aug 19;37(17):2783-90.

PMID:
8064805
18.

The pharmacophore of the human C5a anaphylatoxin.

Toth MJ, Huwyler L, Boyar WC, Braunwalder AF, Yarwood D, Hadala J, Haston WO, Sills MA, Seligmann B, Galakatos N.

Protein Sci. 1994 Aug;3(8):1159-68.

19.

Development of tolerance to the antihypertensive effects of highly selective adenosine A2a agonists upon chronic administration.

Webb RL, Sills MA, Chovan JP, Peppard JV, Francis JE.

J Pharmacol Exp Ther. 1993 Oct;267(1):287-95.

PMID:
8229754
20.

Isolation and structure elucidation of 34-sulfatobastadin 13, an inhibitor of the endothelin A receptor, from a marine sponge of the genus Ianthella.

Gulavita NK, Wright AE, McCarthy PJ, Pomponi SA, Kelly-Borges M, Chin M, Sills MA.

J Nat Prod. 1993 Sep;56(9):1613-7.

PMID:
8254355
21.

Sesquiterpene-derived metabolites from the deep water marine sponge Poecillastra sollasi.

Killday KB, Longley R, McCarthy PJ, Pomponi SA, Wright AE, Neale RF, Sills MA.

J Nat Prod. 1993 Apr;56(4):500-7.

PMID:
8496702
22.

Characterization of the binding of Bolton-Hunter labeled [125I]C5a to human neutrophil, monocyte and U-937 cell membranes.

Braunwalder AF, Musmanno D, Galakatos N, Garlick RH, Haston WO, Rediske JJ, Wennogle L, Seligmann B, Sills MA.

Mol Immunol. 1992 Nov;29(11):1319-24.

PMID:
1406720
23.

[3H]2-phenylaminoadenosine ([3H]CV 1808) labels a novel adenosine receptor in rat brain.

Cornfield LJ, Hu S, Hurt SD, Sills MA.

J Pharmacol Exp Ther. 1992 Nov;263(2):552-61.

PMID:
1331404
24.

Characterization of rat lung endothelin receptor subtypes which are coupled to phosphoinositide hydrolysis.

Cioffi CL, Neale RF Jr, Jackson RH, Sills MA.

J Pharmacol Exp Ther. 1992 Aug;262(2):611-8.

PMID:
1323655
25.

Comparison of antagonist and agonist binding to the leukotriene B4 receptor intact human polymorphonuclear neutrophils (PMN).

Jackson RH, Morrissey MM, Sills MA, Jarvis MF.

J Pharmacol Exp Ther. 1992 Jul;262(1):80-9.

PMID:
1320692
26.

High affinity interleukin-6 binding sites in bovine hypothalamus.

Cornfield LJ, Sills MA.

Eur J Pharmacol. 1991 Sep 4;202(1):113-5.

PMID:
1786797
27.

[3H]CGP 39653: a new N-methyl-D-aspartate antagonist radioligand with low nanomolar affinity in rat brain.

Sills MA, Fagg G, Pozza M, Angst C, Brundish DE, Hurt SD, Wilusz EJ, Williams M.

Eur J Pharmacol. 1991 Jan 3;192(1):19-24.

PMID:
1674916
29.

CGS 18102A, a benzopyranopyridine anxiolytic with 5-HT1 agonist and 5-HT2 antagonist properties.

Sills MA, Bennett DA, Lovell RA, Liebman JM, Wood PL, Glaeser BS, Williams M, Hutchison AJ.

Prog Clin Biol Res. 1990;361:469-75. No abstract available.

PMID:
1981265
30.

[3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain.

Jarvis MF, Schulz R, Hutchison AJ, Do UH, Sills MA, Williams M.

J Pharmacol Exp Ther. 1989 Dec;251(3):888-93.

PMID:
2600819
31.

Benzofuro[2,3-c]pyridin-6-ols: synthesis, affinity for opioid-receptor subtypes, and antinociceptive activity.

Hutchison AJ, de Jesus R, Williams M, Simke JP, Neale RF, Jackson RH, Ambrose F, Barbaz BJ, Sills MA.

J Med Chem. 1989 Sep;32(9):2221-6.

PMID:
2549247
32.

A case of two inversion (10) recombinants in a family.

Roberts P, Williams J, Sills MA.

J Med Genet. 1989 Jul;26(7):461-4.

34.

Synthesis, opioid receptor binding profile, and antinociceptive activity of 1-azaspiro[4.5]decan-10-yl amides.

Fujimoto RA, Boxer J, Jackson RH, Simke JP, Neale RF, Snowhill EW, Barbaz BJ, Williams M, Sills MA.

J Med Chem. 1989 Jun;32(6):1259-65.

PMID:
2542556
35.

2H-[1]benzopyrano[3,4-b]pyridines: synthesis and activity at central monoamine receptors.

Hutchison A, Williams M, de Jesus R, Stone GA, Sylvester L, Clarke FH, Sills MA.

J Med Chem. 1989 Mar;32(3):720-7.

PMID:
2537429
36.

Characterization of the binding of [3H]-CGS 19755: a novel N-methyl-D-aspartate antagonist with nanomolar affinity in rat brain.

Murphy DE, Hutchison AJ, Hurt SD, Williams M, Sills MA.

Br J Pharmacol. 1988 Nov;95(3):932-8.

37.

The NMDA antagonists, CPP and CGS 19755, lack affinity for central benzodiazepine receptors.

Williams M, Loo PS, Sills MA.

Eur J Pharmacol. 1988 Oct 11;155(1-2):185-7.

PMID:
2854072
39.

Central muscarinic cholinergic antagonists block wet-dog shakes produced by the TRH analog MK-771 in the rat.

Sills MA, Mellow AM, Sunderland T, Jacobowitz DM.

Brain Res. 1988 Jun 21;453(1-2):385-8.

PMID:
3135919
40.

Interactions of isamoltane (CGP 361A), an anxiolytic phenoxypropanolamine derivative, with 5-HT1 receptor subtypes in the rat brain.

Waldmeier PC, Williams M, Baumann PA, Bischoff S, Sills MA, Neale RF.

Naunyn Schmiedebergs Arch Pharmacol. 1988 Jun;337(6):609-20.

PMID:
2905765
41.
42.

The N-methyl-D-aspartate receptor complex.

Williams M, Loo PA, Murphy DE, Braunwalder AF, Jarvis MF, Sills MA.

J Recept Res. 1988;8(1-4):195-203.

PMID:
2455046
44.
45.

The novel anticonvulsant MK-801 interacts with central phencyclidine recognition sites in rat brain.

Loo PA, Braunwalder AF, Williams M, Sills MA.

Eur J Pharmacol. 1987 Mar 17;135(2):261-3. No abstract available.

PMID:
3034630
46.
47.

Role of octanoic and decanoic acids in the control of seizures.

Sills MA, Forsythe WI, Haidukewych D.

Arch Dis Child. 1986 Dec;61(12):1173-7.

48.

The medium chain triglyceride diet and intractable epilepsy.

Sills MA, Forsythe WI, Haidukewych D, MacDonald A, Robinson M.

Arch Dis Child. 1986 Dec;61(12):1168-72.

49.

Autoradiographic distribution of 125I-galanin binding sites in the rat central nervous system.

Skofitsch G, Sills MA, Jacobowitz DM.

Peptides. 1986 Nov-Dec;7(6):1029-42.

PMID:
2436195
50.

Iron deficiency alters discrete proteins in rat caudate nucleus and nucleus accumbens.

Youdim MB, Sills MA, Heydorn WE, Creed GJ, Jacobowitz DM.

J Neurochem. 1986 Sep;47(3):794-9.

PMID:
2942640

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