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Items: 28

1.

Assembly of the Entire Carbon Backbone of a Stereoisomer of the Antitumor Marine Natural Product Hemicalide.

Lecourt C, Dhambri S, Yamani K, Boissonnat G, Specklin S, Fleury E, Hammad K, Auclair E, Sablé S, Grondin A, Arimondo PB, Sautel F, Massiot G, Meyer C, Cossy J, Sorin G, Lannou MI, Ardisson J.

Chemistry. 2019 Feb 21;25(11):2745-2749. doi: 10.1002/chem.201806327. Epub 2019 Jan 25.

PMID:
30600846
2.

Intramolecular Diels-Alder Approaches to the Decalin Core of Verongidolide: The Origin of the exo-Selectivity, a DFT Analysis.

Maiga-Wandiam B, Corbu A, Massiot G, Sautel F, Yu P, Lin BW, Houk KN, Cossy J.

J Org Chem. 2018 Jun 1;83(11):5975-5985. doi: 10.1021/acs.joc.8b00566. Epub 2018 May 16.

PMID:
29715016
3.

Elaboration of Sterically Hindered δ-Lactones through Ring-Closing Metathesis: Application to the Synthesis of the C1-C27 Fragment of Hemicalide.

Lecourt C, Boinapally S, Dhambri S, Boissonnat G, Meyer C, Cossy J, Sautel F, Massiot G, Ardisson J, Sorin G, Lannou MI.

J Org Chem. 2016 Dec 16;81(24):12275-12290. Epub 2016 Dec 5.

PMID:
27978725
4.

Anticancer activity of koningic acid and semisynthetic derivatives.

Rahier NJ, Molinier N, Long C, Deshmukh SK, Kate AS, Ranadive P, Verekar SA, Jiotode M, Lavhale RR, Tokdar P, Balakrishnan A, Meignan S, Robichon C, Gomes B, Aussagues Y, Samson A, Sautel F, Bailly C.

Bioorg Med Chem. 2015 Jul 1;23(13):3712-21. doi: 10.1016/j.bmc.2015.04.004. Epub 2015 Apr 9.

PMID:
25937235
5.

Synthetic Studies toward the C32-C46 Segment of Hemicalide. Assignment of the Relative Configuration of the C36-C42 Subunit.

Specklin S, Boissonnat G, Lecourt C, Sorin G, Lannou MI, Ardisson J, Sautel F, Massiot G, Meyer C, Cossy J.

Org Lett. 2015 May 15;17(10):2446-9. doi: 10.1021/acs.orglett.5b00955. Epub 2015 Apr 23.

PMID:
25906322
6.

Cytisine-like alkaloids from Ormosia hosiei Hemsl. & E.H. Wilson.

Pouny I, Batut M, Vendier L, David B, Yi S, Sautel F, Arimondo PB, Massiot G.

Phytochemistry. 2014 Nov;107:97-101. doi: 10.1016/j.phytochem.2014.07.022. Epub 2014 Aug 26.

PMID:
25172516
7.

Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation.

Rilova E, Erdmann A, Gros C, Masson V, Aussagues Y, Poughon-Cassabois V, Rajavelu A, Jeltsch A, Menon Y, Novosad N, Gregoire JM, Vispé S, Schambel P, Ausseil F, Sautel F, Arimondo PB, Cantagrel F.

ChemMedChem. 2014 Mar;9(3):590-601. doi: 10.1002/cmdc.201300420.

8.

Synthetic studies on hemicalide: development of a convergent approach toward the C1-C25 fragment.

Sorin G, Fleury E, Tran C, Prost E, Molinier N, Sautel F, Massiot G, Specklin S, Meyer C, Cossy J, Lannou MI, Ardisson J.

Org Lett. 2013 Sep 20;15(18):4734-7. doi: 10.1021/ol402077e. Epub 2013 Sep 3.

PMID:
24001374
9.

Dichapetalins from Dichapetalum species and their cytotoxic properties.

Long C, Aussagues Y, Molinier N, Marcourt L, Vendier L, Samson A, Poughon V, Chalo Mutiso PB, Ausseil F, Sautel F, Arimondo PB, Massiot G.

Phytochemistry. 2013 Oct;94:184-91. doi: 10.1016/j.phytochem.2013.03.023. Epub 2013 Apr 22.

PMID:
23618620
10.

Relative stereochemical determination and synthesis of the C17-C25 δ-lactone fragment of hemicalide.

Fleury E, Sorin G, Prost E, Pancrazi A, Sautel F, Massiot G, Lannou MI, Ardisson J.

J Org Chem. 2013 Feb 1;78(3):855-64. doi: 10.1021/jo302440a. Epub 2013 Jan 23.

PMID:
23301639
11.

Semisynthetic neoboutomellerone derivatives as ubiquitin-proteasome pathway inhibitors.

Beck J, Guminski Y, Long C, Marcourt L, Derguini F, Plisson F, Grondin A, Vandenberghe I, Vispé S, Brel V, Aussagues Y, Ausseil F, Arimondo PB, Massiot G, Sautel F, Cantagrel F.

Bioorg Med Chem. 2012 Jan 15;20(2):819-31. doi: 10.1016/j.bmc.2011.11.066. Epub 2011 Dec 8.

PMID:
22206869
12.

Proteasome inhibitors from Neoboutonia melleri.

Long C, Beck J, Cantagrel F, Marcourt L, Vendier L, David B, Plisson F, Derguini F, Vandenberghe I, Aussagues Y, Ausseil F, Lavaud C, Sautel F, Massiot G.

J Nat Prod. 2012 Jan 27;75(1):34-47. doi: 10.1021/np200441h. Epub 2011 Dec 14.

PMID:
22168134
13.

Four new carvotanacetone derivatives from Sphaeranthus ukambensis, inhibitors of the ubiquitin-proteasome pathway.

Pouny I, Vispé S, Marcourt L, Long C, Vandenberghe I, Aussagues Y, Raux R, Chalo Mutiso PB, Massiot G, Sautel F.

Planta Med. 2011 Sep;77(14):1605-9. doi: 10.1055/s-0030-1270935. Epub 2011 Mar 21.

PMID:
21425033
14.

Relative stereochemical determination and synthesis of the C1-C17 fragment of a new natural polyketide.

Fleury E, Lannou MI, Bistri O, Sautel F, Massiot G, Pancrazi A, Ardisson J.

J Org Chem. 2009 Sep 18;74(18):7034-45. doi: 10.1021/jo9012833.

PMID:
19694414
15.

F15063, a potential antipsychotic with dopamine D(2)/D(3) antagonist, 5-HT(1A) agonist and D(4) partial agonist properties: (IV) duration of brain D2-like receptor occupancy and antipsychotic-like activity versus plasma concentration in mice.

Assié MB, Bardin L, Auclair A, Consul-Denjean N, Sautel F, Depoortère R, Newman-Tancredi A.

Naunyn Schmiedebergs Arch Pharmacol. 2007 Jun;375(4):241-50. Epub 2007 Apr 24.

PMID:
17453175
16.

Characterization of human cytochrome P450 isoenzymes involved in the metabolism of vinorelbine.

Beulz-Riché D, Grudé P, Puozzo C, Sautel F, Filaquier C, Riché C, Ratanasavanh D.

Fundam Clin Pharmacol. 2005 Oct;19(5):545-53.

PMID:
16176333
18.

High-efficacy 5-HT1A receptor activation causes a curative-like action on allodynia in rats with spinal cord injury.

Colpaert FC, Wu WP, Hao JX, Royer I, Sautel F, Wiesenfeld-Hallin Z, Xu XJ.

Eur J Pharmacol. 2004 Aug 16;497(1):29-33.

PMID:
15321732
19.

Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 receptor agonist.

Pilla M, Perachon S, Sautel F, Garrido F, Mann A, Wermuth CG, Schwartz JC, Everitt BJ, Sokoloff P.

Nature. 1999 Jul 22;400(6742):371-5. Erratum in: Nature 1999 Sep 23;401(6751):403.

PMID:
10432116
20.

Dopamine D3 receptor gene variants and substance abuse in schizophrenia.

Krebs MO, Sautel F, Bourdel MC, Sokoloff P, Schwartz JC, Olié JP, Lôo H, Poirier MF.

Mol Psychiatry. 1998 Jul;3(4):337-41.

PMID:
9702743
21.

Homozygosity at the dopamine D3 receptor gene is associated with opiate dependence.

Duaux E, Gorwood P, Griffon N, Bourdel MC, Sautel F, Sokoloff P, Schwartz JC, Ades J, Lôo H, Poirier MF.

Mol Psychiatry. 1998 Jul;3(4):333-6.

PMID:
9702742
22.

Two intracellular signaling pathways for the dopamine D3 receptor: opposite and synergistic interactions with cyclic AMP.

Griffon N, Pilon C, Sautel F, Schwartz JC, Sokoloff P.

J Neurochem. 1997 Jan;68(1):1-9.

23.

Functional models for the dopamine D3 receptor.

Griffon N, Sautel F, Pilon C, Lévesque D, Sokoloff P, Schwartz JC, Diaz J, Simon P, Costentin J, Mann A, Wermuth CG.

Biochem Soc Trans. 1996 Feb;24(1):193-8. Review. No abstract available.

PMID:
8674660
24.

Antipsychotics with inverse agonist activity at the dopamine D3 receptor.

Griffon N, Pilon C, Sautel F, Schwartz JC, Sokoloff P.

J Neural Transm (Vienna). 1996;103(10):1163-75.

PMID:
9013403
25.

Nafadotride, a potent preferential dopamine D3 receptor antagonist, activates locomotion in rodents.

Sautel F, Griffon N, Sokoloff P, Schwartz JC, Launay C, Simon P, Costentin J, Schoenfelder A, Garrido F, Mann A, et al.

J Pharmacol Exp Ther. 1995 Dec;275(3):1239-46.

PMID:
8531087
26.

The D3 receptor and its relevance in psychiatry.

Schwartz JC, Griffon N, Diaz J, Levesque D, Sautel F, Sokoloff P, Simon P, Costentin J, Garrido F, Mann A, et al.

Int Clin Psychopharmacol. 1995 Sep;10 Suppl 3:15-20. Review.

PMID:
8866761
27.

A functional test identifies dopamine agonists selective for D3 versus D2 receptors.

Sautel F, Griffon N, Lévesque D, Pilon C, Schwartz JC, Sokoloff P.

Neuroreport. 1995 Jan 26;6(2):329-32.

PMID:
7756621
28.

The dopamine D3 receptor and schizophrenia: pharmacological, anatomical and genetic approaches.

Griffon N, Sokoloff P, Diaz J, Lévesque D, Sautel F, Schwartz JC, Simon P, Costentin J, Garrido F, Mann A, et al.

Eur Neuropsychopharmacol. 1995;5 Suppl:3-9. Review.

PMID:
8775753

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