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Items: 16

1.

Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A.

Leaver DJ, Cleary B, Nguyen N, Priebbenow DL, Lagiakos HR, Sanchez J, Xue L, Huang F, Sun Y, Mujumdar P, Mudududdla R, Varghese S, Teguh S, Charman SA, White KL, Katneni K, Cuellar M, Strasser JM, Dahlin JL, Walters MA, Street IP, Monahan BJ, Jarman KE, Sabroux HJ, Falk H, Chung MC, Hermans SJ, Parker MW, Thomas T, Baell JB.

J Med Chem. 2019 Aug 8;62(15):7146-7159. doi: 10.1021/acs.jmedchem.9b00665. Epub 2019 Jul 17.

PMID:
31256587
2.

Carbonic Anhydrase XII Inhibitors Overcome Temozolomide Resistance in Glioblastoma.

Mujumdar P, Kopecka J, Bua S, Supuran CT, Riganti C, Poulsen SA.

J Med Chem. 2019 Apr 25;62(8):4174-4192. doi: 10.1021/acs.jmedchem.9b00282. Epub 2019 Apr 10.

PMID:
30925064
3.

Carbonic Anhydrase XII Inhibitors Overcome P-Glycoprotein-Mediated Resistance to Temozolomide in Glioblastoma.

Salaroglio IC, Mujumdar P, Annovazzi L, Kopecka J, Mellai M, Schiffer D, Poulsen SA, Riganti C.

Mol Cancer Ther. 2018 Dec;17(12):2598-2609. doi: 10.1158/1535-7163.MCT-18-0533. Epub 2018 Sep 25.

PMID:
30254183
4.

Synthesis, structure and bioactivity of primary sulfamate-containing natural products.

Mujumdar P, Bua S, Supuran CT, Peat TS, Poulsen SA.

Bioorg Med Chem Lett. 2018 Sep 15;28(17):3009-3013. doi: 10.1016/j.bmcl.2018.04.038. Epub 2018 Apr 16.

PMID:
29685656
5.

Increasing frequency and spatial extent of concurrent meteorological droughts and heatwaves in India.

Sharma S, Mujumdar P.

Sci Rep. 2017 Nov 14;7(1):15582. doi: 10.1038/s41598-017-15896-3.

6.

Identification of a New Zinc Binding Chemotype by Fragment Screening.

Chrysanthopoulos PK, Mujumdar P, Woods LA, Dolezal O, Ren B, Peat TS, Poulsen SA.

J Med Chem. 2017 Sep 14;60(17):7333-7349. doi: 10.1021/acs.jmedchem.7b00606. Epub 2017 Sep 1.

PMID:
28817930
7.

An Unusual Natural Product Primary Sulfonamide: Synthesis, Carbonic Anhydrase Inhibition, and Protein X-ray Structures of Psammaplin C.

Mujumdar P, Teruya K, Tonissen KF, Vullo D, Supuran CT, Peat TS, Poulsen SA.

J Med Chem. 2016 Jun 9;59(11):5462-70. doi: 10.1021/acs.jmedchem.6b00443. Epub 2016 May 23.

PMID:
27172398
8.

Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases.

Supuran CT, Kalinin S, Tanç M, Sarnpitak P, Mujumdar P, Poulsen SA, Krasavin M.

J Enzyme Inhib Med Chem. 2016;31(sup1):197-202. Epub 2016 May 10.

PMID:
27160030
9.

A hybrid method based upon nonlinear Lamb wave response for locating a delamination in composite laminates.

Yelve NP, Mitra M, Mujumdar PM, Ramadas C.

Ultrasonics. 2016 Aug;70:12-7. doi: 10.1016/j.ultras.2016.04.012. Epub 2016 Apr 19.

PMID:
27115575
10.

Library of diversely substituted 2-(quinolin-4-yl)imidazolines delivers novel non-cytotoxic antitubercular leads.

Krasavin M, Mujumdar P, Parchinsky V, Vinogradova T, Manicheva O, Dogonadze M.

J Enzyme Inhib Med Chem. 2016 Dec;31(6):1146-55. doi: 10.3109/14756366.2015.1101094. Epub 2015 Nov 2.

PMID:
26526717
11.

Natural Product Primary Sulfonamides and Primary Sulfamates.

Mujumdar P, Poulsen SA.

J Nat Prod. 2015 Jun 26;78(6):1470-7. doi: 10.1021/np501015m. Epub 2015 Jun 2. Review.

PMID:
26035239
12.

Panel docking of small-molecule libraries - Prospects to improve efficiency of lead compound discovery.

Sarnpitak P, Mujumdar P, Taylor P, Cross M, Coster MJ, Gorse AD, Krasavin M, Hofmann A.

Biotechnol Adv. 2015 Nov 1;33(6 Pt 1):941-7. doi: 10.1016/j.biotechadv.2015.05.006. Epub 2015 May 27. Review.

13.

Potent, orally available, selective COX-2 inhibitors based on 2-imidazoline core.

Sarnpitak P, Mujumdar P, Morisseau C, Hwang SH, Hammock B, Iurchenko V, Zozulya S, Gavalas A, Geronikaki A, Ivanenkov Y, Krasavin M.

Eur J Med Chem. 2014 Sep 12;84:160-72. doi: 10.1016/j.ejmech.2014.07.023. Epub 2014 Jul 8.

PMID:
25016374
14.

Long-term, progressive, aerobic training increases adiponectin in middle-aged, overweight, untrained males and females.

Mujumdar PP, Duerksen-Hughes PJ, Firek AF, Hessinger DA.

Scand J Clin Lab Invest. 2011 Apr;71(2):101-7. doi: 10.3109/00365513.2011.554995. Epub 2011 Jan 27.

PMID:
21271804
15.

An imprecise fuzzy risk approach for water quality management of a river system.

Rehana S, Mujumdar PP.

J Environ Manage. 2009 Aug;90(11):3653-64. doi: 10.1016/j.jenvman.2009.07.007. Epub 2009 Aug 12.

PMID:
19674829
16.

An inexact optimization approach for river water-quality management.

Karmakar S, Mujumdar PP.

J Environ Manage. 2006 Nov;81(3):233-48. Epub 2006 Mar 20.

PMID:
16545902

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