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Items: 13

1.

Pyrrolidinyl phenylurea derivatives as novel CCR3 antagonists.

Nitta A, Iura Y, Inoue H, Sato I, Morihira K, Kubota H, Morokata T, Takeuchi M, Ohta M, Tsukamoto S, Imaoka T, Takahashi T.

Bioorg Med Chem Lett. 2012 Nov 15;22(22):6876-81. doi: 10.1016/j.bmcl.2012.09.035. Epub 2012 Sep 20.

PMID:
23046963
2.

Discovery and structure-activity relationships of urea derivatives as potent and novel CCR3 antagonists.

Nitta A, Iura Y, Tomioka H, Sato I, Morihira K, Kubota H, Morokata T, Takeuchi M, Ohta M, Tsukamoto S, Imaoka T, Takahashi T.

Bioorg Med Chem Lett. 2012 Aug 1;22(15):4951-4. doi: 10.1016/j.bmcl.2012.06.042. Epub 2012 Jun 20.

PMID:
22749826
3.

Synthesis, biological evaluation, and metabolic stability of acrylamide derivatives as novel CCR3 antagonists.

Sato I, Morihira K, Inami H, Kubota H, Morokata T, Suzuki K, Ohno K, Iura Y, Nitta A, Imaoka T, Takahashi T, Takeuchi M, Ohta M, Tsukamoto S.

Bioorg Med Chem. 2009 Aug 15;17(16):5989-6002. doi: 10.1016/j.bmc.2009.06.066. Epub 2009 Jul 3.

PMID:
19620010
4.

Design and synthesis of 6-fluoro-2-naphthyl derivatives as novel CCR3 antagonists with reduced CYP2D6 inhibition.

Sato I, Morihira K, Inami H, Kubota H, Morokata T, Suzuki K, Iura Y, Nitta A, Imaoka T, Takahashi T, Takeuchi M, Ohta M, Tsukamoto S.

Bioorg Med Chem. 2008 Sep 15;16(18):8607-18. doi: 10.1016/j.bmc.2008.08.006. Epub 2008 Aug 7.

PMID:
18752960
5.

Synthesis and structure-activity relationships of N-{1-[(6-fluoro-2-naphthyl)methyl]piperidin-4-yl}benzamide derivatives as novel CCR3 antagonists.

Sato I, Morihira K, Inami H, Kubota H, Morokata T, Suzuki K, Hamada N, Iura Y, Nitta A, Imaoka T, Takahashi T, Takeuchi M, Ohta M, Tsukamoto S.

Bioorg Med Chem. 2008 Jan 1;16(1):144-56. Epub 2007 Oct 5. Erratum in: Bioorg Med Chem. 2008 Jul 15;16(14):1078.

PMID:
17951061
6.

A dual antagonist for chemokine CCR3 receptor and histamine H1 receptor.

Suzuki K, Morokata T, Morihira K, Sato I, Takizawa S, Kaneko M, Takahashi K, Shimizu Y.

Eur J Pharmacol. 2007 Jun 1;563(1-3):224-32. Epub 2007 Feb 8.

PMID:
17336292
7.

In vitro and in vivo characterization of a novel CCR3 antagonist, YM-344031.

Suzuki K, Morokata T, Morihira K, Sato I, Takizawa S, Kaneko M, Takahashi K, Shimizu Y.

Biochem Biophys Res Commun. 2006 Jan 27;339(4):1217-23. Epub 2005 Dec 5.

PMID:
16343433
8.

A novel, selective, and orally available antagonist for CC chemokine receptor 3.

Morokata T, Suzuki K, Masunaga Y, Taguchi K, Morihira K, Sato I, Fujii M, Takizawa S, Torii Y, Yamamoto N, Kaneko M, Yamada T, Takahashi K, Shimizu Y.

J Pharmacol Exp Ther. 2006 Apr;317(1):244-50. Epub 2005 Dec 9.

PMID:
16339911
9.

Peptide based interleukin-1 beta converting enzyme (ICE) inhibitors: synthesis, structure activity relationships and crystallographic study of the ICE-inhibitor complex.

Okamoto Y, Anan H, Nakai E, Morihira K, Yonetoku Y, Kurihara H, Sakashita H, Terai Y, Takeuchi M, Shibanuma T, Isomura Y.

Chem Pharm Bull (Tokyo). 1999 Jan;47(1):11-21.

PMID:
9987822
10.

Synthesis and evaluation of artificial taxoids with antitumor and multi-drug resistance reversing activities.

Morihira K, Nishimori T, Kusama H, Horiguchi Y, Kuwajima I, Tsuruo T.

Bioorg Med Chem Lett. 1998 Nov 3;8(21):2977-82.

PMID:
9873658
11.

Synthesis of C-ring aromatic taxoids and evaluation of their multi-drug resistance reversing activity.

Morihira K, Nishimori T, Kusama H, Horiguchi Y, Kuwajima I, Tsuruo T.

Bioorg Med Chem Lett. 1998 Nov 3;8(21):2973-6.

PMID:
9873657
12.

Selective muscarinic antagonists. II. Synthesis and antimuscarinic properties of biphenylylcarbamate derivatives.

Naito R, Takeuchi M, Morihira K, Hayakawa M, Ikeda K, Shibanuma T, Isomura Y.

Chem Pharm Bull (Tokyo). 1998 Aug;46(8):1286-94.

PMID:
9734316
13.

Selective muscarinic antagonists. I. Synthesis and antimuscarinic properties of 4-piperidyl benzhydrylcarbamate derivatives.

Naito R, Takeuchi M, Morihira K, Hayakawa M, Ikeda K, Shibanuma T, Isomura Y.

Chem Pharm Bull (Tokyo). 1998 Aug;46(8):1274-85.

PMID:
9734315

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