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Items: 5

1.

A Photoswitchable Agonist for the Histamine H3 Receptor, a prototypic family A G protein-coupled receptor.

Hauwert NJ, Mocking TAM, Da Costa Pereira D, Lion K, Huppelschoten Y, Vischer HF, De Esch IJP, Wijtmans M, Leurs R.

Angew Chem Int Ed Engl. 2019 Feb 8. doi: 10.1002/anie.201813110. [Epub ahead of print]

PMID:
30735597
2.

Homogeneous, Real-Time NanoBRET Binding Assays for the Histamine H3 and H4 Receptors on Living Cells.

Mocking TAM, Verweij EWE, Vischer HF, Leurs R.

Mol Pharmacol. 2018 Dec;94(6):1371-1381. doi: 10.1124/mol.118.113373. Epub 2018 Sep 24.

PMID:
30249614
3.

Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology.

Hauwert NJ, Mocking TAM, Da Costa Pereira D, Kooistra AJ, Wijnen LM, Vreeker GCM, Verweij EWE, De Boer AH, Smit MJ, De Graaf C, Vischer HF, de Esch IJP, Wijtmans M, Leurs R.

J Am Chem Soc. 2018 Mar 28;140(12):4232-4243. doi: 10.1021/jacs.7b11422. Epub 2018 Mar 14.

4.

Structure-kinetics relationships of Capadenoson derivatives as adenosine A1 receptor agonists.

Louvel J, Guo D, Soethoudt M, Mocking TA, Lenselink EB, Mulder-Krieger T, Heitman LH, IJzerman AP.

Eur J Med Chem. 2015 Aug 28;101:681-91. doi: 10.1016/j.ejmech.2015.07.023. Epub 2015 Jul 15.

PMID:
26210506
5.

Agonists for the adenosine A1 receptor with tunable residence time. A Case for nonribose 4-amino-6-aryl-5-cyano-2-thiopyrimidines.

Louvel J, Guo D, Agliardi M, Mocking TA, Kars R, Pham TP, Xia L, de Vries H, Brussee J, Heitman LH, Ijzerman AP.

J Med Chem. 2014 Apr 24;57(8):3213-22. doi: 10.1021/jm401643m. Epub 2014 Apr 3.

PMID:
24669958

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