Format
Sort by
Items per page

Send to

Choose Destination

Search results

Items: 10

1.

From UTP to AR-C118925, the discovery of a potent non nucleotide antagonist of the P2Y2 receptor.

Kindon N, Davis A, Dougall I, Dixon J, Johnson T, Walters I, Thom S, McKechnie K, Meghani P, Stocks MJ.

Bioorg Med Chem Lett. 2017 Nov 1;27(21):4849-4853. doi: 10.1016/j.bmcl.2017.09.043. Epub 2017 Sep 21.

PMID:
28958619
2.

Discovery and evaluation of a novel monocyclic series of CXCR2 antagonists.

Austin RP, Bennion C, Bonnert RV, Cheema L, Cook AR, Cox RJ, Ebden MR, Gaw A, Grime K, Meghani P, Nicholls D, Phillips C, Smith N, Steele J, Stonehouse JP.

Bioorg Med Chem Lett. 2015 Apr 1;25(7):1616-20. doi: 10.1016/j.bmcl.2015.01.067. Epub 2015 Feb 3.

PMID:
25708618
3.

Identification of a putative intracellular allosteric antagonist binding-site in the CXC chemokine receptors 1 and 2.

Nicholls DJ, Tomkinson NP, Wiley KE, Brammall A, Bowers L, Grahames C, Gaw A, Meghani P, Shelton P, Wright TJ, Mallinder PR.

Mol Pharmacol. 2008 Nov;74(5):1193-202. doi: 10.1124/mol.107.044610. Epub 2008 Aug 1.

PMID:
18676678
4.

Novel N-aryl and N-heteroaryl sulfamide synthesis via palladium cross coupling.

Alcaraz L, Bennion C, Morris J, Meghani P, Thom SM.

Org Lett. 2004 Aug 5;6(16):2705-8.

PMID:
15281749
5.

New Lewis-basic N-oxides as chiral organocatalysts in asymmetric allylation of aldehydes.

Malkov AV, Bell M, Orsini M, Pernazza D, Massa A, Herrmann P, Meghani P, Kocovský P.

J Org Chem. 2003 Dec 12;68(25):9659-68.

PMID:
14656092
6.

Synthesis of new chiral 2,2'-bipyridine ligands and their application in copper-catalyzed asymmetric allylic oxidation and cyclopropanation.

Malkov AV, Pernazza D, Bell M, Bella M, Massa A, Teplý F, Meghani P, Kocovský P.

J Org Chem. 2003 Jun 13;68(12):4727-42.

PMID:
12790576
7.

Chiral 2,2'-bipyridine-type N-monoxides as organocatalysts in the enantioselective allylation of aldehydes with allyltrichlorosilane.

Malkov AV, Orsini M, Pernazza D, Muir KW, Langer V, Meghani P, Kocovský P.

Org Lett. 2002 Mar 21;4(6):1047-9.

PMID:
11893218
8.

The medicinal chemistry of the P2 receptor family.

Guile SD, Ince F, Ingall AH, Kindon ND, Meghani P, Mortimore MP.

Prog Med Chem. 2001;38:115-87. Review. No abstract available.

PMID:
11774794
9.

Lead generation using pharmacophore mapping and three-dimensional database searching: application to muscarinic M(3) receptor antagonists.

Marriott DP, Dougall IG, Meghani P, Liu YJ, Flower DR.

J Med Chem. 1999 Aug 26;42(17):3210-6.

PMID:
10464008
10.

(R)-2-(3-mercapto-2(S)-methyl-1-oxo-propoxy)-3-(methylthio)propanoic acid, the first ultra-short-acting angiotensin converting enzyme inhibitor.

Baxter AJ, Carr RD, Eyley SC, Fraser-Rae L, Hallam C, Harper ST, Hurved PA, King SJ, Meghani P.

J Med Chem. 1992 Oct 2;35(20):3718-20. No abstract available.

PMID:
1433185

Supplemental Content

Loading ...
Support Center