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Items: 30

1.

Novel auristatin E-based albumin-binding prodrugs with superior anticancer efficacy in vivo compared to the parent compound.

Pes L, Koester SD, Magnusson JP, Chercheja S, Medda F, Abu Ajaj K, Rognan D, Daum S, Nollmann FI, Garcia Fernandez J, Perez Galan P, Walter HK, Warnecke A, Kratz F.

J Control Release. 2019 Feb 28;296:81-92. doi: 10.1016/j.jconrel.2019.01.010. Epub 2019 Jan 11.

PMID:
30639692
2.

A Versatile Strategy for the Synthesis of 4,5-Dihydroxy-2,3-Pentanedione (DPD) and Related Compounds as Potential Modulators of Bacterial Quorum Sensing.

Stotani S, Gatta V, Medda F, Padmanaban M, Karawajczyk A, Tammela P, Giordanetto F, Tzalis D, Collina S.

Molecules. 2018 Oct 6;23(10). pii: E2545. doi: 10.3390/molecules23102545.

3.

Dataset of the livability performance of the city of Birmingham, UK, as measured by its citizen wellbeing, resource security, resource efficiency and carbon emissions.

Leach JM, Lee SE, Boyko CT, Coulton CJ, Cooper R, Smith N, Joffe H, Büchs M, Hale JD, Sadler JP, Braithwaite PA, Blunden LS, De Laurentiis V, Hunt DVL, Bahaj AS, Barnes K, Bouch CJ, Bourikas L, Cavada M, Chilvers A, Clune SJ, Collins B, Cosgrave E, Dunn N, Falkingham J, James P, Kwami C, Locret-Collet M, Medda F, Ortegon A, Pollastri S, Popan C, Psarikidou K, Tyler N, Urry J, Wu Y, Zeeb V, Rogers CDF.

Data Brief. 2017 Oct 13;15:691-695. doi: 10.1016/j.dib.2017.10.004. eCollection 2017 Dec.

4.

Inhibitors to Overcome Secondary Mutations in the Stem Cell Factor Receptor KIT.

Kaitsiotou H, Keul M, Hardick J, Mühlenberg T, Ketzer J, Ehrt C, Krüll J, Medda F, Koch O, Giordanetto F, Bauer S, Rauh D.

J Med Chem. 2017 Nov 9;60(21):8801-8815. doi: 10.1021/acs.jmedchem.7b00841. Epub 2017 Oct 24.

PMID:
28991465
5.

Assessment of eating disorders with the diabetes eating problems survey - revised (DEPS-R) in a representative sample of insulin-treated diabetic patients: a validation study in Italy.

Pinna F, Diana E, Sanna L, Deiana V, Manchia M, Nicotra E, Fiorillo A, Albert U, Nivoli A, Volpe U, Atti AR, Ferrari S, Medda F, Atzeni MG, Manca D, Mascia E, Farci F, Ghiani M, Cau R, Tuveri M, Cossu E, Loy E, Mereu A, Mariotti S, Carpiniello B.

BMC Psychiatry. 2017 Jul 19;17(1):262. doi: 10.1186/s12888-017-1434-8.

6.

Total synthesis of dehaloperophoramidine using a highly diastereoselective Hosomi-Sakurai reaction.

Wilkie RP, Neal AR, Johnston CA, Voute N, Lancefield CS, Stell MD, Medda F, Makiyi EF, Turner EM, Stephen Ojo O, Slawin AM, Lebl T, Mullen P, Harrison DJ, Ireland CM, Westwood NJ.

Chem Commun (Camb). 2016 Sep 14;52(71):10747-50. doi: 10.1039/c6cc05747k. Epub 2016 Aug 10.

PMID:
27507662
7.

Design and Synthesis of Fsp(3)-Rich, Bis-Spirocyclic-Based Compound Libraries for Biological Screening.

Stotani S, Lorenz C, Winkler M, Medda F, Picazo E, Ortega Martinez R, Karawajczyk A, Sanchez-Quesada J, Giordanetto F.

ACS Comb Sci. 2016 Jun 13;18(6):330-6. doi: 10.1021/acscombsci.6b00005. Epub 2016 May 26.

PMID:
27163646
8.

DYRK1A inhibition as potential treatment for Alzheimer's disease.

Stotani S, Giordanetto F, Medda F.

Future Med Chem. 2016 Apr;8(6):681-96. doi: 10.4155/fmc-2016-0013. Epub 2016 Apr 13. Review.

PMID:
27073990
9.

Branching cascades provide access to two amino-oxazoline compound libraries.

Murali A, Medda F, Winkler M, Giordanetto F, Kumar K.

Bioorg Med Chem. 2015 Jun 1;23(11):2656-65. doi: 10.1016/j.bmc.2015.01.009. Epub 2015 Jan 13.

10.
11.

Synthesis of diverse nitrogen-enriched heterocyclic scaffolds using a suite of tunable one-pot multicomponent reactions.

Martinez-Ariza G, Ayaz M, Medda F, Hulme C.

J Org Chem. 2014 Jun 6;79(11):5153-62. doi: 10.1021/jo500723d. Epub 2014 May 19.

12.

3-(4-Bromo-phen-yl)-1-butyl-5-[1-(2-chloro-6-methyl-phen-yl)-1H-tetra-zol-5-yl]imidazolidine-2,4-dione.

Hall GB, Medda F, Roberts SA, Hulme C.

Acta Crystallogr Sect E Struct Rep Online. 2013 Jun 15;69(Pt 7):o1102-3. doi: 10.1107/S1600536813016000. eCollection 2013.

13.

Synthesis and biological activity of aminophthalazines and aminopyridazines as novel inhibitors of PGE2 production in cells.

Medda F, Sells E, Chang HH, Dietrich J, Chappeta S, Smith B, Gokhale V, Meuillet EJ, Hulme C.

Bioorg Med Chem Lett. 2013 Jan 15;23(2):528-31. doi: 10.1016/j.bmcl.2012.11.030. Epub 2012 Nov 21.

14.

Recent advances in the design, synthesis, and biological evaluation of selective DYRK1A inhibitors: a new avenue for a disease modifying treatment of Alzheimer's?

Smith B, Medda F, Gokhale V, Dunckley T, Hulme C.

ACS Chem Neurosci. 2012 Nov 21;3(11):857-72. doi: 10.1021/cn300094k. Epub 2012 Aug 28. Review.

15.

Synthesis and biological activity of 2-aminothiazoles as novel inhibitors of PGE2 production in cells.

Smith B, Chang HH, Medda F, Gokhale V, Dietrich J, Davis A, Meuillet EJ, Hulme C.

Bioorg Med Chem Lett. 2012 May 15;22(10):3567-70. doi: 10.1016/j.bmcl.2012.03.013. Epub 2012 Mar 28.

16.
17.

Novel cambinol analogs as sirtuin inhibitors: synthesis, biological evaluation, and rationalization of activity.

Medda F, Russell RJ, Higgins M, McCarthy AR, Campbell J, Slawin AM, Lane DP, Lain S, Westwood NJ.

J Med Chem. 2009 May 14;52(9):2673-82. doi: 10.1021/jm8014298.

18.

Gonadotropin-releasing hormone receptor levels and cell context affect tumor cell responses to agonist in vitro and in vivo.

Morgan K, Stewart AJ, Miller N, Mullen P, Muir M, Dodds M, Medda F, Harrison D, Langdon S, Millar RP.

Cancer Res. 2008 Aug 1;68(15):6331-40. doi: 10.1158/0008-5472.CAN-08-0197.

19.

[Congenital malformations of the female genital tract and gestation capacity].

Marcello C, Corda F, Medda F, Silvetti E, Lecca U.

Ann Ostet Ginecol Med Perinat. 1988 Jul-Aug;109(4):219-28. Italian. No abstract available.

PMID:
3232910
20.

HSV2 and cervical intraepithelial neoplasia: cytological, histological and serological features.

Puligheddu P, Nieddu R, Medda F, Marcello C, Lecca U.

Clin Exp Obstet Gynecol. 1988;15(3):88-93.

PMID:
3402090
21.

Activity of interferon beta in condylomata with dysplastic lesion of the uterine cervix.

Puligheddu P, Marcello C, Medda F, Parodo G, Setzu A, Lecca U.

Eur J Gynaecol Oncol. 1988;9(2):161-2.

PMID:
3383896
22.

Hormonal profile and androgen status during the menstrual cycle in women with acne.

Medda F, Nieddu R, Fiore R, Marcello C, Lecca U.

Clin Exp Obstet Gynecol. 1988;15(4):137-42.

PMID:
2976617
23.

Carcinoma IB of the endometrium: spread and prognostic factors.

Lecca U, Medda F, Parodo G, Puligheddu P, Marcello C.

Eur J Gynaecol Oncol. 1987;8(2):127-30.

PMID:
3569330
24.

Management, therapy and outcome of treatment in women with pelvic endometriosis.

Parodo G, Marcello C, Medda F, Puligheddu P, Rassu G, Fiore R, Lecca U.

Clin Exp Obstet Gynecol. 1987;14(3-4):169-74.

PMID:
3454724
25.

Short term treatment with ketoconazole: effects on gonadal and adrenal steroidogenesis in women.

Medda F, Puligheddu P, Parodo G, Marcello C, Aste N, Pascalis P, Pia G, Lecca U.

Clin Exp Obstet Gynecol. 1987;14(3-4):161-6.

PMID:
2970350
26.

Ovarian metastasis in breast cancer.

Lecca U, Medda F, Marcello C, Mattana C, Nasi A, Valdes E, Ferreli A.

Eur J Gynaecol Oncol. 1980 Dec;1(3):168-74. No abstract available.

PMID:
7341266
27.

Variations of plasma CEA levels in gynecologic malignancies: incidence, significance and changes occurring in response to therapy.

Lecca U, Marcello C, Medda F, Mattana C, Manca P, Fodde M, Caminiti F.

Eur J Gynaecol Oncol. 1980 Dec;1(3):150-7.

PMID:
7341264
28.

[Hypophyseal response to the administration of LH-RH based on the plasma level of estradiol in normal women and patients with amenorrhea].

Paoletti AM, Melis GB, Medda F, Genazzani AR, Fioretti P.

Ann Ostet Ginecol Med Perinat. 1978 Jul-Aug;99(4):259-70. Italian. No abstract available.

PMID:
371486
29.

[Circadian changes in protein and steroid hormones in normal females and males].

Melis GB, Paoletti AM, Murru S, Medda F, Fioretti P.

Ann Ostet Ginecol Med Perinat. 1978 Jan-Feb;99(1):47-55. Italian. No abstract available.

PMID:
646280
30.

Inhibitory effect of prostaglandin F2alpha (PgF2alpha) on puerperal lactation.

Fioretti P, Nasi A, Medda F, De Murtas M, Melis GB, Caminiti F.

Acta Eur Fertil. 1977 Sep;8(3):265-71.

PMID:
920042

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