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Items: 1 to 50 of 287

1.

Role of Histamine H₃ Receptor Antagonists on Intraocular Pressure Reduction in Rabbit Models of Transient Ocular Hypertension and Glaucoma.

Lanzi C, Lucarini L, Durante M, Sgambellone S, Pini A, Catarinicchia S, Łażewska D, Kieć-Kononowicz K, Stark H, Masini E.

Int J Mol Sci. 2019 Feb 24;20(4). pii: E981. doi: 10.3390/ijms20040981.

2.

Urban Growth, Land-use Efficiency and Local Socioeconomic Context: A Comparative Analysis of 417 Metropolitan Regions in Europe.

Masini E, Tomao A, Barbati A, Corona P, Serra P, Salvati L.

Environ Manage. 2019 Mar;63(3):322-337. doi: 10.1007/s00267-018-1119-1. Epub 2018 Nov 17.

PMID:
30448998
3.

A Selective Histamine H4 Receptor Antagonist, JNJ7777120, Is Protective in a Rat Model of Transient Cerebral Ischemia.

Dettori I, Gaviano L, Melani A, Lucarini L, Durante M, Masini E, Pedata F.

Front Pharmacol. 2018 Oct 29;9:1231. doi: 10.3389/fphar.2018.01231. eCollection 2018.

4.

Reduced Susceptibility to Sugar-Induced Metabolic Derangements and Impairments of Myocardial Redox Signaling in Mice Chronically Fed with D-Tagatose when Compared to Fructose.

Collotta D, Lucarini L, Chiazza F, Cento AS, Durante M, Sgambellone S, Chini J, Baratta F, Aragno M, Mastrocola R, Masini E, Collino M.

Oxid Med Cell Longev. 2018 Sep 19;2018:5042428. doi: 10.1155/2018/5042428. eCollection 2018.

5.

Relationship between inflammatory parameters and cardiovascular and lifestyle factors in the Mugello study oldest old.

Molino Lova R, Vassalle C, Masini E, Del Ry S, Cabiati M, Pasquini G, Macchi C.

Biomark Med. 2018 Oct;12(10):1115-1124. doi: 10.2217/bmm-2017-0441. Epub 2018 Sep 11.

PMID:
30203672
6.

Identification of Bivalent Ligands with Melatonin Receptor Agonist and Fatty Acid Amide Hydrolase (FAAH) Inhibitory Activity That Exhibit Ocular Hypotensive Effect in the Rabbit.

Spadoni G, Bedini A, Furiassi L, Mari M, Mor M, Scalvini L, Lodola A, Ghidini A, Lucini V, Dugnani S, Scaglione F, Piomelli D, Jung KM, Supuran CT, Lucarini L, Durante M, Sgambellone S, Masini E, Rivara S.

J Med Chem. 2018 Sep 13;61(17):7902-7916. doi: 10.1021/acs.jmedchem.8b00893. Epub 2018 Sep 4.

PMID:
30126274
7.

Variability in distribution and use of tuberculosis diagnostic tests in Kenya: a cross-sectional survey.

Oliwa JN, Maina J, Ayieko P, Gathara D, Kathure IA, Masini E, Van't Hoog AH, van Hensbroek MB, English M.

BMC Infect Dis. 2018 Jul 16;18(1):328. doi: 10.1186/s12879-018-3237-z.

8.

The non-cylindrical crustal architecture of the Pyrenees.

Chevrot S, Sylvander M, Diaz J, Martin R, Mouthereau F, Manatschal G, Masini E, Calassou S, Grimaud F, Pauchet H, Ruiz M.

Sci Rep. 2018 Jun 25;8(1):9591. doi: 10.1038/s41598-018-27889-x.

9.

Epidemiology of Pediatric Tuberculosis in Kenya and Risk Factors for Mortality during Treatment: A National Retrospective Cohort Study.

Onyango DO, Yuen CM, Masini E, Borgdorff MW.

J Pediatr. 2018 Oct;201:115-121. doi: 10.1016/j.jpeds.2018.05.017. Epub 2018 Jun 6.

PMID:
29885751
10.

Targeting Serotonin 2A and Adrenergic α1 Receptors for Ocular Antihypertensive Agents: Discovery of 3,4-Dihydropyrazino[1,2-b]indazol-1(2H)-one Derivatives.

Furlotti G, Alisi MA, Cazzolla N, Ceccacci F, Garrone B, Gasperi T, La Bella A, Leonelli F, Loreto MA, Magarò G, Mangano G, Bettolo RM, Masini E, Miceli M, Migneco LM, Vitiello M.

ChemMedChem. 2018 Aug 10;13(15):1597-1607. doi: 10.1002/cmdc.201800199. Epub 2018 Jul 9.

PMID:
29873449
11.

Impact of a national nutritional support programme on loss to follow-up after tuberculosis diagnosis in Kenya.

Mansour O, Masini EO, Kim BJ, Kamene M, Githiomi MM, Hanson CL.

Int J Tuberc Lung Dis. 2018 Jun 1;22(6):649-654. doi: 10.5588/ijtld.17.0537.

PMID:
29862949
12.

Discovery of β-Adrenergic Receptors Blocker-Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy.

Nocentini A, Ceruso M, Bua S, Lomelino CL, Andring JT, McKenna R, Lanzi C, Sgambellone S, Pecori R, Matucci R, Filippi L, Gratteri P, Carta F, Masini E, Selleri S, Supuran CT.

J Med Chem. 2018 Jun 28;61(12):5380-5394. doi: 10.1021/acs.jmedchem.8b00625. Epub 2018 Jun 13.

PMID:
29851481
13.

2-Benzylpiperazine: A new scaffold for potent human carbonic anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents.

Chiaramonte N, Bua S, Ferraroni M, Nocentini A, Bonardi A, Bartolucci G, Durante M, Lucarini L, Chiapponi D, Dei S, Manetti D, Teodori E, Gratteri P, Masini E, Supuran CT, Romanelli MN.

Eur J Med Chem. 2018 May 10;151:363-375. doi: 10.1016/j.ejmech.2018.04.002. Epub 2018 Apr 3.

PMID:
29635168
14.

Fructose liquid and solid formulations differently affect gut integrity, microbiota composition and related liver toxicity: a comparative in vivo study.

Mastrocola R, Ferrocino I, Liberto E, Chiazza F, Cento AS, Collotta D, Querio G, Nigro D, Bitonto V, Cutrin JC, Rantsiou K, Durante M, Masini E, Aragno M, Cordero C, Cocolin L, Collino M.

J Nutr Biochem. 2018 May;55:185-199. doi: 10.1016/j.jnutbio.2018.02.003. Epub 2018 Feb 13.

PMID:
29539590
15.

ERRATUM.

Mini E, Landini I, Lucarini L, Lapucci A, Napoli C, Perrone G, Tassi R, Masini E, Moroni F, Nobili S.

Oncol Res. 2018 Mar 5;26(2):333-334. doi: 10.3727/096504018X15187172557369.

PMID:
29514732
16.

Methadone Dose Adjustments, Plasma R-Methadone Levels and Therapeutic Outcome of Heroin Users: A Randomized Clinical Trial.

Mannaioni G, Lanzi C, Lotti M, Galli V, Totti A, Pacileo I, Sili M, Pracucci C, Dilaghi A, Bertieri L, Quaranta M, Orsini F, Occupati B, Michahelles A, Ciuti R, Bianchini E, Fabbro G, Biggeri A, Masini E, Moroni F.

Eur Addict Res. 2018;24(1):9-18. doi: 10.1159/000485029. Epub 2018 Jan 31.

PMID:
29393208
17.

Plasmatic carbonic anhydrase IX as a diagnostic marker for clear cell renal cell carcinoma.

Lucarini L, Magnelli L, Schiavone N, Crisci A, Innocenti A, Puccetti L, Cianchi F, Peri S, Supuran CT, Papucci L, Masini E.

J Enzyme Inhib Med Chem. 2018 Dec;33(1):234-240. doi: 10.1080/14756366.2017.1411350.

PMID:
29251173
18.

Reduction of HIV-associated excess mortality by antiretroviral treatment among tuberculosis patients in Kenya.

Onyango DO, Yuen CM, Cain KP, Ngari F, Masini EO, Borgdorff MW.

PLoS One. 2017 Nov 16;12(11):e0188235. doi: 10.1371/journal.pone.0188235. eCollection 2017.

19.

Using Patient-Pathway Analysis to Inform a Differentiated Program Response to Tuberculosis: The Case of Kenya.

Masini E, Hanson C, Ogoro J, Brown J, Ngari F, Mingkwan P, Makayova J, Osberg M.

J Infect Dis. 2017 Nov 6;216(suppl_7):S714-S723. doi: 10.1093/infdis/jix381.

20.

Activation of ERK/CREB pathway in noradrenergic neurons contributes to hypernociceptive phenotype in H4 receptor knockout mice after nerve injury.

Sanna MD, Mello T, Masini E, Galeotti N.

Neuropharmacology. 2018 Jan;128:340-350. doi: 10.1016/j.neuropharm.2017.10.025. Epub 2017 Oct 28.

PMID:
29107625
21.

Paths to Change: Bio-Economic Factors, Geographical Gradients and the Land-Use Structure of Italy.

Masini E, Barbati A, Bencardino M, Carlucci M, Corona P, Salvati L.

Environ Manage. 2018 Jan;61(1):116-131. doi: 10.1007/s00267-017-0950-0. Epub 2017 Oct 25.

PMID:
29071552
22.

gem-Dinitroalkyl Benzenes: A Novel Class of IOP-Lowering Agents for the Treatment of Ocular Hypertension.

Blangetti M, Rolando B, Marini E, Chegaev K, Guglielmo S, Lazzarato L, Lucarini L, Masini E, Fruttero R.

ACS Med Chem Lett. 2017 Sep 13;8(10):1054-1059. doi: 10.1021/acsmedchemlett.7b00264. eCollection 2017 Oct 12.

23.

1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads.

Ferraroni M, Lucarini L, Masini E, Korsakov M, Scozzafava A, Supuran CT, Krasavin M.

Bioorg Med Chem. 2017 Sep 1;25(17):4560-4565. doi: 10.1016/j.bmc.2017.06.054. Epub 2017 Jul 11.

PMID:
28728897
24.

Diabetes and pre-diabetes in tuberculosis patients in western Kenya using point-of-care glycated haemoglobin.

Owiti P, Keter A, Harries AD, Pastakia S, Wambugu C, Kirui N, Kasera G, Momanyi R, Masini E, Some F, Gardner A.

Public Health Action. 2017 Jun 21;7(2):147-154. doi: 10.5588/pha.16.0114.

25.

The Inhibitory Effects of HYDAMTIQ, a Novel PARP Inhibitor, on Growth in Human Tumor Cell Lines With Defective DNA Damage Response Pathways.

Mini E, Landini I, Lucarini L, Lapucci A, Napoli C, Perrone G, Tassi R, Masini E, Moroni F, Nobili S.

Oncol Res. 2017 Nov 2;25(9):1441-1451. doi: 10.3727/096504017X14926854178616. Epub 2017 Apr 20.

PMID:
28429680
26.

New furoxan derivatives for the treatment of ocular hypertension.

Blangetti M, Rolando B, Chegaev K, Guglielmo S, Lazzarato L, Durante M, Masini E, Almirante N, Bastia E, Impagnatiello F, Fruttero R, Gasco A.

Bioorg Med Chem Lett. 2017 Feb 1;27(3):479-483. doi: 10.1016/j.bmcl.2016.12.041. Epub 2016 Dec 18.

27.

Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations.

Nocentini A, Ferraroni M, Carta F, Ceruso M, Gratteri P, Lanzi C, Masini E, Supuran CT.

J Med Chem. 2016 Dec 8;59(23):10692-10704. Epub 2016 Nov 21.

PMID:
27933963
28.

Behavioural phenotype of histamine H4 receptor knockout mice: Focus on central neuronal functions.

Sanna MD, Ghelardini C, Thurmond RL, Masini E, Galeotti N.

Neuropharmacology. 2017 Mar 1;114:48-57. doi: 10.1016/j.neuropharm.2016.11.023. Epub 2016 Nov 27.

PMID:
27899280
29.

Histamine H4 receptor agonist-induced relief from painful peripheral neuropathy is mediated by inhibition of spinal neuroinflammation and oxidative stress.

Sanna MD, Lucarini L, Durante M, Ghelardini C, Masini E, Galeotti N.

Br J Pharmacol. 2017 Jan;174(1):28-40. doi: 10.1111/bph.13644. Epub 2016 Nov 18.

30.

Using Survival Analysis to Identify Risk Factors for Treatment Interruption among New and Retreatment Tuberculosis Patients in Kenya.

Masini EO, Mansour O, Speer CE, Addona V, Hanson CL, Sitienei JK, Kipruto HK, Githiomi MM, Mungai BN.

PLoS One. 2016 Oct 5;11(10):e0164172. doi: 10.1371/journal.pone.0164172. eCollection 2016.

31.

HYDAMTIQ, a selective PARP-1 inhibitor, improves bleomycin-induced lung fibrosis by dampening the TGF-β/SMAD signalling pathway.

Lucarini L, Durante M, Lanzi C, Pini A, Boccalini G, Calosi L, Moroni F, Masini E, Mannaioni G.

J Cell Mol Med. 2017 Feb;21(2):324-335. doi: 10.1111/jcmm.12967. Epub 2016 Oct 4.

32.

Role of histamine H4 receptor ligands in bleomycin-induced pulmonary fibrosis.

Lucarini L, Pini A, Rosa AC, Lanzi C, Durante M, Chazot PL, Krief S, Schreeb A, Stark H, Masini E.

Pharmacol Res. 2016 Sep;111:740-748. doi: 10.1016/j.phrs.2016.07.037. Epub 2016 Jul 27.

PMID:
27475884
33.

Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma.

Vullo D, Durante M, Di Leva FS, Cosconati S, Masini E, Scozzafava A, Novellino E, Supuran CT, Carta F.

J Med Chem. 2016 Jun 23;59(12):5857-67. doi: 10.1021/acs.jmedchem.6b00462. Epub 2016 Jun 13.

PMID:
27253845
34.

Histamine Regulates Actin Cytoskeleton in Human Toll-like Receptor 4-activated Monocyte-derived Dendritic Cells Tuning CD4+ T Lymphocyte Response.

Aldinucci A, Bonechi E, Manuelli C, Nosi D, Masini E, Passani MB, Ballerini C.

J Biol Chem. 2016 Jul 8;291(28):14803-14. doi: 10.1074/jbc.M116.720680. Epub 2016 May 13.

35.

Protection from Cigarette Smoke-Induced Lung Dysfunction and Damage by H2 Relaxin (Serelaxin).

Pini A, Boccalini G, Lucarini L, Catarinicchia S, Guasti D, Masini E, Bani D, Nistri S.

J Pharmacol Exp Ther. 2016 Jun;357(3):451-8. doi: 10.1124/jpet.116.232215. Epub 2016 Apr 5.

PMID:
27048661
36.

Cyclodextrin complexation highly enhances efficacy of arylsulfonylureido benzenesulfonamide carbonic anhydrase inhibitors as a topical antiglaucoma agents.

Bragagni M, Bozdag M, Carta F, Scozzafava A, Lanzi C, Masini E, Mura P, Supuran CT.

Bioorg Med Chem. 2015 Sep 15;23(18):6223-7. doi: 10.1016/j.bmc.2015.07.047. Epub 2015 Jul 29.

PMID:
26319622
37.

Virus-induced gene silencing in Catharanthus roseus by biolistic inoculation of tobacco rattle virus vectors.

Carqueijeiro I, Masini E, Foureau E, Sepúlveda LJ, Marais E, Lanoue A, Besseau S, Papon N, Clastre M, Dugé de Bernonville T, Glévarec G, Atehortùa L, Oudin A, Courdavault V.

Plant Biol (Stuttg). 2015 Nov;17(6):1242-6. doi: 10.1111/plb.12380. Epub 2015 Aug 30.

PMID:
26284695
38.

Histamine H4 receptor activation alleviates neuropathic pain through differential regulation of ERK, JNK, and P38 MAPK phosphorylation.

Sanna MD, Stark H, Lucarini L, Ghelardini C, Masini E, Galeotti N.

Pain. 2015 Dec;156(12):2492-504. doi: 10.1097/j.pain.0000000000000319.

PMID:
26270581
39.

Poly(amidoamine) Dendrimers with Carbonic Anhydrase Inhibitory Activity and Antiglaucoma Action.

Carta F, Osman SM, Vullo D, Gullotto A, Winum JY, AlOthman Z, Masini E, Supuran CT.

J Med Chem. 2015 May 14;58(9):4039-45. doi: 10.1021/acs.jmedchem.5b00383. Epub 2015 Apr 15.

PMID:
25849626
40.

Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action.

Bozdag M, Carta F, Vullo D, Akdemir A, Isik S, Lanzi C, Scozzafava A, Masini E, Supuran CT.

Bioorg Med Chem. 2015 May 15;23(10):2368-76. doi: 10.1016/j.bmc.2015.03.068. Epub 2015 Mar 31.

PMID:
25846066
41.

A class of 4-sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects.

Bozdag M, Pinard M, Carta F, Masini E, Scozzafava A, McKenna R, Supuran CT.

J Med Chem. 2014 Nov 26;57(22):9673-86. doi: 10.1021/jm501497m. Epub 2014 Nov 10.

42.

Structural insights on carbonic anhydrase inhibitory action, isoform selectivity, and potency of sulfonamides and coumarins incorporating arylsulfonylureido groups.

Bozdag M, Ferraroni M, Carta F, Vullo D, Lucarini L, Orlandini E, Rossello A, Nuti E, Scozzafava A, Masini E, Supuran CT.

J Med Chem. 2014 Nov 13;57(21):9152-67. doi: 10.1021/jm501314c. Epub 2014 Oct 17.

PMID:
25310626
43.

Prevention of bleomycin-induced lung inflammation and fibrosis in mice by naproxen and JNJ7777120 treatment.

Rosa AC, Pini A, Lucarini L, Lanzi C, Veglia E, Thurmond RL, Stark H, Masini E.

J Pharmacol Exp Ther. 2014 Nov;351(2):308-16. doi: 10.1124/jpet.114.215152. Epub 2014 Sep 2.

PMID:
25185215
44.

Pharmacokinetics and local safety profile of propranolol eye drops in rabbits.

Padrini L, Isacchi B, Bilia AR, Pini A, Lanzi C, Masini E, Della Bona ML, Calvani AM, Ceccantini R, la Marca G, Filippi L.

Pediatr Res. 2014 Oct;76(4):378-85. doi: 10.1038/pr.2014.108. Epub 2014 Jul 16.

PMID:
25029260
45.

Furazan and furoxan sulfonamides are strong α-carbonic anhydrase inhibitors and potential antiglaucoma agents.

Chegaev K, Lazzarato L, Tamboli Y, Boschi D, Blangetti M, Scozzafava A, Carta F, Masini E, Fruttero R, Supuran CT, Gasco A.

Bioorg Med Chem. 2014 Aug 1;22(15):3913-21. doi: 10.1016/j.bmc.2014.06.016. Epub 2014 Jun 17.

PMID:
25022971
46.

Poly(ADP-ribose) polymerase inhibition with HYDAMTIQ reduces allergen-induced asthma-like reaction, bronchial hyper-reactivity and airway remodelling.

Lucarini L, Pini A, Gerace E, Pellicciari R, Masini E, Moroni F.

J Cell Mol Med. 2014 Mar;18(3):468-79. doi: 10.1111/jcmm.12197. Epub 2014 Jan 20.

47.

Cyclooxygenase-2 and inflammation mediators have a crucial role in reflux-related esophageal histological changes and Barrett's esophagus.

Taddei A, Fabbroni V, Pini A, Lucarini L, Ringressi MN, Fantappiè O, Bani D, Messerini L, Masini E, Bechi P.

Dig Dis Sci. 2014 May;59(5):949-57. doi: 10.1007/s10620-013-2975-4. Epub 2013 Dec 20.

PMID:
24357184
48.

Acute treatment with relaxin protects the kidney against ischaemia/reperfusion injury.

Collino M, Rogazzo M, Pini A, Benetti E, Rosa AC, Chiazza F, Fantozzi R, Bani D, Masini E.

J Cell Mol Med. 2013 Nov;17(11):1494-505. doi: 10.1111/jcmm.12120. Epub 2013 Sep 20.

49.

Outcomes of isoniazid prophylaxis among HIV-infected children attending routine HIV care in Kenya.

Masini EO, Sitienei J, Weyeinga H.

Public Health Action. 2013 Sep 21;3(3):204-8. doi: 10.5588/pha.13.0013.

50.

Effects of a selective histamine H₄R antagonist on inflammation in a model of carrageenan-induced pleurisy in the rat.

Pini A, Somma T, Formicola G, Lucarini L, Bani D, Thurmond R, Masini E.

Curr Pharm Des. 2014;20(9):1338-44.

PMID:
23978101

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