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Items: 1 to 50 of 107

1.

In vivo EPR extracellular pH-metry in tumors using a triphosphonated trityl radical.

Marchand V, Levêque P, Driesschaert B, Marchand-Brynaert J, Gallez B.

Magn Reson Med. 2017 Jun;77(6):2438-2443. doi: 10.1002/mrm.26316. Epub 2016 Jul 1.

PMID:
27364733
2.

Delivery of siRNA targeting tumor metabolism using non-covalent PEGylated chitosan nanoparticles: Identification of an optimal combination of ligand structure, linker and grafting method.

Corbet C, Ragelle H, Pourcelle V, Vanvarenberg K, Marchand-Brynaert J, Préat V, Feron O.

J Control Release. 2016 Feb 10;223:53-63. doi: 10.1016/j.jconrel.2015.12.020. Epub 2015 Dec 14.

PMID:
26699426
3.

Intracellular siRNA delivery dynamics of integrin-targeted, PEGylated chitosan-poly(ethylene imine) hybrid nanoparticles: A mechanistic insight.

Ragelle H, Colombo S, Pourcelle V, Vanvarenberg K, Vandermeulen G, Bouzin C, Marchand-Brynaert J, Feron O, Foged C, Préat V.

J Control Release. 2015 Aug 10;211:1-9. doi: 10.1016/j.jconrel.2015.05.274. Epub 2015 May 16.

PMID:
25989603
4.

Functionalization of the PEG Corona of Nanoparticles by Clip Photochemistry in Water: Application to the Grafting of RGD Ligands on PEGylated USPIO Imaging Agent.

Pourcelle V, Laurent S, Welle A, Vriamont N, Stanicki D, Vander Elst L, Muller RN, Marchand-Brynaert J.

Bioconjug Chem. 2015 May 20;26(5):822-9. doi: 10.1021/acs.bioconjchem.5b00041. Epub 2015 Apr 14.

PMID:
25853330
5.

Self-assembling doxorubicin-tocopherol succinate prodrug as a new drug delivery system: synthesis, characterization, and in vitro and in vivo anticancer activity.

Duhem N, Danhier F, Pourcelle V, Schumers JM, Bertrand O, Leduff CS, Hoeppener S, Schubert US, Gohy JF, Marchand-Brynaert J, Préat V.

Bioconjug Chem. 2014 Jan 15;25(1):72-81. doi: 10.1021/bc400326y. Epub 2013 Dec 23.

PMID:
24328289
6.

(S)-1-(Pent-4'-enoyl)-4-(hydroxymethyl)-azetidin-2-one derivatives as inhibitors of human fatty acid amide hydrolase (hFAAH): synthesis, biological evaluation and molecular modelling.

Caruano J, Feledziak M, Labar G, Michaux C, Perpète EA, Muccioli GG, Robiette R, Marchand-Brynaert J.

J Enzyme Inhib Med Chem. 2014 Oct;29(5):654-62. doi: 10.3109/14756366.2013.837900. Epub 2013 Oct 9.

PMID:
24102523
7.

Macrocycle-embedded β-lactams as novel inhibitors of the Penicillin Binding Protein PBP2a from MRSA.

Dive G, Bouillon C, Sliwa A, Valet B, Verlaine O, Sauvage E, Marchand-Brynaert J.

Eur J Med Chem. 2013 Jun;64:365-76. doi: 10.1016/j.ejmech.2013.03.052. Epub 2013 Apr 15.

PMID:
23648973
8.

Polyethylene terephthalate membrane grafted with peptidomimetics: endothelial cell compatibility and retention under shear stress.

Rémy M, Bareille R, Rerat V, Bourget C, Marchand-Brynaert J, Bordenave L.

J Biomater Sci Polym Ed. 2013;24(3):269-86. doi: 10.1080/09205063.2012.690275. Epub 2012 Aug 13.

PMID:
23565647
9.

Targeted nanoparticles with novel non-peptidic ligands for oral delivery.

des Rieux A, Pourcelle V, Cani PD, Marchand-Brynaert J, Préat V.

Adv Drug Deliv Rev. 2013 Jun 15;65(6):833-44. doi: 10.1016/j.addr.2013.01.002. Epub 2013 Feb 20. Review.

PMID:
23454185
10.

A pyrene- and phosphonate-containing fluorescent probe as guest molecule in a host polymer matrix.

Villemin E, Elias B, Devillers M, Marchand-Brynaert J.

Molecules. 2013 Feb 1;18(2):1897-915. doi: 10.3390/molecules18021897.

11.

An unprecedented reversible mode of action of β-lactams for the inhibition of human fatty acid amide hydrolase (hFAAH).

Feledziak M, Michaux C, Lambert DM, Marchand-Brynaert J.

Eur J Med Chem. 2013 Feb;60:101-11. doi: 10.1016/j.ejmech.2012.11.035. Epub 2012 Nov 29.

PMID:
23287055
12.

Surface modification of polypropylene nonwovens with LDV peptidomimetics and their application in the leukodepletion of blood products.

Gérard E, Bessy E, Hénard G, Verpoort T, Marchand-Brynaert J.

J Biomed Mater Res B Appl Biomater. 2012 Aug;100(6):1513-23. doi: 10.1002/jbm.b.32720. Epub 2012 Jun 12.

PMID:
22689380
13.

Vibrational circular dichroism versus optical rotation dispersion and electronic circular dichroism for diastereomers: the stereochemistry of 3-(1'-hydroxyethyl)-1-(3'-phenylpropanoyl)-azetidin-2-one.

Gussem ED, Bultinck P, Feledziak M, Marchand-Brynaert J, Stevens CV, Herrebout W.

Phys Chem Chem Phys. 2012 Jun 28;14(24):8562-71. doi: 10.1039/c2cp40617a. Epub 2012 May 17.

PMID:
22596178
14.

Degradation of bare and silanized silicon wafer surfaces by constituents of biological fluids.

Dekeyser CM, Buron CC, Derclaye SR, Jonas AM, Marchand-Brynaert J, Rouxhet PG.

J Colloid Interface Sci. 2012 Jul 15;378(1):77-82. doi: 10.1016/j.jcis.2012.04.022. Epub 2012 Apr 19.

PMID:
22560491
15.

Characterization of an endophytic whorl-forming Streptomyces from Catharanthus roseus stems producing polyene macrolide antibiotic.

Rakotoniriana EF, Chataigné G, Raoelison G, Rabemanantsoa C, Munaut F, El Jaziri M, Urveg-Ratsimamanga S, Marchand-Brynaert J, Corbisier AM, Declerck S, Quetin-Leclercq J.

Can J Microbiol. 2012 May;58(5):617-27. doi: 10.1139/w2012-034. Epub 2012 Apr 23.

PMID:
22524528
16.

Targeting of tumor endothelium by RGD-grafted PLGA-nanoparticles.

Danhier F, Pourcelle V, Marchand-Brynaert J, Jérôme C, Feron O, Préat V.

Methods Enzymol. 2012;508:157-75. doi: 10.1016/B978-0-12-391860-4.00008-2.

PMID:
22449925
17.

Synthesis of poly(lactide-co-glycolide-co-ε-caprolactone)-graft-mannosylated poly(ethylene oxide) copolymers by combination of "clip" and "click" chemistries.

Freichels H, Pourcelle V, Auzély-Velty R, Marchand-Brynaert J, Jérôme C.

Biomacromolecules. 2012 Mar 12;13(3):760-8. doi: 10.1021/bm201690w. Epub 2012 Feb 27.

PMID:
22329463
18.

A phosphonated triarylmethyl radical as a probe for measurement of pH by EPR.

Driesschaert B, Marchand V, Levêque P, Gallez B, Marchand-Brynaert J.

Chem Commun (Camb). 2012 Apr 28;48(34):4049-51. doi: 10.1039/c2cc00025c. Epub 2012 Feb 8.

PMID:
22314917
19.

Inhibitors of the endocannabinoid-degrading enzymes, or how to increase endocannabinoid's activity by preventing their hydrolysis.

Feledziak M, Lambert DM, Marchand-Brynaert J, Muccioli GG.

Recent Pat CNS Drug Discov. 2012 Apr 1;7(1):49-70. Review.

PMID:
22280341
20.

Non-symmetrically substituted phenoxazinones from laccase-mediated oxidative cross-coupling of aminophenols: an experimental and theoretical insight.

Bruyneel F, Dive G, Marchand-Brynaert J.

Org Biomol Chem. 2012 Mar 7;10(9):1834-46. doi: 10.1039/c1ob05795b. Epub 2012 Jan 18.

PMID:
22257991
21.

12- to 22-membered bridged β-lactams as potential penicillin-binding protein inhibitors.

Sliwa A, Dive G, Marchand-Brynaert J.

Chem Asian J. 2012 Feb 6;7(2):425-34. doi: 10.1002/asia.201100732. Epub 2011 Dec 8.

22.

LDV peptidomimetics equipped with biotinylated spacer-arms: synthesis and biological evaluation on CCRF-CEM cell line.

Gérard E, Meulle A, Feron O, Marchand-Brynaert J.

Bioorg Med Chem Lett. 2012 Jan 1;22(1):586-90. doi: 10.1016/j.bmcl.2011.10.078. Epub 2011 Oct 31.

PMID:
22101134
23.

DOSY-NMR analysis of ring-closing metathesis (RCM) products from β-lactam precursors.

Sliwa A, Marchand-Brynaert J, Luhmer M.

Magn Reson Chem. 2011 Dec;49(12):812-5. doi: 10.1002/mrc.2808. Epub 2011 Nov 17.

PMID:
22095794
24.

Benzisothiazolinone as a useful template for the design of new monoacylglycerol lipase inhibitors: investigation of the target residues and comparison with octhilinone.

Matuszak N, Es Saadi B, Labar G, Marchand-Brynaert J, Lambert DM.

Bioorg Med Chem Lett. 2011 Dec 15;21(24):7321-4. doi: 10.1016/j.bmcl.2011.10.026. Epub 2011 Oct 18.

PMID:
22056744
25.

Spin transition sensors based on β-amino-acid 1,2,4-triazole derivative.

Dîrtu MM, Schmit F, Naik AD, Rotaru A, Marchand-Brynaert J, Garcia Y.

Int J Mol Sci. 2011;12(8):5339-51. doi: 10.3390/ijms12085339. Epub 2011 Aug 18.

26.

SAR and LC/MS studies of β-lactamic inhibitors of human fatty acid amide hydrolase (hFAAH): evidence of a nonhydrolytic process.

Feledziak M, Muccioli GG, Lambert DM, Marchand-Brynaert J.

J Med Chem. 2011 Oct 13;54(19):6812-23. doi: 10.1021/jm200723m. Epub 2011 Sep 20.

PMID:
21899370
27.

Role of oxidative stress in lysosomal membrane permeabilization and apoptosis induced by gentamicin, an aminoglycoside antibiotic.

Denamur S, Tyteca D, Marchand-Brynaert J, Van Bambeke F, Tulkens PM, Courtoy PJ, Mingeot-Leclercq MP.

Free Radic Biol Med. 2011 Nov 1;51(9):1656-65. doi: 10.1016/j.freeradbiomed.2011.07.015. Epub 2011 Jul 23.

PMID:
21835240
28.

Structure-activity relationships of various amino-hydroxy-benzenesulfonic acids and sulfonamides as tyrosinase substrates.

Rescigno A, Bruyneel F, Padiglia A, Sollai F, Salis A, Marchand-Brynaert J, Sanjust E.

Biochim Biophys Acta. 2011 Aug;1810(8):799-807. doi: 10.1016/j.bbagen.2011.05.002. Epub 2011 May 13.

PMID:
21605629
29.

"Clip" and "click" chemistries combination: toward easy PEGylation of degradable aliphatic polyesters.

Freichels H, Pourcelle V, Le Duff CS, Marchand-Brynaert J, Jérôme C.

Macromol Rapid Commun. 2011 Apr 4;32(7):616-21. doi: 10.1002/marc.201000803. Epub 2011 Mar 7.

PMID:
21438062
30.

Chiral properties of tetrathiatriarylmethyl spin probes.

Driesschaert B, Robiette R, Lucaccioni F, Gallez B, Marchand-Brynaert J.

Chem Commun (Camb). 2011 Apr 28;47(16):4793-5. doi: 10.1039/c1cc10988j. Epub 2011 Mar 15.

PMID:
21409216
31.

Combined experimental and theoretical study on the Raman and Raman optical activity signatures of pentamethylundecane diastereoisomers.

Drooghaag X, Marchand-Brynaert J, Champagne B, Liégeois V.

J Phys Chem B. 2010 Sep 16;114(36):11753-60. doi: 10.1021/jp105028q.

PMID:
20731402
32.

[4 + 2] Cycloadditions of 1-phosphono-1,3-butadienes with nitroso heterodienophiles: a versatile synthetic route for polyfunctionalized aminophosphonic derivatives.

Monbaliu JC, Tinant B, Marchand-Brynaert J.

J Org Chem. 2010 Aug 20;75(16):5478-86. doi: 10.1021/jo100230r.

PMID:
20704424
33.

Calcium and zinc complexes of pyrroglutamate analogs detected by electrospray ionization mass spectrometry.

Beck J, Maton L, Habib Jiwan JL, Marchand-Brynaert J.

Amino Acids. 2011 Feb;40(2):679-87. doi: 10.1007/s00726-010-0697-x. Epub 2010 Jul 27.

PMID:
20661759
34.

Chemistry around imidazopyrazine and ibuprofen: discovery of novel fatty acid amide hydrolase (FAAH) inhibitors.

De Wael F, Muccioli GG, Lambert DM, Sergent T, Schneider YJ, Rees JF, Marchand-Brynaert J.

Eur J Med Chem. 2010 Sep;45(9):3564-74. doi: 10.1016/j.ejmech.2010.04.040. Epub 2010 May 11.

PMID:
20570023
35.

Live-cell imaging with water-soluble aminophenoxazinone dyes synthesised through laccase biocatalysis.

Bruyneel F, D'Auria L, Payen O, Courtoy PJ, Marchand-Brynaert J.

Chembiochem. 2010 Jul 5;11(10):1451-7. doi: 10.1002/cbic.201000145.

PMID:
20533495
36.

Stability of meropenem and doripenem solutions for administration by continuous infusion.

Berthoin K, Le Duff CS, Marchand-Brynaert J, Carryn S, Tulkens PM.

J Antimicrob Chemother. 2010 May;65(5):1073-5. doi: 10.1093/jac/dkq044. Epub 2010 Feb 21. No abstract available.

PMID:
20176578
37.

Ultrasmall particle of iron oxide--RGD peptidomimetic conjugate: synthesis and characterisation.

Rerat V, Laurent S, Burtéa C, Driesschaert B, Pourcelle V, Vander Elst L, Muller RN, Marchand-Brynaert J.

Bioorg Med Chem Lett. 2010 Mar 15;20(6):1861-5. doi: 10.1016/j.bmcl.2010.01.150. Epub 2010 Feb 4.

PMID:
20172716
38.

beta-Lactams derived from a carbapenem chiron are selective inhibitors of human fatty acid amide hydrolase versus human monoacylglycerol lipase.

Feledziak M, Michaux C, Urbach A, Labar G, Muccioli GG, Lambert DM, Marchand-Brynaert J.

J Med Chem. 2009 Nov 26;52(22):7054-68. doi: 10.1021/jm9008532.

PMID:
19877691
39.

alphavbeta3 Integrin-targeting Arg-Gly-Asp (RGD) peptidomimetics containing oligoethylene glycol (OEG) spacers.

Rerat V, Dive G, Cordi AA, Tucker GC, Bareille R, Amédée J, Bordenave L, Marchand-Brynaert J.

J Med Chem. 2009 Nov 26;52(22):7029-43. doi: 10.1021/jm901133z.

40.

Targeting of tumor endothelium by RGD-grafted PLGA-nanoparticles loaded with paclitaxel.

Danhier F, Vroman B, Lecouturier N, Crokart N, Pourcelle V, Freichels H, Jérôme C, Marchand-Brynaert J, Feron O, Préat V.

J Control Release. 2009 Dec 3;140(2):166-73. doi: 10.1016/j.jconrel.2009.08.011. Epub 2009 Aug 20.

PMID:
19699245
41.

Laccase-mediated synthesis of novel substituted phenoxazine chromophores featuring tuneable water solubility.

Bruyneel F, Payen O, Rescigno A, Tinant B, Marchand-Brynaert J.

Chemistry. 2009 Aug 17;15(33):8283-95. doi: 10.1002/chem.200900681.

PMID:
19623587
42.

In vitro and in vivo studies of 6,8-(diaryl)imidazo[1,2-a]pyrazin-3(7H)-ones as new antioxidants.

De Wael F, Jeanjot P, Moens C, Verbeuren T, Cordi A, Bouskela E, Rees JF, Marchand-Brynaert J.

Bioorg Med Chem. 2009 Jul 1;17(13):4336-44. doi: 10.1016/j.bmc.2009.05.025. Epub 2009 May 15.

PMID:
19477651
43.

Discovery of novel lipophilic inhibitors of OXA-10 enzyme (class D beta-lactamase) by screening amino analogs and homologs of citrate and isocitrate.

Beck J, Vercheval L, Bebrone C, Herteg-Fernea A, Lassaux P, Marchand-Brynaert J.

Bioorg Med Chem Lett. 2009 Jul 1;19(13):3593-7. doi: 10.1016/j.bmcl.2009.04.149. Epub 2009 May 6.

44.

Targeting nanoparticles to M cells with non-peptidic ligands for oral vaccination.

Fievez V, Plapied L, des Rieux A, Pourcelle V, Freichels H, Wascotte V, Vanderhaeghen ML, Jerôme C, Vanderplasschen A, Marchand-Brynaert J, Schneider YJ, Préat V.

Eur J Pharm Biopharm. 2009 Sep;73(1):16-24. doi: 10.1016/j.ejpb.2009.04.009. Epub 2009 May 4.

45.

Light induced functionalization of PCL-PEG block copolymers for the covalent immobilization of biomolecules.

Pourcelle V, Freichels H, Stoffelbach F, Auzély-Velty R, Jérôme C, Marchand-Brynaert J.

Biomacromolecules. 2009 Apr 13;10(4):966-74. doi: 10.1021/bm900027r.

PMID:
19226175
46.

Surface functionalization of germanium ATR devices for use in FTIR-biosensors.

Devouge S, Conti J, Goldsztein A, Gosselin E, Brans A, Voué M, De Coninck J, Homblé F, Goormaghtigh E, Marchand-Brynaert J.

J Colloid Interface Sci. 2009 Apr 15;332(2):408-15. doi: 10.1016/j.jcis.2008.12.045. Epub 2008 Dec 24.

47.

Nano-emulsions of fluorinated trityl radicals as sensors for EPR oximetry.

Charlier N, Driesschaert B, Wauthoz N, Beghein N, Préat V, Amighi K, Marchand-Brynaert J, Gallez B.

J Magn Reson. 2009 Apr;197(2):176-80. doi: 10.1016/j.jmr.2008.12.013. Epub 2008 Dec 24.

PMID:
19128993
48.

Large ring 1,3-bridged 2-azetidinones: experimental and theoretical studies.

Urbach A, Dive G, Tinant B, Duval V, Marchand-Brynaert J.

Eur J Med Chem. 2009 May;44(5):2071-80. doi: 10.1016/j.ejmech.2008.10.016. Epub 2008 Oct 26.

49.

Ligand-receptor interactions in complex media: a new type of biosensors for the detection of coagulation factor VIII.

Goldzstein A, Aamouche A, Homblé F, Voué M, Conti J, De Coninck J, Devouge S, Marchand-Brynaert J, Goormaghtigh E.

Biosens Bioelectron. 2009 Mar 15;24(7):1831-6. doi: 10.1016/j.bios.2008.09.013. Epub 2008 Sep 24.

PMID:
18977650
50.

Paclitaxel-loaded PEGylated PLGA-based nanoparticles: in vitro and in vivo evaluation.

Danhier F, Lecouturier N, Vroman B, Jérôme C, Marchand-Brynaert J, Feron O, Préat V.

J Control Release. 2009 Jan 5;133(1):11-7. doi: 10.1016/j.jconrel.2008.09.086. Epub 2008 Oct 9.

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