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Items: 17


Enantiomeric characterization and structure elucidation of LH601A using vibrational circular dichroism spectroscopy.

Shen J, Magesh S, Chen L, Hu L, He Y.

Spectrochim Acta A Mol Biomol Spectrosc. 2018 Mar 5;192:312-317. doi: 10.1016/j.saa.2017.11.033. Epub 2017 Nov 21.


The NEU1-selective sialidase inhibitor, C9-butyl-amide-DANA, blocks sialidase activity and NEU1-mediated bioactivities in human lung in vitro and murine lung in vivo.

Hyun SW, Liu A, Liu Z, Cross AS, Verceles AC, Magesh S, Kommagalla Y, Kona C, Ando H, Luzina IG, Atamas SP, Piepenbrink KH, Sundberg EJ, Guang W, Ishida H, Lillehoj EP, Goldblum SE.

Glycobiology. 2016 Aug;26(8):834-49. doi: 10.1093/glycob/cww060. Epub 2016 May 25.


A Novel Potent and Highly Specific Inhibitor against Influenza Viral N1-N9 Neuraminidases: Insight into Neuraminidase-Inhibitor Interactions.

Sriwilaijaroen N, Magesh S, Imamura A, Ando H, Ishida H, Sakai M, Ishitsubo E, Hori T, Moriya S, Ishikawa T, Kuwata K, Odagiri T, Tashiro M, Hiramatsu H, Tsukamoto K, Miyagi T, Tokiwa H, Kiso M, Suzuki Y.

J Med Chem. 2016 May 26;59(10):4563-77. doi: 10.1021/acs.jmedchem.5b01863. Epub 2016 May 4.


Insilico docking study of compounds elucidated from helicteres isora fruits with ampkinase- insulin receptor.

Vennila S, Bupesh G, Saravanamurali K, SenthilKumar V, SenthilRaja R, Saran N, Magesh S.

Bioinformation. 2014 May 20;10(5):263-6. doi: 10.6026/97320630010263. eCollection 2014.


Design and synthesis of novel iminothiazinylbutadienols and divinylpyrimidinethiones as ARE inducers.

Chen L, Magesh S, Wang H, Yang CS, Kong AN, Hu L.

Bioorg Med Chem Lett. 2014 Feb 1;24(3):940-3. doi: 10.1016/j.bmcl.2013.12.072. Epub 2013 Dec 24.


In vitro and in vivo anti-inflammatory effects of a novel 4,6-bis ((E)-4-hydroxy-3-methoxystyryl)-1-phenethylpyrimidine-2(1H)-thione.

Lee JH, Lee KR, Su ZY, Boyanapalli SS, Barman DN, Huang MT, Chen L, Magesh S, Hu L, Kong AN.

Chem Res Toxicol. 2014 Jan 21;27(1):34-41. doi: 10.1021/tx400315u. Epub 2013 Dec 17.


The identification and characterization of non-reactive inhibitor of Keap1-Nrf2 interaction through HTS using a fluorescence polarization assay.

Wang L, Lewis T, Zhang YL, Khodier C, Magesh S, Chen L, Inoyama D, Chen Y, Zhen J, Hu L, Beamer LJ, Faloon PW, Dandapani S, Perez JR, Munoz B, Palmer M, Schreiber S.

Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010-.
2012 Dec 17 [updated 2013 Sep 16].


Discovery of a small-molecule inhibitor and cellular probe of Keap1-Nrf2 protein-protein interaction.

Hu L, Magesh S, Chen L, Wang L, Lewis TA, Chen Y, Khodier C, Inoyama D, Beamer LJ, Emge TJ, Shen J, Kerrigan JE, Kong AN, Dandapani S, Palmer M, Schreiber SL, Munoz B.

Bioorg Med Chem Lett. 2013 May 15;23(10):3039-43. doi: 10.1016/j.bmcl.2013.03.013. Epub 2013 Mar 14.


Small molecule modulators of Keap1-Nrf2-ARE pathway as potential preventive and therapeutic agents.

Magesh S, Chen Y, Hu L.

Med Res Rev. 2012 Jul;32(4):687-726. doi: 10.1002/med.21257. Epub 2012 May 1. Review.


High-affinity ligands of Siglec receptors and their therapeutic potentials.

Magesh S, Ando H, Tsubata T, Ishida H, Kiso M.

Curr Med Chem. 2011;18(23):3537-50. Review.


Evaluation of a Set of C9 N-acyl Neu5Ac2en Mimetics as Viral Sialidase Selective Inhibitors.

Magesh S, Sriwilaijaroen N, Moriya S, Ando H, Miyagi T, Suzuki Y, Ishida H, Kiso M.

Int J Med Chem. 2011;2011:539245. doi: 10.1155/2011/539245. Epub 2010 Dec 8.


Human sialidase inhibitors: design, synthesis, and biological evaluation of 4-acetamido-5-acylamido-2-fluoro benzoic acids.

Magesh S, Savita V, Moriya S, Suzuki T, Miyagi T, Ishida H, Kiso M.

Bioorg Med Chem. 2009 Jul 1;17(13):4595-603. doi: 10.1016/j.bmc.2009.04.065. Epub 2009 May 4.


Design, synthesis, and biological evaluation of human sialidase inhibitors. Part 1: selective inhibitors of lysosomal sialidase (NEU1).

Magesh S, Moriya S, Suzuki T, Miyagi T, Ishida H, Kiso M.

Bioorg Med Chem Lett. 2008 Jan 15;18(2):532-7. Epub 2007 Nov 28.


Impurity profile study of zaleplon.

Bharathi Ch, Prabahar KJ, Prasad ChS, Kumar MS, Magesh S, Handa VK, Dandala R, Naidu A.

J Pharm Biomed Anal. 2007 May 9;44(1):101-9. Epub 2007 Feb 6.


Acute toxicity of endosulfan to the milkfish, Chanos chanos, of the Southeast Coast of India.

Magesh S, Kumaraguru AK.

Bull Environ Contam Toxicol. 2006 Apr;76(4):622-8. No abstract available.


Homology modeling of human sialidase enzymes NEU1, NEU3 and NEU4 based on the crystal structure of NEU2: hints for the design of selective NEU3 inhibitors.

Magesh S, Suzuki T, Miyagi T, Ishida H, Kiso M.

J Mol Graph Model. 2006 Oct;25(2):196-207. Epub 2006 Jan 19.


An outbreak of food poisoning in Tamil Nadu associated with Yersinia enterocolitica.

Abraham M, Pai M, Kang G, Asokan GV, Magesh SR, Bhattacharji S, Ramakrishna BS.

Indian J Med Res. 1997 Nov;106:465-8.


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