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Items: 13

1.

Novel BQCA and TBPB derived M1 Receptor Hybrid-Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism.

Schramm S, Agnetta L, Bermudez M, Gerwe H, Littmann T, Irmen M, Holze J, Wolber G, Tränkle C, Decker M.

ChemMedChem. 2019 Jun 5. doi: 10.1002/cmdc.201900283. [Epub ahead of print]

PMID:
31166078
2.

Split luciferase-based assay for simultaneous analyses of the ligand concentration- and time-dependent recruitment of β-arrestin2.

Littmann T, Buschauer A, Bernhardt G.

Anal Biochem. 2019 May 15;573:8-16. doi: 10.1016/j.ab.2019.02.023. Epub 2019 Mar 8.

PMID:
30853375
3.

Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties.

Agnetta L, Bermudez M, Riefolo F, Matera C, Claro E, Messerer R, Littmann T, Wolber G, Holzgrabe U, Decker M.

J Med Chem. 2019 Mar 28;62(6):3009-3020. doi: 10.1021/acs.jmedchem.8b01822. Epub 2019 Mar 19.

PMID:
30827105
4.

A split luciferase-based probe for quantitative proximal determination of Gαq signalling in live cells.

Littmann T, Ozawa T, Hoffmann C, Buschauer A, Bernhardt G.

Sci Rep. 2018 Nov 21;8(1):17179. doi: 10.1038/s41598-018-35615-w.

5.

In Search of NPY Y4R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or d-Amino Acids into Oligopeptides Derived from the C-Termini of the Endogenous Agonists.

Kuhn KK, Littmann T, Dukorn S, Tanaka M, Keller M, Ozawa T, Bernhardt G, Buschauer A.

ACS Omega. 2017 Jul 31;2(7):3616-3631. doi: 10.1021/acsomega.7b00451. Epub 2017 Jul 14.

6.

Structural basis of ligand binding modes at the neuropeptide Y Y1 receptor.

Yang Z, Han S, Keller M, Kaiser A, Bender BJ, Bosse M, Burkert K, Kögler LM, Wifling D, Bernhardt G, Plank N, Littmann T, Schmidt P, Yi C, Li B, Ye S, Zhang R, Xu B, Larhammar D, Stevens RC, Huster D, Meiler J, Zhao Q, Beck-Sickinger AG, Buschauer A, Wu B.

Nature. 2018 Apr;556(7702):520-524. doi: 10.1038/s41586-018-0046-x. Epub 2018 Apr 18.

7.

Establishing a Split Luciferase Assay for Proteinkinase G (PKG) Interaction Studies.

Schramm A, Mueller-Thuemen P, Littmann T, Harloff M, Ozawa T, Schlossmann J.

Int J Mol Sci. 2018 Apr 12;19(4). pii: E1180. doi: 10.3390/ijms19041180.

8.

Fluorescence- and Radiolabeling of [Lys4,Nle17,30]hPP Yields Molecular Tools for the NPY Y4 Receptor.

Dukorn S, Littmann T, Keller M, Kuhn K, Cabrele C, Baumeister P, Bernhardt G, Buschauer A.

Bioconjug Chem. 2017 Apr 19;28(4):1291-1304. doi: 10.1021/acs.bioconjchem.7b00103. Epub 2017 Apr 5.

PMID:
28345900
9.

Label-free versus conventional cellular assays: Functional investigations on the human histamine H1 receptor.

Lieb S, Littmann T, Plank N, Felixberger J, Tanaka M, Schäfer T, Krief S, Elz S, Friedland K, Bernhardt G, Wegener J, Ozawa T, Buschauer A.

Pharmacol Res. 2016 Dec;114:13-26. doi: 10.1016/j.phrs.2016.10.010. Epub 2016 Oct 15.

PMID:
27751876
10.

Recruitment of β-arrestin 1 and 2 to the β2-adrenoceptor: analysis of 65 ligands.

Littmann T, Göttle M, Reinartz MT, Kälble S, Wainer IW, Ozawa T, Seifert R.

J Pharmacol Exp Ther. 2015 Nov;355(2):183-90. doi: 10.1124/jpet.115.227959. Epub 2015 Aug 25.

11.

Structure-bias relationships for fenoterol stereoisomers in six molecular and cellular assays at the β2-adrenoceptor.

Reinartz MT, Kälble S, Littmann T, Ozawa T, Dove S, Kaever V, Wainer IW, Seifert R.

Naunyn Schmiedebergs Arch Pharmacol. 2015 Jan;388(1):51-65. doi: 10.1007/s00210-014-1054-5. Epub 2014 Oct 24.

PMID:
25342094
12.

The P2Y(2) nucleotide receptor mediates tissue factor expression in human coronary artery endothelial cells.

Ding L, Ma W, Littmann T, Camp R, Shen J.

J Biol Chem. 2011 Jul 29;286(30):27027-38. doi: 10.1074/jbc.M111.235176. Epub 2011 Jun 7.

13.

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