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Items: 10

1.

Novel SAR for quinazoline inhibitors of EHMT1 and EHMT2.

Leenders R, Zijlmans R, van Bree B, van de Sande M, Trivarelli F, Damen E, Wegert A, Müller D, Ehlert JE, Feger D, Heidemann-Dinger C, Kubbutat M, Schächtele C, Lenstra DC, Mecinović J, Müller G.

Bioorg Med Chem Lett. 2019 Sep 1;29(17):2516-2524. doi: 10.1016/j.bmcl.2019.06.012. Epub 2019 Jun 14.

PMID:
31350126
2.

Lysine Ethylation by Histone Lysine Methyltransferases.

Al Temimi AHK, Martin M, Meng Q, Lenstra DC, Qian P, Guo H, Weinhold E, Mecinovic J.

Chembiochem. 2019 Jul 9. doi: 10.1002/cbic.201900359. [Epub ahead of print]

PMID:
31287209
3.

Importance of the main chain of lysine for histone lysine methyltransferase catalysis.

Al Temimi AHK, Teeuwen RS, Tran V, Altunc AJ, Lenstra DC, Ren W, Qian P, Guo H, Mecinović J.

Org Biomol Chem. 2019 Jun 12;17(23):5693-5697. doi: 10.1039/c9ob01038f.

PMID:
31134245
4.

Catalytic Staudinger Reduction at Room Temperature.

Lenstra DC, Wolf JJ, Mecinović J.

J Org Chem. 2019 May 17;84(10):6536-6545. doi: 10.1021/acs.joc.9b00831. Epub 2019 May 9.

PMID:
31050295
5.

Investigating the active site of human trimethyllysine hydroxylase.

Wang Y, Reddy YV, Al Temimi AHK, Venselaar H, Nelissen FHT, Lenstra DC, Mecinović J.

Biochem J. 2019 Apr 10;476(7):1109-1119. doi: 10.1042/BCJ20180857.

PMID:
30898847
6.

Structure-Activity Relationship Studies on (R)-PFI-2 Analogues as Inhibitors of Histone Lysine Methyltransferase SETD7.

Lenstra DC, Damen E, Leenders RGG, Blaauw RH, Rutjes FPJT, Wegert A, Mecinović J.

ChemMedChem. 2018 Jul 18;13(14):1405-1413. doi: 10.1002/cmdc.201800242. Epub 2018 Jun 25.

PMID:
29869845
7.

Inhibition of histone lysine methyltransferases G9a and GLP by ejection of structural Zn(II).

Lenstra DC, Al Temimi AHK, Mecinović J.

Bioorg Med Chem Lett. 2018 Apr 15;28(7):1234-1238. doi: 10.1016/j.bmcl.2018.02.043. Epub 2018 Feb 24.

8.

Poly(methylhydrosiloxane) as a green reducing agent in organophosphorus-catalysed amide bond formation.

Hamstra DFJ, Lenstra DC, Koenders TJ, Rutjes FPJT, Mecinović J.

Org Biomol Chem. 2017 Aug 2;15(30):6426-6432. doi: 10.1039/c7ob01510k.

PMID:
28737181
9.

One-Pot Sulfoxide Synthesis Exploiting a Sulfinyl-Dication Equivalent Generated from a DABSO/Trimethylsilyl Chloride Sequence.

Lenstra DC, Vedovato V, Ferrer Flegeau E, Maydom J, Willis MC.

Org Lett. 2016 May 6;18(9):2086-9. doi: 10.1021/acs.orglett.6b00712. Epub 2016 Apr 15.

10.

Triphenylphosphine-catalysed amide bond formation between carboxylic acids and amines.

Lenstra DC, Rutjes FP, Mecinović J.

Chem Commun (Camb). 2014 Jun 1;50(43):5763-6. doi: 10.1039/c4cc01861c. Epub 2014 Apr 22.

PMID:
24752820

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