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Items: 9


A NanoBRET-based binding assay for Smoothened allows real time analysis of ligand binding and distinction of two binding sites for BODIPY-cyclopamine.

Kozielewicz P, Bowin CF, Turku A, Schulte G.

Mol Pharmacol. 2019 Nov 9. pii: mol.119.118158. doi: 10.1124/mol.119.118158. [Epub ahead of print]


Molecular Pharmacology of Class F Receptor Activation.

Kozielewicz P, Turku A, Schulte G.

Mol Pharmacol. 2019 Oct 7. pii: mol.119.117986. doi: 10.1124/mol.119.117986. [Epub ahead of print]


Overexpression of Orphan Receptor GPR61 Increases cAMP Levels upon Forskolin Stimulation in HEK293 Cells: in vitro and in silico Validation of 5-(Nonyloxy)Tryptamine as a Low-Affinity Inverse Agonist.

Kozielewicz P, Grafton G, Sajkowska-Kozielewicz JJ, Barnes NM.

Pharmacology. 2019 Jul 26:1-6. doi: 10.1159/000501926. [Epub ahead of print]


Comment on: Triazoles bind the C-terminal domain of SMO: Illustration by docking and molecular dynamics simulations the binding between SMO and triazoles.

Kozielewicz P.

Life Sci. 2019 May 15;225:132. doi: 10.1016/j.lfs.2019.03.075. Epub 2019 Apr 6. No abstract available.


Structural insight into Class F receptors - What have we learnt regarding agonist-induced activation?

Schulte G, Kozielewicz P.

Basic Clin Pharmacol Toxicol. 2019 Mar 29. doi: 10.1111/bcpt.13235. [Epub ahead of print]


A conserved molecular switch in Class F receptors regulates receptor activation and pathway selection.

Wright SC, Kozielewicz P, Kowalski-Jahn M, Petersen J, Bowin CF, Slodkowicz G, Marti-Solano M, Rodríguez D, Hot B, Okashah N, Strakova K, Valnohova J, Babu MM, Lambert NA, Carlsson J, Schulte G.

Nat Commun. 2019 Feb 8;10(1):667. doi: 10.1038/s41467-019-08630-2.


N-glycosylation and expression in human tissues of the orphan GPR61 receptor.

Kozielewicz P, Alomar H, Yusof S, Grafton G, Cooper AJ, Curnow SJ, Ironside JW, Pall H, Barnes NM.

FEBS Open Bio. 2017 Nov 20;7(12):1982-1993. doi: 10.1002/2211-5463.12339. eCollection 2017 Dec.


Antioxidant, Cytotoxic, and Antiproliferative Activities and Total Polyphenol Contents of the Extracts of Geissospermum reticulatum Bark.

Sajkowska-Kozielewicz JJ, Kozielewicz P, Barnes NM, Wawer I, Paradowska K.

Oxid Med Cell Longev. 2016;2016:2573580. Epub 2016 Jun 29.


Novel vitamin D analogues; cytotoxic and anti-proliferative activity against a diffuse large B-cell lymphoma cell line and B-cells from healthy donors.

Kozielewicz P, Grafton G, Kutner A, Curnow SJ, Gordon J, Barnes NM.

J Steroid Biochem Mol Biol. 2016 Nov;164:98-105. doi: 10.1016/j.jsbmb.2015.10.015. Epub 2015 Oct 17.


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