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Items: 1 to 50 of 97

1.

Acute salt loading and cardiotonic steroids in resistant hypertension.

Emelyanov IV, Konradi AO, Lakatta EG, Fedorova OV, Bagrov AY.

Curr Top Membr. 2019;83:1-13. doi: 10.1016/bs.ctm.2019.01.005. Epub 2019 Feb 18.

PMID:
31196601
2.

May Measurement Month 2017 in Russia: hypertension treatment and control-Europe.

Rotar O, Konradi A, Tanicheva A, Nakonechnikov S, Blinova N, Beaney T, Xia X, Poulter NR, Chazova I, Shlyakhto E.

Eur Heart J Suppl. 2019 Apr;21(Suppl D):D101-D103. doi: 10.1093/eurheartj/suz068. Epub 2019 Apr 24.

3.

Vascular Age Concept: Which Approach Is Preferable in Clinical Practice?

Rotar OP, Alieva AS, Boiarinova MA, Tolkunova KM, Konradi AO.

Kardiologiia. 2019 Mar 7;59(2):45-53. doi: 10.18087/cardio.2019.2.10229. Russian.

PMID:
30853021
4.

Porphyromonas gingivalis in Alzheimer's disease brains: Evidence for disease causation and treatment with small-molecule inhibitors.

Dominy SS, Lynch C, Ermini F, Benedyk M, Marczyk A, Konradi A, Nguyen M, Haditsch U, Raha D, Griffin C, Holsinger LJ, Arastu-Kapur S, Kaba S, Lee A, Ryder MI, Potempa B, Mydel P, Hellvard A, Adamowicz K, Hasturk H, Walker GD, Reynolds EC, Faull RLM, Curtis MA, Dragunow M, Potempa J.

Sci Adv. 2019 Jan 23;5(1):eaau3333. doi: 10.1126/sciadv.aau3333. eCollection 2019 Jan.

5.

The prevalence of abdominal obesity and the association with socioeconomic status in Regions of the Russian Federation, the results of the epidemiological study - ESSE-RF.

Zhernakova YV, Zheleznova EA, Chazova IE, Oshchepkova EV, Dolgusheva YA, Yarovaya EB, Blinova NV, Orlovsky AA, Konosova ID, Shalnova SA, Rotar' OP, Konradi AO, Shlyakhto EV, Boytsov SA.

Ter Arkh. 2018 Nov 22;90(10):14-22. doi: 10.26442/terarkh2018901014-22.

PMID:
30701790
6.

MASked-unconTrolled hypERtension management based on office BP or on ambulatory blood pressure measurement (MASTER) Study: a randomised controlled trial protocol.

Parati G, Agabiti-Rosei E, Bakris GL, Bilo G, Branzi G, Cecchi F, Chrostowska M, De la Sierra A, Domenech M, Dorobantu M, Faria T, Huo Y, Jelaković B, Kahan T, Konradi A, Laurent S, Li N, Madan K, Mancia G, McManus RJ, Modesti PA, Ochoa JE, Octavio JA, Omboni S, Palatini P, Park JB, Pellegrini D, Perl S, Podoleanu C, Pucci G, Redon J, Renna N, Rhee MY, Rodilla Sala E, Sanchez R, Schmieder R, Soranna D, Stergiou G, Stojanovic M, Tsioufis K, Valsecchi MG, Veglio F, Waisman GD, Wang JG, Wijnmaalen P, Zambon A, Zanchetti A, Zhang Y.

BMJ Open. 2018 Dec 19;8(12):e021038. doi: 10.1136/bmjopen-2017-021038.

7.

Large artery stiffness according to different assessment methods in adult population of St.Petersburg.

Alieva AS, Rotar OP, Orlov AV, Boyarinova MA, Moguchaya EV, Rogoza AN, Konradi AO, Shlyakhto EV.

Atheroscler Suppl. 2018 Sep;35:e1-e5. doi: 10.1016/j.atherosclerosissup.2018.08.001. Epub 2018 Aug 24.

PMID:
30197020
8.

Epidemiology of cardiovascular risk factors in two population-based studies.

Olmastroni E, Shlyakhto EV, Konradi AO, Rotar OP, Alieva AS, Boyarinova MA, Baragetti A, Grigore L, Pellegatta F, Tragni E, Catapano AL, Casula M.

Atheroscler Suppl. 2018 Sep;35:e14-e20. doi: 10.1016/j.atherosclerosissup.2018.08.003. Epub 2018 Aug 25.

PMID:
30177370
9.

[Stress levels and coping behavior in patients with chronic insomnia].

Zhuravlyova EV, Dubinina EA, Korostovtseva LS, Filchenko IA, Bochkarev MV, Stankova EP, Sviryaev YV, Alekhin AN, Konradi AO.

Zh Nevrol Psikhiatr Im S S Korsakova. 2018;118(4. Vyp. 2):35-42. doi: 10.17116/jnevro20181184235. Russian.

PMID:
30059050
10.

[Social-demographic aspects of insomnia in the Russian population according to ESSE-RF study].

Bochkarev MV, Korostovtseva LS, Filchenko IA, Rotar OP, Sviryaev YV, Zhernakova YV, Shalnova SA, Konradi AO, Boitsov SA, Chazova IE, Shlyakhto EV.

Zh Nevrol Psikhiatr Im S S Korsakova. 2018;118(4. Vyp. 2):26-34. doi: 10.17116/jnevro20181184226. Russian.

PMID:
30059049
11.

Haplotype Sharing Provides Insights into Fine-Scale Population History and Disease in Finland.

Martin AR, Karczewski KJ, Kerminen S, Kurki MI, Sarin AP, Artomov M, Eriksson JG, Esko T, Genovese G, Havulinna AS, Kaprio J, Konradi A, Korányi L, Kostareva A, Männikkö M, Metspalu A, Perola M, Prasad RB, Raitakari O, Rotar O, Salomaa V, Groop L, Palotie A, Neale BM, Ripatti S, Pirinen M, Daly MJ.

Am J Hum Genet. 2018 May 3;102(5):760-775. doi: 10.1016/j.ajhg.2018.03.003. Epub 2018 Apr 26.

12.

Autoantibodies to endothelial cells in patients with hypertensive disorders during pregnancy.

Ziganshina MM, Amiraslanov EY, Yarotskaya EL, Dolgushina NV, Sergunina OA, Nikolaeva MA, Kan NE, Tyutyunnik VL, Mantrova DA, Loginova NS, Konradi AO, Sukhikh GT.

Pregnancy Hypertens. 2018 Apr;12:65-70. doi: 10.1016/j.preghy.2018.02.010. Epub 2018 Mar 3. No abstract available.

PMID:
29674202
13.

[Elevated Level of the Natriuretic Peptide Among Adult Population in Regions Participating in the ESSE-RF Study and Its Association With Cardiovascular Diseases and Risk Factors].

Shalnova SA, Imaeva AE, Deev AD, Metelskaya VA, Muromtseva GA, Konradi AO, Masenko VP, Efanov AY, Kulakova NV, Rotar OP, Trubacheva IA, Shabunova AA, SHlyakhto EV, Boytsov SA.

Kardiologiia. 2017 Dec;57(12):43-52. Russian.

PMID:
29466210
14.

Effects of metabolic syndrome on arterial function in different age groups: the Advanced Approach to Arterial Stiffness study.

Topouchian J, Labat C, Gautier S, Bäck M, Achimastos A, Blacher J, Cwynar M, de la Sierra A, Pall D, Fantin F, Farkas K, Garcia-Ortiz L, Hakobyan Z, Jankowski P, Jelakovic A, Kobalava Z, Konradi A, Kotovskaya Y, Kotsani M, Lazareva I, Litvin A, Milyagin V, Mintale I, Persson O, Ramos R, Rogoza A, Ryliskyte L, Scuteri A, Sirenko Y, Soulis G, Tasic N, Udovychenko M, Urazalina S, Wohlfahrt P, Zelveian P, Benetos A, Asmar R.

J Hypertens. 2018 Apr;36(4):824-833. doi: 10.1097/HJH.0000000000001631.

15.

Predictors of heart rhythm disturbances in hypertensive obese patients with obstructive sleep apnea.

Korostovtseva LS, Zvartau NE, Rotar OP, Sviryaev YV, Konradi AO.

J Geriatr Cardiol. 2017 Sep;14(9):553-562. doi: 10.11909/j.issn.1671-5411.2017.09.010.

16.

Subclinical target organ damage in subjects with different components of metabolic syndrome.

Rotar OP, Boyarinova MA, Moguchaia EV, Kolesova EP, Erina AM, Solntsev VN, Konradi AO, Shlyakhto EV.

Clin Exp Hypertens. 2018;40(5):421-426. doi: 10.1080/10641963.2017.1384488. Epub 2017 Oct 25.

PMID:
29068233
17.

[The role of subjective methods for the evaluation of sleep quality].

Gortseva AY, Korostovtseva LS, Bochkarev MV, Sviryaev YV, Konradi AO.

Zh Nevrol Psikhiatr Im S S Korsakova. 2017;117(4. Vyp. 2):34-41. doi: 10.17116/jnevro20171174234-41. Russian.

PMID:
28777362
18.

[Optimization of BP Control and Arterial Elasticity With Fixed Combination Therapy Perindopril and Amlodipine In Patients With Arterial Hypertension and Increased Pulse Wave Velocity].

Nedogoda SV, Konradi AO, Zvartau NE, Chumachek EV, Ledyaeva AA, Tsoma VV, Salasyuk AS, Judina JS, Smirnova VO, Khripaeva VJ, Palashkin RV.

Kardiologiia. 2017 Mar;57(3):31-38. Russian.

PMID:
28762933
19.

[Adipokines Level in Metabolically Healthy Obese Saint-Petersburg Inhabitants (ESSE-RF)].

Boyarinova MA, Orlov AV, Rotar OP, Alieva AS, Moguchaya EV, Vasileva EU, Soltsev VN, Baranova EI, Konradi AO.

Kardiologiia. 2016 Aug;56(8):40-45. Russian.

PMID:
28290879
20.

Metabolically healthy obese and metabolically unhealthy non-obese phenotypes in a Russian population.

Rotar O, Boyarinova M, Orlov A, Solntsev V, Zhernakova Y, Shalnova S, Deev A, Konradi A, Baranova E, Chazova I, Boytsov S, Shlyakhto E.

Eur J Epidemiol. 2017 Mar;32(3):251-254. doi: 10.1007/s10654-016-0221-z. Epub 2016 Dec 30.

PMID:
28039558
21.

[BRADY-ARRHYTHMIAS IN THE OBSTRUCTIVE SLEEP APNEA SYNDROME: DANGEROUS COMPLICATION OR DEFENSE MECHANISM?].

Korostovtseva LS, Kravchenko SO, Sviryaev YV, Konradi AO, Oganesyan GA.

Zh Evol Biokhim Fiziol. 2016 Jul;52(4):275-280. Review. Russian.

PMID:
30695298
22.

Lifetime Prevalence of Transient Loss of Consciousness in an Urban Russian Population.

Gudkova S, Cherepanova N, Duplyakov D, Golovina G, Khokhlunov S, Surkova E, Rotar O, Konradi A, Shlyakhto E.

Arq Bras Cardiol. 2016 May;106(5):382-8. doi: 10.5935/abc.20160056. Epub 2016 Apr 15. English, Portuguese.

23.

[Gender Differences of Behavioral Risk Factors in Saint-Petersburg Inhabitants].

Orlov AV, Rotar OP, Boyarinova MA, Alieva AS, Dudorova EA, Kolesova EP, Moguchaya EV, Paskar NA, Solntsev VN, Baranova EA, Konradi AO.

Vestn Ross Akad Med Nauk. 2015;(5):585-91. Russian.

PMID:
26846085
24.

Continuation of the ESH-CHL-SHOT trial after publication of the SPRINT: rationale for further study on blood pressure targets of antihypertensive treatment after stroke.

Zanchetti A, Liu L, Mancia G, Parati G, Grassi G, Stramba-Badiale M, Silani V, Bilo G, Corrao G, Zambon A, Scotti L, Zhang X, Guan TR, Zhang Y, Zhang X, Berge E, Redon J, Narkiewicz K, Dominiczak A, Nilsson P, Viigimaa M, Laurent S, Agabiti-Rosei E, Wu Z, Zhu D, Rodicio JL, Ruilope LM, Martell-Claros N, Pinto F, Schmieder RE, Burnier M, Banach M, Cifkova R, Farsang C, Konradi A, Lazareva I, Sirenko Y, Dorobantu M, Postadzhiyan A, Accetto R, Jelakovic B, Lovic D, Manolis AJ, Stylianou P, Dicker D, Wei G, Xu C, Xie H, Coca A, O'Brien J, Ford G; ESH-CHL-SHOT trial investigators.

J Hypertens. 2016 Mar;34(3):393-6. doi: 10.1097/HJH.0000000000000853. No abstract available.

PMID:
26780185
25.

[AGED CARDIOHEMODYNAMICS COMPLICATED BY STROKE].

Nesterov VP, Ballyzek MF, Konradi AO, Burdygin AI, Korotkov SM, Shemarova IV, Cygvinzev SN, Nesterov SV.

Adv Gerontol. 2016;29(1):107-115. Russian.

PMID:
28423255
26.

Is Mixed Apnea Associated with Non-Rapid Eye Movement Sleep a Reversible Compensatory Sign of Heart Failure?

Korostovtseva L, Sazonova Y, Zvartau N, Semenov A, Nepran V, Bochkarev M, Nikolaev G, Mitrofanova L, Sviryaev Y, Gordeev M, Konradi A.

Am J Case Rep. 2015 Dec 18;16:886-92.

27.

Siege of Leningrad Survivors Phenotyping and Biospecimen Collection.

Rotar OP, Moguchaya EV, Boyarinova MA, Alieva AS, Orlov AV, Vasilieva EY, Yudina VA, Anisimov SV, Konradi AO.

Biopreserv Biobank. 2015 Oct;13(5):371-5. doi: 10.1089/bio.2015.0018. Epub 2015 Sep 29.

PMID:
26417917
28.

Seventy years after the siege of Leningrad: does early life famine still affect cardiovascular risk and aging?

Rotar O, Moguchaia E, Boyarinova M, Kolesova E, Khromova N, Freylikhman O, Smolina N, Solntsev V, Kostareva A, Konradi A, Shlyakhto E.

J Hypertens. 2015 Sep;33(9):1772-9; discussion 1779. doi: 10.1097/HJH.0000000000000640.

PMID:
26136204
29.

Marinobufagenin-induced vascular fibrosis is a likely target for mineralocorticoid antagonists.

Fedorova OV, Emelianov IV, Bagrov KA, Grigorova YN, Wei W, Juhasz O, Frolova EV, Marshall CA, Lakatta EG, Konradi AO, Bagrov AY.

J Hypertens. 2015 Aug;33(8):1602-10. doi: 10.1097/HJH.0000000000000591.

30.

[Clinical features of obstructive sleep apnea syndrome in patients with acromegaly].

Tsoy UA, Sviryaev YV, Korostovtseva LS, Semenov AP, Vaulina DA, Nepran VI, Kravchenko SO, Konradi AO, Grineva EN.

Ter Arkh. 2015;87(4):47-52. doi: 10.17116/terarkh201587447-52. Russian.

PMID:
26087634
31.

Association of adipokines with metabolic disorders in patients with schizophrenia: Results of comparative study with mental healthy cohort.

Tanyanskiy DA, Martynikhin IA, Rotar OP, Konradi AO, Sokolian NA, Neznanov NG, Denisenko AD.

Diabetes Metab Syndr. 2015 Jul-Sep;9(3):163-7. doi: 10.1016/j.dsx.2015.04.009. Epub 2015 Apr 24.

PMID:
25952038
32.

[Prevalence of cardiiovascular risk factors in Russian population of patients with arterial hypertension].

Chazova IE, Zhernakova IuV, Oshchepkova EV, Shal'nova SA, Iarovaia EB, Konradi AO, Boĭtsov SA.

Kardiologiia. 2014;54(10):4-12. Russian.

PMID:
25675714
33.

WISP1 is a novel adipokine linked to inflammation in obesity.

Murahovschi V, Pivovarova O, Ilkavets I, Dmitrieva RM, Döcke S, Keyhani-Nejad F, Gögebakan Ö, Osterhoff M, Kemper M, Hornemann S, Markova M, Klöting N, Stockmann M, Weickert MO, Lamounier-Zepter V, Neuhaus P, Konradi A, Dooley S, von Loeffelholz C, Blüher M, Pfeiffer AF, Rudovich N.

Diabetes. 2015 Mar;64(3):856-66. doi: 10.2337/db14-0444. Epub 2014 Oct 3.

34.

Blood pressure and LDL-cholesterol targets for prevention of recurrent strokes and cognitive decline in the hypertensive patient: design of the European Society of Hypertension-Chinese Hypertension League Stroke in Hypertension Optimal Treatment randomized trial.

Zanchetti A, Liu L, Mancia G, Parati G, Grassi G, Stramba-Badiale M, Silani V, Bilo G, Corrao G, Zambon A, Scotti L, Zhang X, Wang H, Zhang Y, Zhang X, Guan TR, Berge E, Redon J, Narkiewicz K, Dominiczak A, Nilsson P, Viigimaa M, Laurent S, Agabiti-Rosei E, Wu Z, Zhu D, Rodicio JL, Ruilope LM, Martell-Claros N, Pinto F, Schmieder RE, Burnier M, Banach M, Cifkova R, Farsang C, Konradi A, Lazareva I, Sirenko Y, Dorobantu M, Postadzhiyan A, Accetto R, Jelakovic B, Lovic D, Manolis AJ, Stylianou P, Erdine S, Dicker D, Wei G, Xu C, Xie H, Coca A, O'Brien J, Ford G.

J Hypertens. 2014 Sep;32(9):1888-97. doi: 10.1097/HJH.0000000000000254.

PMID:
24979303
35.

Blood pressure and low-density lipoprotein-cholesterol lowering for prevention of strokes and cognitive decline: a review of available trial evidence.

Zanchetti A, Liu L, Mancia G, Parati G, Grassi G, Stramba-Badiale M, Silani V, Bilo G, Corrao G, Zambon A, Scotti L, Zhang X, Wang H, Zhang Y, Zhang X, Guan TR, Berge E, Redon J, Narkiewicz K, Dominiczak A, Nilsson P, Viigimaa M, Laurent S, Agabiti-Rosei E, Wu Z, Zhu D, Rodicio JL, Ruilope LM, Martell-Claros N, Pinto F, Schmieder RE, Burnier M, Banach M, Cifkova R, Farsang C, Konradi A, Lazareva I, Sirenko Y, Dorobantu M, Postadzhiyan A, Accetto R, Jelakovic B, Lovic D, Manolis AJ, Stylianou P, Erdine S, Dicker D, Wei G, Xu C, Xie H, Coca A, O'Brien J, Ford G.

J Hypertens. 2014 Sep;32(9):1741-50. doi: 10.1097/HJH.0000000000000253. Review.

PMID:
24979302
36.

New insights into the management of rhythm and conduction disorders after acute myocardial infarction.

Korostovtseva L, Sviryaev Y, Zvartau N, Druzhkova T, Tikhonenko V, Konradi A.

Am J Case Rep. 2014 Apr 19;15:159-62. doi: 10.12659/AJCR.890357. eCollection 2014.

37.

Day-to-day repeatability of the Pulse Time Index of Norm.

Posokhov IN, Konradi AO, Shlyakhto EV, Mamontov OV, Orlov AV, Rogoza AN.

Med Devices (Auckl). 2014 Feb 27;7:29-33. doi: 10.2147/MDER.S58507. eCollection 2014.

38.

Effects of rituximab therapy on elastic properties of vascular wall in patients with progressive systemic sclerosis.

Maslyanskiy AL, Lapin SV, Kolesova EP, Penin IN, Cheshuina MD, Feist E, Konradi AO.

Clin Exp Rheumatol. 2014 Nov-Dec;32(6 Suppl 86):S-228. Epub 2014 Jan 30. No abstract available.

PMID:
24480389
39.

[The prevalence of anxiety and depression in different regions of the Russian Federation and its association with sociodemographic factors (according to the data of the ESSE-RF study)].

Shal'nova SA, Evstifeeva SE, Deev AD, Artamova GV, Gatagonova TM, Dupliakov DV, Efanov AIu, Zhernakova IuV, Konradi AO, Libis RA, Minakov EV, Nedogoda SV, Oshchepkova EV, Romanchuk SV, Rotar' OP, Trubacheva IA, SHliakhto EV, Boitsov SA.

Ter Arkh. 2014;86(12):53-60. Russian.

PMID:
25804041
40.

[Effectiveness of diagnostics and treatment of complicated hypertensive disease taking into account results of 3 day arterial pressure monitoring].

Mamontov OV, Katinas GS, Konradi AO, Shliakhto EV, Emel'ianov IV, Bogachev MI, Markelov OA.

Klin Med (Mosk). 2014;92(9):33-8. Russian.

PMID:
25790709
41.

High prevalence of human cytomegalovirus in carotid atherosclerotic plaques obtained from Russian patients undergoing carotid endarterectomy.

Yaiw KC, Ovchinnikova O, Taher C, Mohammad AA, Davoudi B, Shlyakhto E, Rotar O, Konradi A, Wilhelmi V, Rahbar A, Butler L, Assinger A, Söderberg-Nauclér C.

Herpesviridae. 2013 Nov 14;4(1):3. doi: 10.1186/2042-4280-4-3.

42.

Label free fragment screening using surface plasmon resonance as a tool for fragment finding - analyzing parkin, a difficult CNS target.

Regnström K, Yan J, Nguyen L, Callaway K, Yang Y, Diep L, Xing W, Adhikari A, Beroza P, Hom RK, Riley B, Rudolph D, Jobling MF, Baker J, Johnston J, Konradi A, Bova MP, Artis DR.

PLoS One. 2013 Jul 5;8(7):e66879. doi: 10.1371/journal.pone.0066879. Print 2013. Erratum in: PLoS One. 2013;8(7). doi:10.1371/annotation/590bbe38-3a12-45bd-bc5d-83b766c968b3. Artis, Rick D [corrected to Artis, Dean R].

43.

Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: prime side chromane-containing inhibitors.

Ng RA, Sun M, Bowers S, Hom RK, Probst GD, John V, Fang LY, Maillard M, Gailunas A, Brogley L, Neitz RJ, Tung JS, Pleiss MA, Konradi AW, Sham HL, Dappen MS, Adler M, Yao N, Zmolek W, Nakamura D, Quinn KP, Sauer JM, Bova MP, Ruslim L, Artis DR, Yednock TA.

Bioorg Med Chem Lett. 2013 Aug 15;23(16):4674-9. doi: 10.1016/j.bmcl.2013.06.006. Epub 2013 Jun 11.

PMID:
23856050
44.

[Estimation of the information value of diagnostic data obtained by bio-radiolocation pneumography in non-contact screening of sleep apnea syndrome].

Alekhin MD, Anishchenko LN, Zhuravlev AV, Ivashov SI, Korostovtseva LS, Sviriaev IuV, Konradi AO, Parashin VB, Bogomolov AV.

Med Tekh. 2013 Mar-Apr;(2):36-8. Russian. No abstract available.

PMID:
23789156
45.

Selective and brain-permeable polo-like kinase-2 (Plk-2) inhibitors that reduce α-synuclein phosphorylation in rat brain.

Aubele DL, Hom RK, Adler M, Galemmo RA Jr, Bowers S, Truong AP, Pan H, Beroza P, Neitz RJ, Yao N, Lin M, Tonn G, Zhang H, Bova MP, Ren Z, Tam D, Ruslim L, Baker J, Diep L, Fitzgerald K, Hoffman J, Motter R, Fauss D, Tanaka P, Dappen M, Jagodzinski J, Chan W, Konradi AW, Latimer L, Zhu YL, Sham HL, Anderson JP, Bergeron M, Artis DR.

ChemMedChem. 2013 Aug;8(8):1295-313. doi: 10.1002/cmdc.201300166. Epub 2013 Jun 21.

PMID:
23794260
46.

Orally available and efficacious α4β1/α4β7 integrin inhibitors.

Xu YZ, Smith JL, Semko CM, Rossiter KI, Fukuda JY, Dappen MS, Quincy DA, Konradi AW, Mao W, Welch B, Dreyer ML, Samant B, Zhang H, Lugar J, Liao Z, Henschel C, Petersen E, Vandevert C, Shoemaker M, Wehner N, Mutter L, Shopp G, Krimm M, Chen L, Wipke B, Dofiles L, Gallager I, Sauer JM, Messersmith EK, Pleiss MA, Bard F, Yednock TA.

Bioorg Med Chem Lett. 2013 Aug 1;23(15):4370-3. doi: 10.1016/j.bmcl.2013.05.076. Epub 2013 May 31.

PMID:
23777782
47.

PEG conjugates of potent α4 integrin inhibitors, maintaining sustained levels and bioactivity in vivo, following subcutaneous administration.

Smith JL, Rossiter KI, Semko CM, Xu YZ, Quincy DA, Jagodzinski J, Dappen MS, Konradi AW, Vandevert C, Garrido C, Mao W, San Pablo FB, Wipke B, Dofiles L, Wadsworth A, Peterson E, Lorenzana C, Simmonds S, Messersmith EK, Bard F, Pleiss MA, Yednock TA.

Bioorg Med Chem Lett. 2013 Jul 15;23(14):4117-9. doi: 10.1016/j.bmcl.2013.05.048. Epub 2013 May 24.

PMID:
23743283
48.

Discovery of (R)-4-cyclopropyl-7,8-difluoro-5-(4-(trifluoromethyl)phenylsulfonyl)-4,5-dihydro-1H-pyrazolo[4,3-c]quinoline (ELND006) and (R)-4-cyclopropyl-8-fluoro-5-(6-(trifluoromethyl)pyridin-3-ylsulfonyl)-4,5-dihydro-2H-pyrazolo[4,3-c]quinoline (ELND007): metabolically stable γ-secretase Inhibitors that selectively inhibit the production of amyloid-β over Notch.

Probst G, Aubele DL, Bowers S, Dressen D, Garofalo AW, Hom RK, Konradi AW, Marugg JL, Mattson MN, Neitzel ML, Semko CM, Sham HL, Smith J, Sun M, Truong AP, Ye XM, Xu YZ, Dappen MS, Jagodzinski JJ, Keim PS, Peterson B, Latimer LH, Quincy D, Wu J, Goldbach E, Ness DK, Quinn KP, Sauer JM, Wong K, Zhang H, Zmolek W, Brigham EF, Kholodenko D, Hu K, Kwong GT, Lee M, Liao A, Motter RN, Sacayon P, Santiago P, Willits C, Bard F, Bova MP, Hemphill SS, Nguyen L, Ruslim L, Tanaka K, Tanaka P, Wallace W, Yednock TA, Basi GS.

J Med Chem. 2013 Jul 11;56(13):5261-74. doi: 10.1021/jm301741t. Epub 2013 Jun 20.

PMID:
23713656
49.

Arylsulfonamide pyrimidines as VLA-4 antagonists.

Xu YZ, Konradi AW, Bard F, Dappen M, Dofiles L, Dreyer M, Gallager I, Garrido C, Krimm M, Liao Z, Messersmith E, Mutter L, Pleiss MA, Samant B, Semko CM, Smith J, Stappenbeck F, Stupi B, Vandervert C, Welch B, Wipke B, Yednock T.

Bioorg Med Chem Lett. 2013 May 15;23(10):3070-4. doi: 10.1016/j.bmcl.2013.03.010. Epub 2013 Mar 15.

PMID:
23562062
50.

Cross-linking density and temperature effects on the self-assembly of SiO2-PNIPAAm core-shell particles at interfaces.

Nazli KO, Pester CW, Konradi A, Böker A, van Rijn P.

Chemistry. 2013 Apr 26;19(18):5586-94. doi: 10.1002/chem.201203900. Epub 2013 Mar 28.

PMID:
23554025

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