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Items: 1 to 50 of 74

1.

Polyoxygenated Tertiary Alcohols: A Kiyooka Approach.

Lücke D, Kalesse M.

Chemistry. 2019 Jun 7. doi: 10.1002/chem.201902589. [Epub ahead of print]

PMID:
31173411
2.

Synthesis of sulfonamide, amide and amine hybrid pharmacophore, an entry of new class of carbonic anhydrase II inhibitors and evaluation of chemo-informatics and binding analysis.

Ahmed A, Channar PA, Saeed A, Kalesse M, Kazi MA, Larik FA, Abbas Q, Hassan M, Raza H, Seo SY.

Bioorg Chem. 2019 May;86:624-630. doi: 10.1016/j.bioorg.2019.01.060. Epub 2019 Feb 10.

PMID:
30807935
3.

Resolving Inflammation: Synthesis, Configurational Assignment, and Biological Evaluations of RvD1n-3 DPA.

Tungen JE, Gerstmann L, Vik A, De Matteis R, Colas RA, Dalli J, Chiang N, Serhan CN, Kalesse M, Hansen TV.

Chemistry. 2019 Jan 28;25(6):1476-1480. doi: 10.1002/chem.201806029. Epub 2018 Dec 20.

PMID:
30511787
4.

Corrigendum to "Bumepamine, a brain-permeant benzylamine derivative of bumetanide, does not inhibit NKCC1 but is more potent to enhance phenobarbital's antiseizure efficacy" [Neuropharmacology 143 (2018) 186-204].

Brandt C, Seja P, Töllner K, Römermann K, Hampel P, Kalesse M, Kipper A, Feit PW, Lykke K, Toft-Bertelsen TL, Paavilainen P, Spoljaric I, Puskarjov M, MacAulay N, Kaila K, Löscher W.

Neuropharmacology. 2018 Dec;143:349-350. doi: 10.1016/j.neuropharm.2018.10.012. Epub 2018 Oct 19. No abstract available.

PMID:
30343990
5.

Bumepamine, a brain-permeant benzylamine derivative of bumetanide, does not inhibit NKCC1 but is more potent to enhance phenobarbital's anti-seizure efficacy.

Brandt C, Seja P, Töllner K, Römermann K, Hampel P, Kalesse M, Kipper A, Feit PW, Lykke K, Toft-Bertelsen TL, Paavilainen P, Spoljaric I, Puskarjov M, MacAulay N, Kaila K, Löscher W.

Neuropharmacology. 2018 Dec;143:186-204. doi: 10.1016/j.neuropharm.2018.09.025. Epub 2018 Sep 21. Erratum in: Neuropharmacology. 2018 Oct 18;:.

PMID:
30248303
6.

Total Synthesis of Pericoannosin A.

Lücke D, Linne Y, Hempel K, Kalesse M.

Org Lett. 2018 Aug 3;20(15):4475-4477. doi: 10.1021/acs.orglett.8b01768. Epub 2018 Jul 13.

PMID:
30003789
7.

Painting argyrins blue: Negishi cross-coupling for synthesis of deep-blue tryptophan analogue β-(1-azulenyl)-l alanine and its incorporation into argyrin C.

Stempel E, Kaml RF, Budisa N, Kalesse M.

Bioorg Med Chem. 2018 Oct 15;26(19):5259-5269. doi: 10.1016/j.bmc.2018.03.037. Epub 2018 Mar 26.

PMID:
29729984
8.

The Rickiols: 20-, 22-, and 24-membered Macrolides from the Ascomycete Hypoxylon rickii.

Surup F, Kuhnert E, Böhm A, Pendzialek T, Solga D, Wiebach V, Engler H, Berkessel A, Stadler M, Kalesse M.

Chemistry. 2018 Feb 9;24(9):2200-2213. doi: 10.1002/chem.201704928. Epub 2018 Jan 19.

PMID:
29168908
9.

Biosynthesis and Total Synthesis of Pyrronazol B: a Secondary Metabolite from Nannocystis pusilla.

Witte SNR, Hug JJ, Géraldy MNE, Müller R, Kalesse M.

Chemistry. 2017 Nov 13;23(63):15917-15921. doi: 10.1002/chem.201703782. Epub 2017 Oct 24.

PMID:
28944573
10.

Total Synthesis of Nannocystin Ax.

Poock C, Kalesse M.

Org Lett. 2017 Sep 1;19(17):4536-4539. doi: 10.1021/acs.orglett.7b02112. Epub 2017 Aug 15.

PMID:
28809579
11.

RNA polymerase motions during promoter melting.

Feklistov A, Bae B, Hauver J, Lass-Napiorkowska A, Kalesse M, Glaus F, Altmann KH, Heyduk T, Landick R, Darst SA.

Science. 2017 May 26;356(6340):863-866. doi: 10.1126/science.aam7858.

12.

Therapeutic effects of Argyrin F in pancreatic adenocarcinoma.

Chen X, Bui KC, Barat S, Thi Nguyen ML, Bozko P, Sipos B, Kalesse M, Malek NP, Plentz RR.

Cancer Lett. 2017 Jul 28;399:20-28. doi: 10.1016/j.canlet.2017.04.003. Epub 2017 Apr 10.

PMID:
28408354
13.

Pinacol Coupling Strategy for the Construction of the Bicyclo[6.4.1]tridecane Framework of Schiglautone A.

Werner B, Kalesse M.

Org Lett. 2017 Apr 7;19(7):1524-1526. doi: 10.1021/acs.orglett.7b00288. Epub 2017 Mar 16.

PMID:
28300417
14.

Synthesis of Antibiotics.

Kalesse M, Böhm A, Kipper A, Wandelt V.

Curr Top Microbiol Immunol. 2016;398:419-445. doi: 10.1007/82_2016_502. Review.

PMID:
27704271
15.

Isolation, Structure Elucidation, and (Bio)Synthesis of Haprolid, a Cell-Type-Specific Myxobacterial Cytotoxin.

Steinmetz H, Li J, Fu C, Zaburannyi N, Kunze B, Harmrolfs K, Schmitt V, Herrmann J, Reichenbach H, Höfle G, Kalesse M, Müller R.

Angew Chem Int Ed Engl. 2016 Aug 16;55(34):10113-7. doi: 10.1002/anie.201603288. Epub 2016 Jul 12.

PMID:
27404448
16.

Total Synthesis of Aetheramide A.

Gerstmann L, Kalesse M.

Chemistry. 2016 Aug 1;22(32):11210-2. doi: 10.1002/chem.201602682. Epub 2016 Jul 4.

PMID:
27303862
17.

Isolation, Structure Elucidation, Biosynthesis, and Synthesis of Antalid, a Secondary Metabolite from Polyangium species.

Tautz T, Hoffmann J, Hoffmann T, Steinmetz H, Washausen P, Kunze B, Huch V, Kitsche A, Reichenbach H, Höfle G, Müller R, Kalesse M.

Org Lett. 2016 Jun 3;18(11):2560-3. doi: 10.1021/acs.orglett.6b00810. Epub 2016 May 24.

PMID:
27220069
18.

Correction to Synthesis of Omphadiol and Pyxidatol C.

Parthasarathy G, Eggert U, Kalesse M.

Org Lett. 2016 Jun 3;18(11):2792. doi: 10.1021/acs.orglett.6b01361. Epub 2016 May 17. No abstract available.

PMID:
27187085
19.

Synthesis of (+)-Omphadiol and (+)-Pyxidatol C.

Parthasarathy G, Eggert U, Kalesse M.

Org Lett. 2016 May 6;18(9):2320-2. doi: 10.1021/acs.orglett.6b00814. Epub 2016 Apr 22. Erratum in: Org Lett. 2016 Jun 3;18(11):2792.

PMID:
27105390
20.

Paleo-soraphens: chemical total syntheses and biological studies.

Lu HH, Hinkelmann B, Tautz T, Li J, Sasse F, Franke R, Kalesse M.

Org Biomol Chem. 2015 Aug 7;13(29):8029-36. doi: 10.1039/c5ob01249j. Epub 2015 Jun 29.

PMID:
26119264
21.

Soraphen A: A broad-spectrum antiviral natural product with potent anti-hepatitis C virus activity.

Koutsoudakis G, Romero-Brey I, Berger C, Pérez-Vilaró G, Monteiro Perin P, Vondran FW, Kalesse M, Harmrolfs K, Müller R, Martinez JP, Pietschmann T, Bartenschlager R, Brönstrup M, Meyerhans A, Díez J.

J Hepatol. 2015 Oct;63(4):813-21. doi: 10.1016/j.jhep.2015.06.002. Epub 2015 Jun 10.

PMID:
26070407
22.

The synthesis and biological evaluation of desepoxyisotedanolide and a comparison with desepoxytedanolide.

Naini A, Muthukumar Y, Raja A, Franke R, Harrier I, Smith AB 3rd, Lee D, Taylor RE, Sasse F, Kalesse M.

Angew Chem Int Ed Engl. 2015 Jun 1;54(23):6935-9. doi: 10.1002/anie.201501526. Epub 2015 Apr 27.

PMID:
25914374
23.

Ekkehard Winterfeldt (1932-2014).

Kalesse M.

Angew Chem Int Ed Engl. 2015 Jan 2;54(1):35. doi: 10.1002/anie.201410838. Epub 2014 Dec 4.

PMID:
25476468
24.

Antimalarial activity of the myxobacterial macrolide chlorotonil a.

Held J, Gebru T, Kalesse M, Jansen R, Gerth K, Müller R, Mordmüller B.

Antimicrob Agents Chemother. 2014 Nov;58(11):6378-84. doi: 10.1128/AAC.03326-14. Epub 2014 Aug 11.

25.

The structure elucidation and total synthesis of β-lipomycin.

Hartmann O, Kalesse M.

Angew Chem Int Ed Engl. 2014 Jul 7;53(28):7335-8. doi: 10.1002/anie.201402259. Epub 2014 May 21.

PMID:
24850084
26.

Baceridin, a cyclic hexapeptide from an epiphytic bacillus strain, inhibits the proteasome.

Niggemann J, Bozko P, Bruns N, Wodtke A, Gieseler MT, Thomas K, Jahns C, Nimtz M, Reupke I, Brüser T, Auling G, Malek N, Kalesse M.

Chembiochem. 2014 May 5;15(7):1021-9. doi: 10.1002/cbic.201300778. Epub 2014 Apr 1.

PMID:
24692199
27.

The vinylogous Mukaiyama aldol reaction (VMAR) in natural product synthesis.

Kalesse M, Cordes M, Symkenberg G, Lu HH.

Nat Prod Rep. 2014 Apr;31(4):563-94. doi: 10.1039/c3np70102f. Epub 2014 Mar 5. Review.

PMID:
24595879
28.

Structure elucidation and total synthesis of kulkenon.

Symkenberg G, Kalesse M.

Angew Chem Int Ed Engl. 2014 Feb 10;53(7):1795-8. doi: 10.1002/anie.201309386. Epub 2014 Jan 13.

PMID:
24420412
29.

Synthesis and biological evaluation of paleo-soraphens.

Lu HH, Raja A, Franke R, Landsberg D, Sasse F, Kalesse M.

Angew Chem Int Ed Engl. 2013 Dec 16;52(51):13549-52. doi: 10.1002/anie.201305331. Epub 2013 Nov 7.

PMID:
24346938
30.

Synthesis of angiolam A.

Gieseler MT, Kalesse M.

Org Lett. 2014 Jan 17;16(2):548-51. doi: 10.1021/ol403423r. Epub 2013 Dec 16.

PMID:
24341445
31.

Configurational assignment of secondary hydroxyl groups and methyl branches in polyketide natural products through bioinformatic analysis of the ketoreductase domain.

Kitsche A, Kalesse M.

Chembiochem. 2013 May 10;14(7):851-61. doi: 10.1002/cbic.201300063. Epub 2013 Apr 10.

PMID:
23576424
32.

Synthesis and pharmacology of proteasome inhibitors.

Rentsch A, Landsberg D, Brodmann T, Bülow L, Girbig AK, Kalesse M.

Angew Chem Int Ed Engl. 2013 May 17;52(21):5450-88. doi: 10.1002/anie.201207900. Epub 2013 Mar 25. Review.

PMID:
23526565
33.

The human cytomegalovirus UL51 protein is essential for viral genome cleavage-packaging and interacts with the terminase subunits pUL56 and pUL89.

Borst EM, Kleine-Albers J, Gabaev I, Babic M, Wagner K, Binz A, Degenhardt I, Kalesse M, Jonjic S, Bauerfeind R, Messerle M.

J Virol. 2013 Feb;87(3):1720-32. doi: 10.1128/JVI.01955-12. Epub 2012 Nov 21.

34.

The total synthesis of corallopyronin A and myxopyronin B.

Rentsch A, Kalesse M.

Angew Chem Int Ed Engl. 2012 Nov 5;51(45):11381-4. doi: 10.1002/anie.201206560. Epub 2012 Oct 8.

PMID:
23042599
35.

The total synthesis of (-)-aurafuron A.

Hartmann O, Kalesse M.

Org Lett. 2012 Jun 15;14(12):3064-7. doi: 10.1021/ol3011387. Epub 2012 May 25.

PMID:
22632656
36.

Pellasoren: structure elucidation, biosynthesis, and total synthesis of a cytotoxic secondary metabolite from Sorangium cellulosum.

Jahns C, Hoffmann T, Müller S, Gerth K, Washausen P, Höfle G, Reichenbach H, Kalesse M, Müller R.

Angew Chem Int Ed Engl. 2012 May 21;51(21):5239-43. doi: 10.1002/anie.201200327. Epub 2012 Apr 5. No abstract available.

PMID:
22488911
37.

Sulfangolids, macrolide sulfate esters from Sorangium cellulosum.

Zander W, Irschik H, Augustiniak H, Herrmann M, Jansen R, Steinmetz H, Gerth K, Kessler W, Kalesse M, Höfle G, Müller R.

Chemistry. 2012 May 14;18(20):6264-71. doi: 10.1002/chem.201100851. Epub 2012 Apr 4.

PMID:
22488821
38.

Syn-selective vinylogous Kobayashi aldol reaction.

Symkenberg G, Kalesse M.

Org Lett. 2012 Mar 16;14(6):1608-11. doi: 10.1021/ol300353w. Epub 2012 Mar 8.

PMID:
22400997
39.

An improved route to (+)-tedanolide and analysis of its subtle effects controlling conformation and biological behaviour.

Diaz N, Zhu M, Ehrlich G, Eggert U, Muthukumar Y, Sasse F, Kalesse M.

Chemistry. 2012 Apr 16;18(16):4946-52. doi: 10.1002/chem.201103038. Epub 2012 Mar 5.

PMID:
22392854
40.

Synthesis of simplified tedanolide analogues--connecting tedanolide to myriaporone and gephyronic acid.

Diaz N, Naini A, Muthukumar Y, Sasse F, Kalesse M.

ChemMedChem. 2012 May;7(5):771-5. doi: 10.1002/cmdc.201100576. Epub 2012 Mar 1.

PMID:
22383258
41.

A Kiyooka aldol approach for the synthesis of the C(14)-C(23) segment of the diastereomeric analog of tedanolide C.

Bülow L, Naini A, Fohrer J, Kalesse M.

Org Lett. 2011 Nov 18;13(22):6038-41. doi: 10.1021/ol202515x. Epub 2011 Oct 25.

PMID:
22026452
42.

Asymmetric vinylogous Mukaiyama aldol reaction of aldehyde-derived dienolates.

Gieseler MT, Kalesse M.

Org Lett. 2011 May 6;13(9):2430-2. doi: 10.1021/ol2006727. Epub 2011 Apr 7.

PMID:
21473644
43.

Mode of action of epoxyphomalins A and B and characterization of related metabolites from the marine-derived fungus Paraconiothyrium sp.

Mohamed IE, Kehraus S, Krick A, König GM, Kelter G, Maier A, Fiebig HH, Kalesse M, Malek NP, Gross H.

J Nat Prod. 2010 Dec 27;73(12):2053-6. doi: 10.1021/np100310k. Epub 2010 Nov 29.

PMID:
21114274
44.

Intramolecular stereoselective protonation of aldehyde-derived enolates.

Kena Diba A, Noll C, Richter M, Gieseler MT, Kalesse M.

Angew Chem Int Ed Engl. 2010 Nov 2;49(45):8367-9. doi: 10.1002/anie.201004619. No abstract available.

PMID:
20878962
45.

Total synthesis of chivosazole F.

Brodmann T, Janssen D, Kalesse M.

J Am Chem Soc. 2010 Oct 6;132(39):13610-1. doi: 10.1021/ja107290s.

PMID:
20836495
46.

Elucidation of the structure and intermolecular interactions of a reversible cyclic-peptide inhibitor of the proteasome by NMR spectroscopy and molecular modeling.

Stauch B, Simon B, Basile T, Schneider G, Malek NP, Kalesse M, Carlomagno T.

Angew Chem Int Ed Engl. 2010 May 25;49(23):3934-8. doi: 10.1002/anie.201000140. No abstract available.

PMID:
20408152
47.

Synthesis and biological characterization of argyrin F.

Bülow L, Nickeleit I, Girbig AK, Brodmann T, Rentsch A, Eggert U, Sasse F, Steinmetz H, Frank R, Carlomagno T, Malek NP, Kalesse M.

ChemMedChem. 2010 Jun 7;5(6):832-6. doi: 10.1002/cmdc.201000080. No abstract available. Erratum in: ChemMedChem. 2010 Jun 7;5(6):805.

PMID:
20358576
48.

The synthesis of novel disorazoles.

Schäckel R, Hinkelmann B, Sasse F, Kalesse M.

Angew Chem Int Ed Engl. 2010 Feb 22;49(9):1619-22. doi: 10.1002/anie.200906450. No abstract available.

PMID:
20099286
49.

The oxygen-independent coproporphyrinogen III oxidase HemN utilizes harderoporphyrinogen as a reaction intermediate during conversion of coproporphyrinogen III to protoporphyrinogen IX.

Rand K, Noll C, Schiebel HM, Kemken D, Dülcks T, Kalesse M, Heinz DW, Layer G.

Biol Chem. 2010 Jan;391(1):55-63. doi: 10.1515/BC.2010.006.

PMID:
19919179
50.

The absolute configuration of rhizopodin and its inhibition of actin polymerization by dimerization.

Hagelueken G, Albrecht SC, Steinmetz H, Jansen R, Heinz DW, Kalesse M, Schubert WD.

Angew Chem Int Ed Engl. 2009;48(3):595-8. doi: 10.1002/anie.200802915. No abstract available.

PMID:
19035596

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