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Items: 1 to 50 of 117

2.

Reactions of Piperazin-2-one, Morpholin-3-one, and Thiomorpholin-3-one with Triethyl Phosphite Prompted by Phosphoryl Chloride: Scope and Limitations.

Argüello-Velasco RO, Dziuk B, Zarychta B, Ordóñez M, Kafarski P.

ACS Omega. 2019 May 22;4(5):9056-9064. doi: 10.1021/acsomega.9b01137. eCollection 2019 May 31.

3.

Development of a high performance thin layer chromatography method for the rapid qualification and quantification of phenolic compounds and abscisic acid in honeys.

Stanek N, Kafarski P, Jasicka-Misiak I.

J Chromatogr A. 2019 Aug 2;1598:209-215. doi: 10.1016/j.chroma.2019.04.052. Epub 2019 Apr 19.

PMID:
31023479
4.

Recent advances in design of new urease inhibitors: A review.

Kafarski P, Talma M.

J Adv Res. 2018 Jan 31;13:101-112. doi: 10.1016/j.jare.2018.01.007. eCollection 2018 Sep. Review.

5.

HPTLC Fingerprinting-Rapid Method for the Differentiation of Honeys of Different Botanical Origin Based on the Composition of the Lipophilic Fractions.

Makowicz E, Jasicka-Misiak I, Teper D, Kafarski P.

Molecules. 2018 Jul 21;23(7). pii: E1811. doi: 10.3390/molecules23071811.

6.

Substituted phosphonic analogues of phenylglycine as inhibitors of phenylalanine ammonia lyase from potatoes.

Wanat W, Talma M, Hurek J, Pawełczak M, Kafarski P.

Biochimie. 2018 Aug;151:119-127. doi: 10.1016/j.biochi.2018.06.005. Epub 2018 Jun 15.

PMID:
29890205
7.

Addition of thiols to the double bond of dipeptide C-terminal dehydroalanine as a source of new inhibitors of cathepsin C.

Lenartowicz P, Makowski M, Oszywa B, Haremza K, Latajka R, Pawełczak M, Kafarski P.

Biochimie. 2017 Aug;139:46-55. doi: 10.1016/j.biochi.2017.05.011. Epub 2017 May 17.

PMID:
28528273
8.
9.

Biodegradation of the aminopolyphosphonate DTPMP by the cyanobacterium Anabaena variabilis proceeds via a C-P lyase-independent pathway.

Drzyzga D, Forlani G, Vermander J, Kafarski P, Lipok J.

Environ Microbiol. 2017 Mar;19(3):1065-1076. doi: 10.1111/1462-2920.13616. Epub 2017 Jan 23.

PMID:
27907245
10.

Synthetic Procedures Leading towards Aminobisphosphonates.

Chmielewska E, Kafarski P.

Molecules. 2016 Nov 4;21(11). pii: E1474. Review.

11.

Whole-cell Proteus mirabilis urease inhibition by aminophosphinates for the control of struvite formation.

Grela E, Dziełak A, Szydłowska K, Mucha A, Kafarski P, Grabowiecka AM.

J Med Microbiol. 2016 Oct;65(10):1123-1129. doi: 10.1099/jmm.0.000342. Epub 2016 Aug 22.

PMID:
27550502
12.

Structural Analogues of Selfotel.

Dziuganowska ZA, Ślepokura K, Volle JN, Virieux D, Pirat JL, Kafarski P.

J Org Chem. 2016 Jun 17;81(12):4947-54. doi: 10.1021/acs.joc.6b00220. Epub 2016 Jun 1.

PMID:
27187758
13.

Phytotoxicity of aminobisphosphonates targeting both δ1 -pyrroline-5-carboxylate reductase and glutamine synthetase.

Giberti S, Bertazzini M, Liboni M, Berlicki Ł, Kafarski P, Forlani G.

Pest Manag Sci. 2017 Feb;73(2):435-443. doi: 10.1002/ps.4299. Epub 2016 May 23.

PMID:
27103608
14.

The experimental osteoporosis in sheep--clinical approach.

Kiełbowicz Z, Piątek A, Bieżyński J, Skrzypczak P, Kuropka P, Kuryszko J, Nikodem A, Kafarski P, Pezowicz C.

Pol J Vet Sci. 2015;18(3):645-54. doi: 10.1515/pjvs-2015-0083.

PMID:
26618599
15.

Bisphosphonic acids as effective inhibitors of Mycobacterium tuberculosis glutamine synthetase.

Kosikowska P, Bochno M, Macegoniuk K, Forlani G, Kafarski P, Berlicki Ł.

J Enzyme Inhib Med Chem. 2016 Dec;31(6):931-8. doi: 10.3109/14756366.2015.1070846. Epub 2015 Aug 3.

PMID:
26235917
16.

Synthesis of dehydrodipeptide esters and their evaluation as inhibitors of cathepsin C.

Makowski M, Lenartowicz P, Oszywa B, Jewgiński M, Pawełczak M, Kafarski P.

Med Chem Res. 2015;24(8):3157-3165. Epub 2015 Apr 16.

17.

Do differences in chemical composition of stem and cap of Amanita muscaria fruiting bodies correlate with topsoil type?

Deja S, Wieczorek PP, Halama M, Jasicka-Misiak I, Kafarski P, Poliwoda A, Młynarz P.

PLoS One. 2014 Dec 1;9(12):e104084. doi: 10.1371/journal.pone.0104084. eCollection 2014.

18.

The overproduction of 2,4-DTBP accompanying to the lack of available form of phosphorus during the biodegradative utilization of aminophosphonates by Aspergillus terreus.

Lenartowicz P, Kafarski P, Lipok J.

Biodegradation. 2015 Feb;26(1):65-76. doi: 10.1007/s10532-014-9716-z. Epub 2014 Nov 12.

PMID:
25385070
19.

Amino polyphosphonates - chemical features and practical uses, environmental durability and biodegradation.

Studnik H, Liebsch S, Forlani G, Wieczorek D, Kafarski P, Lipok J.

N Biotechnol. 2015 Jan 25;32(1):1-6. doi: 10.1016/j.nbt.2014.06.007. Epub 2014 Jul 30. Review.

PMID:
25086362
20.

Rapid determination of ibotenic acid and muscimol in human urine.

Deja S, Jawień E, Jasicka-Misiak I, Halama M, Wieczorek P, Kafarski P, Młynarz P.

Magn Reson Chem. 2014 Nov;52(11):711-4. doi: 10.1002/mrc.4104. Epub 2014 Jul 20. No abstract available.

PMID:
25042675
21.

Addition of H-phosphonates to quinine-derived carbonyl compounds. An unexpected C9 phosphonate-phosphate rearrangement and tandem intramolecular piperidine elimination.

Górecki L, Mucha A, Kafarski P.

Beilstein J Org Chem. 2014 Apr 17;10:883-9. doi: 10.3762/bjoc.10.85. eCollection 2014.

22.

Synthesis of fluorescent (benzyloxycarbonylamino)(aryl)methylphosphonates.

Górniak MG, Czernicka A, Młynarz P, Balcerzak W, Kafarski P.

Beilstein J Org Chem. 2014 Mar 28;10:741-5. doi: 10.3762/bjoc.10.68. eCollection 2014.

23.

Conformation of dehydropentapeptides containing four achiral amino acid residues - controlling the role of L-valine.

Jewgiński M, Krzciuk-Gula J, Makowski M, Latajka R, Kafarski P.

Beilstein J Org Chem. 2014 Mar 14;10:660-6. doi: 10.3762/bjoc.10.58. eCollection 2014.

24.

Chemometrics as a tool of origin determination of Polish monofloral and multifloral honeys.

Zieliński L, Deja S, Jasicka-Misiak I, Kafarski P.

J Agric Food Chem. 2014 Apr 2;62(13):2973-81. doi: 10.1021/jf4056715. Epub 2014 Mar 18.

PMID:
24641200
25.

Mannitol in Amanita muscaria--an osmotic blood-brain barrier disruptor enhancing its hallucinogenic action?

Maciejczyk E, Kafarski P.

Med Hypotheses. 2013 Nov;81(5):766-7. doi: 10.1016/j.mehy.2013.07.048. Epub 2013 Aug 8.

PMID:
23932733
26.

Hydrophosphonylation of nanoparticle Schiff bases as a mean for preparation of aminophosphonate-functionalized nanoparticles.

Siemieniec J, Kafarski P, Plucinski P.

Molecules. 2013 Jul 18;18(7):8473-84. doi: 10.3390/molecules18078473.

27.

Synthesis and evaluation of effective inhibitors of plant δ1-pyrroline-5-carboxylate reductase.

Forlani G, Berlicki L, Duò M, Dziędzioła G, Giberti S, Bertazzini M, Kafarski P.

J Agric Food Chem. 2013 Jul 17;61(28):6792-8. doi: 10.1021/jf401234s. Epub 2013 Jul 3.

PMID:
23790100
28.

Toward very potent, non-covalent organophosphonate inhibitors of cathepsin C and related enzymes by 2-amino-1-hydroxy-alkanephosphonates dipeptides.

Drąg M, Wieczerzak E, Pawełczak M, Berlicki Ł, Grzonka Z, Kafarski P.

Biochimie. 2013 Aug;95(8):1640-9. doi: 10.1016/j.biochi.2013.05.006. Epub 2013 May 24.

PMID:
23712251
29.

Sublethal detergent concentrations increase metabolization of recalcitrant polyphosphonates by the cyanobacterium Spirulina platensis.

Forlani G, Bertazzini M, Giberti S, Wieczorek D, Kafarski P, Lipok J.

Environ Sci Pollut Res Int. 2013 May;20(5):3263-70. doi: 10.1007/s11356-012-1253-x. Epub 2012 Oct 23.

PMID:
23089958
30.

Phosphorylation as a method of tuning the enantiodiscrimination potency of quinine--an NMR study.

Górecki Ł, Berlicki Ł, Mucha A, Kafarski P, Ślepokura K, Rudzińska-Szostak E.

Chirality. 2012 Apr;24(4):318-28. doi: 10.1002/chir.22000. Epub 2012 Feb 17.

PMID:
22344893
31.

Phosphonate degradation by Spirulina strains: cyanobacterial biofilters for the removal of anticorrosive polyphosphonates from wastewater.

Forlani G, Prearo V, Wieczorek D, Kafarski P, Lipok J.

Enzyme Microb Technol. 2011 Mar 7;48(3):299-305. doi: 10.1016/j.enzmictec.2010.12.005. Epub 2010 Dec 21.

PMID:
22112915
32.

Comparative study of fungal cell disruption--scope and limitations of the methods.

Klimek-Ochab M, Brzezińska-Rodak M, Zymańczyk-Duda E, Lejczak B, Kafarski P.

Folia Microbiol (Praha). 2011 Sep;56(5):469-75. doi: 10.1007/s12223-011-0069-2. Epub 2011 Sep 8.

33.

Vibrational characterization of L-leucine phosphonate analogues: FT-IR, FT-Raman, and SERS spectroscopy studies and DFT calculations.

Podstawka-Proniewicz E, Piergies N, Skołuba D, Kafarski P, Kim Y, Proniewicz LM.

J Phys Chem A. 2011 Oct 13;115(40):11067-78. doi: 10.1021/jp207101m. Epub 2011 Sep 19.

PMID:
21888349
34.

Remarkable potential of the α-aminophosphonate/phosphinate structural motif in medicinal chemistry.

Mucha A, Kafarski P, Berlicki Ł.

J Med Chem. 2011 Sep 8;54(17):5955-80. doi: 10.1021/jm200587f. Epub 2011 Aug 5. No abstract available.

PMID:
21780776
35.

Biocatalytic resolution of enantiomeric mixtures of 1-aminoethanephosphonic acid.

Brzezińska-Rodak M, Klimek-Ochab M, Zymańczyk-Duda E, Kafarski P.

Molecules. 2011 Jul 14;16(7):5896-904. doi: 10.3390/molecules16075896.

36.

Δ1-pyrroline-5-carboxylate reductase as a new target for therapeutics: inhibition of the enzyme from Streptococcus pyogenes and effects in vivo.

Forlani G, Petrollino D, Fusetti M, Romanini L, Nocek B, Joachimiak A, Berlicki L, Kafarski P.

Amino Acids. 2012 Jun;42(6):2283-91. doi: 10.1007/s00726-011-0970-7. Epub 2011 Jul 9.

37.

N-substituted aminomethanephosphonic and aminomethane-P-methylphosphinic acids as inhibitors of ureases.

Berlicki L, Bochno M, Grabowiecka A, Białas A, Kosikowska P, Kafarski P.

Amino Acids. 2012 May;42(5):1937-45. doi: 10.1007/s00726-011-0920-4. Epub 2011 May 11.

38.

Selective synthesis of α-fluoro-β-keto- and α-fluoro-β-aminophosphonates via electrophilic fluorination by selectfluor.

Radwan-Olszewska K, Palacios F, Kafarski P.

J Org Chem. 2011 Feb 18;76(4):1170-3. doi: 10.1021/jo102276y. Epub 2011 Jan 18.

PMID:
21244062
39.

Computer-aided optimization of phosphinic inhibitors of bacterial ureases.

Vassiliou S, Kosikowska P, Grabowiecka A, Yiotakis A, Kafarski P, Berlicki L.

J Med Chem. 2010 Aug 12;53(15):5597-606. doi: 10.1021/jm100340m.

PMID:
20684601
40.

Possible fungistatic implications of betulin presence in betulaceae plants and their hymenochaetaceae parasitic fungi.

Jasicka-Misiak I, Lipok J, Swider IA, Kafarski P.

Z Naturforsch C J Biosci. 2010 Mar-Apr;65(3-4):201-6.

PMID:
20469638
41.

Metallo-aminopeptidase inhibitors.

Mucha A, Drag M, Dalton JP, Kafarski P.

Biochimie. 2010 Nov;92(11):1509-29. doi: 10.1016/j.biochi.2010.04.026. Epub 2010 May 10. Review.

PMID:
20457213
42.

Structure of the Plasmodium falciparum M17 aminopeptidase and significance for the design of drugs targeting the neutral exopeptidases.

McGowan S, Oellig CA, Birru WA, Caradoc-Davies TT, Stack CM, Lowther J, Skinner-Adams T, Mucha A, Kafarski P, Grembecka J, Trenholme KR, Buckle AM, Gardiner DL, Dalton JP, Whisstock JC.

Proc Natl Acad Sci U S A. 2010 Feb 9;107(6):2449-54. doi: 10.1073/pnas.0911813107. Epub 2010 Jan 21.

43.

Specificity of the zinc(II), magnesium(II) and calcium(II) complexation by (pyridin-2-yl)aminomethane-1,1-diphosphonic acids and related 1,3-(thiazol-2-yl) and 1,3-(benzothiazol-2-yl) derivatives.

Matczak-Jon E, Kowalik-Jankowska T, Slepokura K, Kafarski P, Rajewska A.

Dalton Trans. 2010 Feb 7;39(5):1207-21. doi: 10.1039/b914647d. Epub 2009 Nov 19.

PMID:
20104347
44.

Plasmodium falciparum neutral aminopeptidases: new targets for anti-malarials.

Skinner-Adams TS, Stack CM, Trenholme KR, Brown CL, Grembecka J, Lowther J, Mucha A, Drag M, Kafarski P, McGowan S, Whisstock JC, Gardiner DL, Dalton JP.

Trends Biochem Sci. 2010 Jan;35(1):53-61. doi: 10.1016/j.tibs.2009.08.004. Epub 2009 Sep 30. Review.

PMID:
19796954
45.

Effectiveness and mode of action of phosphonate inhibitors of plant glutamine synthetase.

Occhipinti A, Berlicki Ł, Giberti S, Dziedzioła G, Kafarski P, Forlani G.

Pest Manag Sci. 2010 Jan;66(1):51-8. doi: 10.1002/ps.1830.

46.

Proteases as anti-cancer targets--molecular and biological basis for development of inhibitor-like drugs against cancer.

Białas A, Kafarski P.

Anticancer Agents Med Chem. 2009 Sep;9(7):728-62. Epub 2009 Sep 1. Review.

PMID:
19538170
47.

Conformational isomers of the [(5-methyl-2-pyridinio)aminomethylene]diphosphonate dianion and [(5-methyl-2-pyridyl)aminomethylene]diphosphonate trianion in salts with 4-aminopyridine and ammonia.

Matczak-Jon E, Slepokura K, Kafarski P, Skrzyńska I, Jon M.

Acta Crystallogr C. 2009 Jun;65(Pt 6):o261-6. doi: 10.1107/S0108270109010683. Epub 2009 May 2.

PMID:
19498233
48.

Enantiodifferentiation of alpha-hydroxyalkanephosphonic acids in 31P NMR with application of alpha-cyclodextrin as chiral discriminating agent.

Rudzińska E, Dziedzioła G, Berlicki L, Kafarski P.

Chirality. 2010 Jan;22(1):63-8. doi: 10.1002/chir.20707.

PMID:
19306429
49.

Theoretical study of spin-spin coupling across the hydrogen (O-H...N) bond in adenosine derivatives.

Doskocz M, Strupińska A, Roszak S, Prokopowicz M, Koole LH, Kafarski P.

J Mol Model. 2009 Jun;15(6):651-8. doi: 10.1007/s00894-009-0473-6. Epub 2009 Feb 24.

PMID:
19238462
50.

Structural basis for the inhibition of the essential Plasmodium falciparum M1 neutral aminopeptidase.

McGowan S, Porter CJ, Lowther J, Stack CM, Golding SJ, Skinner-Adams TS, Trenholme KR, Teuscher F, Donnelly SM, Grembecka J, Mucha A, Kafarski P, Degori R, Buckle AM, Gardiner DL, Whisstock JC, Dalton JP.

Proc Natl Acad Sci U S A. 2009 Feb 24;106(8):2537-42. doi: 10.1073/pnas.0807398106. Epub 2009 Feb 5.

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