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Items: 10

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1.

Identification of novel PDEδ interacting proteins.

Küchler P, Zimmermann G, Winzker M, Janning P, Waldmann H, Ziegler S.

Bioorg Med Chem. 2018 May 1;26(8):1426-1434. doi: 10.1016/j.bmc.2017.08.033. Epub 2017 Aug 31.

PMID:
28935183
2.

A Specific and Covalent JNK-1 Ligand Selected from an Encoded Self-Assembling Chemical Library.

Zimmermann G, Rieder U, Bajic D, Vanetti S, Chaikuad A, Knapp S, Scheuermann J, Mattarella M, Neri D.

Chemistry. 2017 Jun 16;23(34):8152-8155. doi: 10.1002/chem.201701644. Epub 2017 May 30.

3.

Quantitative PCR is a Valuable Tool to Monitor the Performance of DNA-Encoded Chemical Library Selections.

Li Y, Zimmermann G, Scheuermann J, Neri D.

Chembiochem. 2017 May 4;18(9):848-852. doi: 10.1002/cbic.201600626. Epub 2017 Mar 16.

4.

Hit-Validation Methodologies for Ligands Isolated from DNA-Encoded Chemical Libraries.

Zimmermann G, Li Y, Rieder U, Mattarella M, Neri D, Scheuermann J.

Chembiochem. 2017 May 4;18(9):853-857. doi: 10.1002/cbic.201600637. Epub 2017 Jan 30.

5.

DNA-encoded chemical libraries: foundations and applications in lead discovery.

Zimmermann G, Neri D.

Drug Discov Today. 2016 Nov;21(11):1828-1834. doi: 10.1016/j.drudis.2016.07.013. Epub 2016 Jul 28. Review.

6.

Identification of pyrazolopyridazinones as PDEδ inhibitors.

Papke B, Murarka S, Vogel HA, Martín-Gago P, Kovacevic M, Truxius DC, Fansa EK, Ismail S, Zimmermann G, Heinelt K, Schultz-Fademrecht C, Al Saabi A, Baumann M, Nussbaumer P, Wittinghofer A, Waldmann H, Bastiaens PI.

Nat Commun. 2016 Apr 20;7:11360. doi: 10.1038/ncomms11360.

7.

Small-molecule modulation of Ras signaling.

Spiegel J, Cromm PM, Zimmermann G, Grossmann TN, Waldmann H.

Nat Chem Biol. 2014 Aug;10(8):613-22. doi: 10.1038/nchembio.1560. Epub 2014 Jun 15. Review.

PMID:
24929527
8.

Structure guided design and kinetic analysis of highly potent benzimidazole inhibitors targeting the PDEδ prenyl binding site.

Zimmermann G, Schultz-Fademrecht C, Küchler P, Murarka S, Ismail S, Triola G, Nussbaumer P, Wittinghofer A, Waldmann H.

J Med Chem. 2014 Jun 26;57(12):5435-48. doi: 10.1021/jm500632s. Epub 2014 Jun 11.

PMID:
24884780
9.

Small molecule inhibition of the KRAS-PDEδ interaction impairs oncogenic KRAS signalling.

Zimmermann G, Papke B, Ismail S, Vartak N, Chandra A, Hoffmann M, Hahn SA, Triola G, Wittinghofer A, Bastiaens PI, Waldmann H.

Nature. 2013 May 30;497(7451):638-42. doi: 10.1038/nature12205. Epub 2013 May 22.

PMID:
23698361
10.

Dissociation of the K-Ras4B/PDEδ complex upon contact with lipid membranes: membrane delivery instead of extraction.

Weise K, Kapoor S, Werkmüller A, Möbitz S, Zimmermann G, Triola G, Waldmann H, Winter R.

J Am Chem Soc. 2012 Jul 18;134(28):11503-10. doi: 10.1021/ja305518h. Epub 2012 Jul 10.

PMID:
22721555

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