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Items: 14

1.

Establish an automated flow injection ESI-MS method for the screening of fragment based libraries: Application to Hsp90.

Riccardi Sirtori F, Caronni D, Colombo M, Dalvit C, Paolucci M, Regazzoni L, Visco C, Fogliatto G.

Eur J Pharm Sci. 2015 Aug 30;76:83-94. doi: 10.1016/j.ejps.2015.05.001. Epub 2015 May 4.

PMID:
25952103
2.

Effective immuno-targeting of the IDH1 mutation R132H in a murine model of intracranial glioma.

Pellegatta S, Valletta L, Corbetta C, Patanè M, Zucca I, Riccardi Sirtori F, Bruzzone MG, Fogliatto G, Isacchi A, Pollo B, Finocchiaro G.

Acta Neuropathol Commun. 2015 Jan 21;3:4. doi: 10.1186/s40478-014-0180-0.

3.

Fragment-based hit discovery and structure-based optimization of aminotriazoloquinazolines as novel Hsp90 inhibitors.

Casale E, Amboldi N, Brasca MG, Caronni D, Colombo N, Dalvit C, Felder ER, Fogliatto G, Galvani A, Isacchi A, Polucci P, Riceputi L, Sola F, Visco C, Zuccotto F, Casuscelli F.

Bioorg Med Chem. 2014 Aug 1;22(15):4135-50. doi: 10.1016/j.bmc.2014.05.056. Epub 2014 Jun 14.

PMID:
24980703
4.

Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases.

Casuscelli F, Ardini E, Avanzi N, Casale E, Cervi G, D'Anello M, Donati D, Faiardi D, Ferguson RD, Fogliatto G, Galvani A, Marsiglio A, Mirizzi DG, Montemartini M, Orrenius C, Papeo G, Piutti C, Salom B, Felder ER.

Bioorg Med Chem. 2013 Dec 1;21(23):7364-80. doi: 10.1016/j.bmc.2013.09.054. Epub 2013 Oct 2.

PMID:
24139169
5.

Discovery of NMS-E973 as novel, selective and potent inhibitor of heat shock protein 90 (Hsp90).

Brasca MG, Mantegani S, Amboldi N, Bindi S, Caronni D, Casale E, Ceccarelli W, Colombo N, De Ponti A, Donati D, Ermoli A, Fachin G, Felder ER, Ferguson RD, Fiorelli C, Guanci M, Isacchi A, Pesenti E, Polucci P, Riceputi L, Sola F, Visco C, Zuccotto F, Fogliatto G.

Bioorg Med Chem. 2013 Nov 15;21(22):7047-63. doi: 10.1016/j.bmc.2013.09.018. Epub 2013 Sep 19. Erratum in: Bioorg Med Chem. 2014 Jan 1;22(1):662.

PMID:
24100158
6.

NMS-E973, a novel synthetic inhibitor of Hsp90 with activity against multiple models of drug resistance to targeted agents, including intracranial metastases.

Fogliatto G, Gianellini L, Brasca MG, Casale E, Ballinari D, Ciomei M, Degrassi A, De Ponti A, Germani M, Guanci M, Paolucci M, Polucci P, Russo M, Sola F, Valsasina B, Visco C, Zuccotto F, Donati D, Felder E, Pesenti E, Galvani A, Mantegani S, Isacchi A.

Clin Cancer Res. 2013 Jul 1;19(13):3520-32. doi: 10.1158/1078-0432.CCR-12-3512. Epub 2013 May 14.

7.

Crystal structures of anaplastic lymphoma kinase in complex with ATP competitive inhibitors.

Bossi RT, Saccardo MB, Ardini E, Menichincheri M, Rusconi L, Magnaghi P, Orsini P, Avanzi N, Borgia AL, Nesi M, Bandiera T, Fogliatto G, Bertrand JA.

Biochemistry. 2010 Aug 17;49(32):6813-25. doi: 10.1021/bi1005514.

PMID:
20695522
8.

Reliable high-throughput functional screening with 3-FABS.

Dalvit C, Ardini E, Fogliatto GP, Mongelli N, Veronesi M.

Drug Discov Today. 2004 Jul 15;9(14):595-602. Review.

PMID:
15239978
9.

3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 1. Lead finding.

Pevarello P, Brasca MG, Amici R, Orsini P, Traquandi G, Corti L, Piutti C, Sansonna P, Villa M, Pierce BS, Pulici M, Giordano P, Martina K, Fritzen EL, Nugent RA, Casale E, Cameron A, Ciomei M, Roletto F, Isacchi A, Fogliatto G, Pesenti E, Pastori W, Marsiglio A, Leach KL, Clare PM, Fiorentini F, Varasi M, Vulpetti A, Warpehoski MA.

J Med Chem. 2004 Jun 17;47(13):3367-80.

PMID:
15189033
10.

A general NMR method for rapid, efficient, and reliable biochemical screening.

Dalvit C, Ardini E, Flocco M, Fogliatto GP, Mongelli N, Veronesi M.

J Am Chem Soc. 2003 Nov 26;125(47):14620-5.

PMID:
14624613
11.

WaterLOGSY as a method for primary NMR screening: practical aspects and range of applicability.

Dalvit C, Fogliatto G, Stewart A, Veronesi M, Stockman B.

J Biomol NMR. 2001 Dec;21(4):349-59.

PMID:
11824754
12.

Correction of dyslipoproteinaemia of casein-fed rabbit by FCE 27677, a potent novel ACAT inhibitor.

Chiari A, Lovisolo P, Fogliatto G, Fancelli D, Ghiselli G.

Pharmacol Res. 1996 Mar;33(3):181-9.

PMID:
8880889
13.

Oxidized lipoproteins induce long-lasting inhibition of nitric oxide synthase from a murine endothelioma cell line (bEnd.4).

Fogliatto G, Musanti R, Pirillo A, Ghiselli G.

J Cardiovasc Risk. 1995 Apr;2(2):123-30.

PMID:
7541706
14.

Prolonged in vitro exposure of rat brain slices to adenosine analogues: selective desensitization of adenosine A1 but not A2 receptors.

Abbracchio MP, Fogliatto G, Paoletti AM, Rovati GE, Cattabeni F.

Eur J Pharmacol. 1992 Nov 2;227(3):317-24.

PMID:
1473554

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