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Items: 14

1.

Discovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor-Prolyl Hydroxylase Inhibitor for Anemia.

Ariazi JL, Duffy KJ, Adams DF, Fitch DM, Luo L, Pappalardi M, Biju M, DiFilippo EH, Shaw T, Wiggall K, Erickson-Miller C.

J Pharmacol Exp Ther. 2017 Dec;363(3):336-347. doi: 10.1124/jpet.117.242503. Epub 2017 Sep 19.

PMID:
28928122
2.

Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295.

Qian X, McDonald A, Zhou HJ, Adams ND, Parrish CA, Duffy KJ, Fitch DM, Tedesco R, Ashcraft LW, Yao B, Jiang H, Huang JK, Marin MV, Aroyan CE, Wang J, Ahmed S, Burgess JL, Chaudhari AM, Donatelli CA, Darcy MG, Ridgers LH, Newlander KA, Schmidt SJ, Chai D, Colón M, Zimmerman MN, Lad L, Sakowicz R, Schauer S, Belmont L, Baliga R, Pierce DW, Finer JT, Wang Z, Morgan BP, Morgans DJ Jr, Auger KR, Sung CM, Carson JD, Luo L, Hugger ED, Copeland RA, Sutton D, Elliott JD, Jackson JR, Wood KW, Dhanak D, Bergnes G, Knight SD.

ACS Med Chem Lett. 2010 Jan 19;1(1):30-4. doi: 10.1021/ml900018m. eCollection 2010 Apr 8.

3.

Substituted benzothiadizine inhibitors of Hepatitis C virus polymerase.

Shaw AN, Tedesco R, Bambal R, Chai D, Concha NO, Darcy MG, Dhanak D, Duffy KJ, Fitch DM, Gates A, Johnston VK, Keenan RM, Lin-Goerke J, Liu N, Sarisky RT, Wiggall KJ, Zimmerman MN.

Bioorg Med Chem Lett. 2009 Aug 1;19(15):4350-3. doi: 10.1016/j.bmcl.2009.05.091. Epub 2009 May 28.

PMID:
19515564
4.

Synthesis and biological activity of heteroaryl 3-(1,1-dioxo-2H-(1,2,4)-benzothiadizin-3-yl)-4-hydroxy-2(1H)-quinolinone derivatives as hepatitis C virus NS5B polymerase inhibitors.

Tedesco R, Chai D, Darcy MG, Dhanak D, Fitch DM, Gates A, Johnston VK, Keenan RM, Lin-Goerke J, Sarisky RT, Shaw AN, Valko KL, Wiggall KJ, Zimmerman MN, Duffy KJ.

Bioorg Med Chem Lett. 2009 Aug 1;19(15):4354-8. doi: 10.1016/j.bmcl.2009.05.080. Epub 2009 May 27.

PMID:
19505821
5.

3-(1,1-dioxo-2H-(1,2,4)-benzothiadiazin-3-yl)-4-hydroxy-2(1H)-quinolinones, potent inhibitors of hepatitis C virus RNA-dependent RNA polymerase.

Tedesco R, Shaw AN, Bambal R, Chai D, Concha NO, Darcy MG, Dhanak D, Fitch DM, Gates A, Gerhardt WG, Halegoua DL, Han C, Hofmann GA, Johnston VK, Kaura AC, Liu N, Keenan RM, Lin-Goerke J, Sarisky RT, Wiggall KJ, Zimmerman MN, Duffy KJ.

J Med Chem. 2006 Feb 9;49(3):971-83.

PMID:
16451063
9.

Enantioselective Synthesis of the Elaiophylin Aglycon.

Evans DA, Fitch DM.

J Org Chem. 1997 Feb 7;62(3):454-455. No abstract available.

PMID:
11671433
10.

Some effects of vitamin E deficiency on in vitro cholesterol metabolism.

Eskelson CD, Jacobi HP, Fitch DM.

Physiol Chem Phys. 1973;5(4):319-29. No abstract available.

PMID:
4753996
11.

Meningitis due to Neisseria catarrhalis.

Elston HR, Quigley HJ Jr, Fitch DM.

Nebr Med J. 1970 Jun;55(6):369-71. No abstract available.

PMID:
5524857
12.

Vasculitis with allopurinol therapy.

Jarzobski J, Ferry J, Wombolt D, Fitch DM, Egan JD.

Am Heart J. 1970 Jan;79(1):116-21. No abstract available.

PMID:
5410273
13.

A distinctive myocardiopathy occurring in Omaha, Nebraska: pathological aspects.

Grinvalsky HT, Fitch DM.

Ann N Y Acad Sci. 1969 Jan 31;156(1):544-65. No abstract available.

PMID:
4110944
14.

DETERMINATION OF POTENTIAL PATHOGENICITY OF STAPHYLOCOCCI.

ELSTON HR, FITCH DM.

Am J Clin Pathol. 1964 Oct;42:346-8. No abstract available.

PMID:
14237391

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