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Items: 9

1.

Bioavailability, Biotransformation, and Excretion of the Covalent Bruton Tyrosine Kinase Inhibitor Acalabrutinib in Rats, Dogs, and Humans.

Podoll T, Pearson PG, Evarts J, Ingallinera T, Bibikova E, Sun H, Gohdes M, Cardinal K, Sanghvi M, Slatter JG.

Drug Metab Dispos. 2019 Feb;47(2):145-154. doi: 10.1124/dmd.118.084459. Epub 2018 Nov 15.

PMID:
30442651
2.

Discovery of a Phosphoinositide 3-Kinase (PI3K) β/δ Inhibitor for the Treatment of Phosphatase and Tensin Homolog (PTEN) Deficient Tumors: Building PI3Kβ Potency in a PI3Kδ-Selective Template by Targeting Nonconserved Asp856.

Perreault S, Chandrasekhar J, Cui ZH, Evarts J, Hao J, Kaplan JA, Kashishian A, Keegan KS, Kenney T, Koditek D, Lad L, Lepist EI, McGrath ME, Patel L, Phillips B, Therrien J, Treiberg J, Yahiaoui A, Phillips G.

J Med Chem. 2017 Feb 23;60(4):1555-1567. doi: 10.1021/acs.jmedchem.6b01821. Epub 2017 Feb 7.

PMID:
28106991
3.

Discovery of Orally Efficacious Phosphoinositide 3-Kinase δ Inhibitors with Improved Metabolic Stability.

Patel L, Chandrasekhar J, Evarts J, Forseth K, Haran AC, Ip C, Kashishian A, Kim M, Koditek D, Koppenol S, Lad L, Lepist EI, McGrath ME, Perreault S, Puri KD, Villaseñor AG, Somoza JR, Steiner BH, Therrien J, Treiberg J, Phillips G.

J Med Chem. 2016 Oct 3. [Epub ahead of print]

PMID:
27660855
4.

2,4,6-Triaminopyrimidine as a Novel Hinge Binder in a Series of PI3Kδ Selective Inhibitors.

Patel L, Chandrasekhar J, Evarts J, Haran AC, Ip C, Kaplan JA, Kim M, Koditek D, Lad L, Lepist EI, McGrath ME, Novikov N, Perreault S, Puri KD, Somoza JR, Steiner BH, Stevens KL, Therrien J, Treiberg J, Villaseñor AG, Yeung A, Phillips G.

J Med Chem. 2016 Apr 14;59(7):3532-48. doi: 10.1021/acs.jmedchem.6b00213. Epub 2016 Mar 29.

PMID:
26980109
5.

Accuracy of EMS Trauma Transport Destination Plans in North Carolina.

Moss C, Cowden CS, Atterton LM, Arasaratnam MH, Fernandez AR, Evarts JS, Barrier B, Lerner EB, Mann NC, Lohmeier C, Shofer FS, Brice JH.

Prehosp Emerg Care. 2015 January-March;19(1):53-60. Epub 2014 May 30.

PMID:
24878396
6.

A morphological and immunohistochemical comparison of mammary tissues from the short-tailed fruit bat (Carollia perspicillata) and the mouse.

Evarts JL, Rasweiler JJ 4th, Behringer RR, Hennighausen L, Robinson GW.

Biol Reprod. 2004 Jun;70(6):1573-9. Epub 2004 Jan 28.

PMID:
14749297
7.
8.

Syntheses of highly substituted enantiopure C6 and C7 enones(1).

Evarts J, Torres E, Fuchs PL.

J Am Chem Soc. 2002 Sep 18;124(37):11093-101.

PMID:
12224957
9.

Cyclic AMP-binding proteins in human blood platelets detected by photoaffinity labelling.

Chambers DA, Nachman RL, Evarts J, Kinoshita T.

Biochim Biophys Acta. 1982 Nov 24;719(2):208-14.

PMID:
6295503

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