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Items: 33

1.

Tryptophan Fluorescence Quenching in β-Lactam-Interacting Proteins Is Modulated by the Structure of Intermediates and Final Products of the Acylation Reaction.

Triboulet S, Edoo Z, Compain F, Ourghanlian C, Dupuis A, Dubée V, Sutterlin L, Atze H, Etheve-Quelquejeu M, Hugonnet JE, Arthur M.

ACS Infect Dis. 2019 Jul 12;5(7):1169-1176. doi: 10.1021/acsinfecdis.9b00023. Epub 2019 May 14.

PMID:
31056908
2.

Bisubstrate analogues as structural tools to investigate m6A methyltransferase active sites.

Oerum S, Catala M, Atdjian C, Brachet F, Ponchon L, Barraud P, Iannazzo L, Droogmans L, Braud E, Ethève-Quelquejeu M, Tisné C.

RNA Biol. 2019 Jun;16(6):798-808. doi: 10.1080/15476286.2019.1589360. Epub 2019 Mar 17.

3.

Negative Impact of Carbapenem Methylation on the Reactivity of β-Lactams for Cysteine Acylation as Revealed by Quantum Calculations and Kinetic Analyses.

Bhattacharjee N, Triboulet S, Dubée V, Fonvielle M, Edoo Z, Hugonnet JE, Ethève-Quelquejeu M, Simorre JP, Field MJ, Arthur M, Bougault CM.

Antimicrob Agents Chemother. 2019 Mar 27;63(4). pii: e02039-18. doi: 10.1128/AAC.02039-18. Print 2019 Apr.

4.

Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat.

Atehortua-Martinez LA, Masniere C, Campolongo P, Chasseigneaux S, Callebert J, Zwergel C, Mai A, Laplanche JL, Chen H, Etheve-Quelquejeu M, Mégarbane B, Benturquia N.

J Psychopharmacol. 2019 Mar;33(3):392-405. doi: 10.1177/0269881118822151. Epub 2019 Jan 15.

PMID:
30644332
5.

Synthesis of Lipid-Carbohydrate-Peptidyl-RNA Conjugates to Explore the Limits Imposed by the Substrate Specificity of Cell Wall Enzymes on the Acquisition of Drug Resistance.

Fonvielle M, Bouhss A, Hoareau C, Patin D, Mengin-Lecreulx D, Iannazzo L, Sakkas N, El Sagheer A, Brown T, Ethève-Quelquejeu M, Arthur M.

Chemistry. 2018 Oct 9;24(56):14911-14915. doi: 10.1002/chem.201802360. Epub 2018 Sep 6.

6.

Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships.

Benturquia N, Chevillard L, Poiré C, Roussel O, Cohier C, Declèves X, Laplanche JL, Etheve-Quelquejeu M, Chen H, Mégarbane B.

Psychopharmacology (Berl). 2019 Mar;236(3):891-901. doi: 10.1007/s00213-018-4962-0. Epub 2018 Jul 3.

PMID:
29971461
7.

Structure-Based Design, Synthesis, and Characterization of the First Irreversible Inhibitor of Focal Adhesion Kinase.

Yen-Pon E, Li B, Acebrón-Garcia-de-Eulate M, Tomkiewicz-Raulet C, Dawson J, Lietha D, Frame MC, Coumoul X, Garbay C, Etheve-Quelquejeu M, Chen H.

ACS Chem Biol. 2018 Aug 17;13(8):2067-2073. doi: 10.1021/acschembio.8b00250. Epub 2018 Jun 22.

8.

Synthesis of Avibactam Derivatives and Activity on β-Lactamases and Peptidoglycan Biosynthesis Enzymes of Mycobacteria.

Edoo Z, Iannazzo L, Compain F, Li de la Sierra Gallay I, van Tilbeurgh H, Fonvielle M, Bouchet F, Le Run E, Mainardi JL, Arthur M, Ethève-Quelquejeu M, Hugonnet JE.

Chemistry. 2018 Jun 7;24(32):8081-8086. doi: 10.1002/chem.201800923. Epub 2018 May 14.

PMID:
29601108
9.

Synthesis of tRNA analogues containing a terminal ribose locked in the South conformation to study tRNA-dependent enzymes.

Iannazzo L, Fonvielle M, Braud E, Hřebabecký H, Procházková E, Nencka R, Mathé C, Arthur M, Etheve-Quelquejeu M.

Org Biomol Chem. 2018 Mar 14;16(11):1903-1911. doi: 10.1039/c8ob00019k.

PMID:
29484333
10.

Critical Impact of Peptidoglycan Precursor Amidation on the Activity of l,d-Transpeptidases from Enterococcus faecium and Mycobacterium tuberculosis.

Ngadjeua F, Braud E, Saidjalolov S, Iannazzo L, Schnappinger D, Ehrt S, Hugonnet JE, Mengin-Lecreulx D, Patin D, Ethève-Quelquejeu M, Fonvielle M, Arthur M.

Chemistry. 2018 Apr 17;24(22):5743-5747. doi: 10.1002/chem.201706082. Epub 2018 Feb 21.

PMID:
29389045
11.

Synthesis of novel 1,2,4-triazine scaffold as FAK inhibitors with antitumor activity.

Dao P, Lietha D, Etheve-Quelquejeu M, Garbay C, Chen H.

Bioorg Med Chem Lett. 2017 Apr 15;27(8):1727-1730. doi: 10.1016/j.bmcl.2017.02.072. Epub 2017 Feb 28.

PMID:
28284808
12.

Insights into the interaction of high potency inhibitor IRC-083864 with phosphatase CDC25.

Sarkis M, Miteva MA, Dasso Lang MC, Jaouen M, Sari MA, Galcéra MO, Ethève-Quelquejeu M, Garbay C, Bertho G, Braud E.

Proteins. 2017 Apr;85(4):593-601. doi: 10.1002/prot.25236. Epub 2017 Jan 18.

PMID:
28056492
13.

Electrophilic RNA for Peptidyl-RNA Synthesis and Site-Specific Cross-Linking with tRNA-Binding Enzymes.

Fonvielle M, Sakkas N, Iannazzo L, Le Fournis C, Patin D, Mengin-Lecreulx D, El-Sagheer A, Braud E, Cardon S, Brown T, Arthur M, Etheve-Quelquejeu M.

Angew Chem Int Ed Engl. 2016 Oct 17;55(43):13553-13557. doi: 10.1002/anie.201606843. Epub 2016 Sep 26.

PMID:
27667506
14.

Routes of Synthesis of Carbapenems for Optimizing Both the Inactivation of L,D-Transpeptidase LdtMt1 of Mycobacterium tuberculosis and the Stability toward Hydrolysis by β-Lactamase BlaC.

Iannazzo L, Soroka D, Triboulet S, Fonvielle M, Compain F, Dubée V, Mainardi JL, Hugonnet JE, Braud E, Arthur M, Etheve-Quelquejeu M.

J Med Chem. 2016 Apr 14;59(7):3427-38. doi: 10.1021/acs.jmedchem.6b00096. Epub 2016 Mar 18.

PMID:
26937999
15.

Monitoring of reversible boronic acid-diol interactions by fluorine NMR spectroscopy in aqueous media.

Iannazzo L, Benedetti E, Catala M, Etheve-Quelquejeu M, Tisné C, Micouin L.

Org Biomol Chem. 2015 Sep 7;13(33):8817-21. doi: 10.1039/c5ob01362c. Epub 2015 Jul 30.

PMID:
26224410
16.

Transformation of Plasmacytoid Dendritic Cells into Giant Multinuclear Cells by HIV-1.

Smith N, Etheve-Quelquejeu M, Herbeuval JP.

AIDS Res Hum Retroviruses. 2015 Oct;31(10):959-60. doi: 10.1089/aid.2015.0082. Epub 2015 May 18. No abstract available.

PMID:
26060879
17.

Synthesis of 3'-fluoro-tRNA analogues for exploring non-ribosomal peptide synthesis in bacteria.

Iannazzo L, Laisné G, Fonvielle M, Braud E, Herbeuval JP, Arthur M, Etheve-Quelquejeu M.

Chembiochem. 2015 Feb 9;16(3):477-86. doi: 10.1002/cbic.201402523. Epub 2015 Jan 13.

PMID:
25586254
18.

CD4 and Tumor Necrosis Factor-Related Apoptosis Ligand (TRAIL) localization in HIV-stimulated plasmacytoid dendritic cells by three-dimensional microscopy.

Smith N, Etheve-Quelquejeu M, Herbeuval JP.

AIDS Res Hum Retroviruses. 2014 Dec;30(12):1158-9. doi: 10.1089/aid.2014.0125. No abstract available.

PMID:
25343561
19.

gem-Difluorocarbadisaccharides: restoring the exo-anomeric effect.

Xu B, Unione L, Sardinha J, Wu S, Ethève-Quelquejeu M, Pilar Rauter A, Blériot Y, Zhang Y, Martín-Santamaría S, Díaz D, Jiménez-Barbero J, Sollogoub M.

Angew Chem Int Ed Engl. 2014 Sep 1;53(36):9597-602. doi: 10.1002/anie.201405008. Epub 2014 Jul 15.

PMID:
25044775
20.

Synthesis of 3'-triazoyl-dinucleotides as precursors of stable Phe-tRNA(Phe) and Leu-tRNA(Leu) analogues.

Santarem M, Fonvielle M, Sakkas N, Laisné G, Chemama M, Herbeuval JP, Braud E, Arthur M, Etheve-Quelquejeu M.

Bioorg Med Chem Lett. 2014 Aug 1;24(15):3231-3. doi: 10.1016/j.bmcl.2014.06.027. Epub 2014 Jun 19.

PMID:
24986659
21.

Synthesis and biological evaluation of non-isomerizable analogues of Ala-tRNA(Ala).

Mellal D, Fonvielle M, Santarem M, Chemama M, Schneider Y, Iannazzo L, Braud E, Arthur M, Etheve-Quelquejeu M.

Org Biomol Chem. 2013 Sep 28;11(36):6161-9. doi: 10.1039/c3ob41206g.

PMID:
23925523
22.

Kinetic features of L,D-transpeptidase inactivation critical for β-lactam antibacterial activity.

Triboulet S, Dubée V, Lecoq L, Bougault C, Mainardi JL, Rice LB, Ethève-Quelquejeu M, Gutmann L, Marie A, Dubost L, Hugonnet JE, Simorre JP, Arthur M.

PLoS One. 2013 Jul 4;8(7):e67831. doi: 10.1371/journal.pone.0067831. Print 2013.

23.

The structure of FemX(Wv) in complex with a peptidyl-RNA conjugate: mechanism of aminoacyl transfer from Ala-tRNA(Ala) to peptidoglycan precursors.

Fonvielle M, Li de La Sierra-Gallay I, El-Sagheer AH, Lecerf M, Patin D, Mellal D, Mayer C, Blanot D, Gale N, Brown T, van Tilbeurgh H, Ethève-Quelquejeu M, Arthur M.

Angew Chem Int Ed Engl. 2013 Jul 8;52(28):7278-81. doi: 10.1002/anie.201301411. Epub 2013 Jun 6. No abstract available.

PMID:
23744707
24.

Fluoro-C-glycosides and fluoro-carbasugars, hydrolytically stable and synthetically challenging glycomimetics.

Leclerc E, Pannecoucke X, Ethève-Quelquejeu M, Sollogoub M.

Chem Soc Rev. 2013 May 21;42(10):4270-83. doi: 10.1039/c2cs35403a. Epub 2012 Dec 4. Review.

PMID:
23212149
25.

Efficient access to peptidyl-RNA conjugates for picomolar inhibition of non-ribosomal FemX(Wv) aminoacyl transferase.

Fonvielle M, Mellal D, Patin D, Lecerf M, Blanot D, Bouhss A, Santarem M, Mengin-Lecreulx D, Sollogoub M, Arthur M, Ethève-Quelquejeu M.

Chemistry. 2013 Jan 21;19(4):1357-63. doi: 10.1002/chem.201201999. Epub 2012 Nov 29.

PMID:
23197408
26.

Inactivation of Mycobacterium tuberculosis l,d-transpeptidase LdtMt₁ by carbapenems and cephalosporins.

Dubée V, Triboulet S, Mainardi JL, Ethève-Quelquejeu M, Gutmann L, Marie A, Dubost L, Hugonnet JE, Arthur M.

Antimicrob Agents Chemother. 2012 Aug;56(8):4189-95. doi: 10.1128/AAC.00665-12. Epub 2012 May 21.

27.

Kinetic analysis of Enterococcus faecium L,D-transpeptidase inactivation by carbapenems.

Dubée V, Arthur M, Fief H, Triboulet S, Mainardi JL, Gutmann L, Sollogoub M, Rice LB, Ethève-Quelquejeu M, Hugonnet JE.

Antimicrob Agents Chemother. 2012 Jun;56(6):3409-12. doi: 10.1128/AAC.06398-11. Epub 2012 Mar 26.

28.

Synthesis of stable aminoacyl-tRNA analogs.

Chemama M, Fonvielle M, Lecerf M, Mellal D, Fief H, Arthur M, Etheve-Quelquejeu M.

Curr Protoc Nucleic Acid Chem. 2011 Mar;Chapter 4:Unit 4.44. doi: 10.1002/0471142700.nc0444s44.

PMID:
21400704
29.

Decoding the logic of the tRNA regiospecificity of nonribosomal FemX(Wv) aminoacyl transferase.

Fonvielle M, Chemama M, Lecerf M, Villet R, Busca P, Bouhss A, Ethève-Quelquejeu M, Arthur M.

Angew Chem Int Ed Engl. 2010 Jul 12;49(30):5115-9. doi: 10.1002/anie.201001473. No abstract available.

PMID:
20572225
30.

Aminoacyl-tRNA recognition by the FemXWv transferase for bacterial cell wall synthesis.

Fonvielle M, Chemama M, Villet R, Lecerf M, Bouhss A, Valéry JM, Ethève-Quelquejeu M, Arthur M.

Nucleic Acids Res. 2009 Apr;37(5):1589-601. doi: 10.1093/nar/gkn1039. Epub 2009 Jan 16.

31.

Synthesis of stable aminoacyl-tRNA analogues containing triazole as a bioisoster of esters.

Chemama M, Fonvielle M, Arthur M, Valéry JM, Etheve-Quelquejeu M.

Chemistry. 2009;15(8):1929-38. doi: 10.1002/chem.200801563.

PMID:
19035586
32.

Idiosyncratic features in tRNAs participating in bacterial cell wall synthesis.

Villet R, Fonvielle M, Busca P, Chemama M, Maillard AP, Hugonnet JE, Dubost L, Marie A, Josseaume N, Mesnage S, Mayer C, Valéry JM, Ethève-Quelquejeu M, Arthur M.

Nucleic Acids Res. 2007;35(20):6870-83. Epub 2007 Oct 11.

33.

Stable analogues of aminoacyl-tRNA for inhibition of an essential step of bacterial cell-wall synthesis.

Chemama M, Fonvielle M, Villet R, Arthur M, Valéry JM, Etheve-Quelquejeu M.

J Am Chem Soc. 2007 Oct 24;129(42):12642-3. Epub 2007 Oct 2. No abstract available. Erratum in: J Am Chem Soc. 2008 Mar 26;130(12):4203.

PMID:
17910455

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