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Items: 24

1.

Inhibition of CPAP-tubulin interaction prevents proliferation of centrosome-amplified cancer cells.

Mariappan A, Soni K, Schorpp K, Zhao F, Minakar A, Zheng X, Mandad S, Macheleidt I, Ramani A, Kubelka T, Dawidowski M, Golfmann K, Wason A, Yang C, Simons J, Schmalz HG, Hyman AA, Aneja R, Ullrich R, Urlaub H, Odenthal M, Büttner R, Li H, Sattler M, Hadian K, Gopalakrishnan J.

EMBO J. 2019 Jan 15;38(2). pii: e99876. doi: 10.15252/embj.201899876. Epub 2018 Dec 10.

2.

Synthesis and biological investigations of 3β-aminotropane arylamide derivatives with atypical antipsychotic profile.

Stefanowicz J, Słowiński T, Wróbel MZ, Ślifirski G, Dawidowski M, Stefanowicz Z, Jastrzębska-Więsek M, Partyka A, Wesołowska A, Turło J.

Med Chem Res. 2018;27(8):1906-1928. doi: 10.1007/s00044-018-2203-z. Epub 2018 Jun 22.

3.

Selenized polysaccharides - Biosynthesis and structural analysis.

Malinowska E, Klimaszewska M, Strączek T, Schneider K, Kapusta C, Podsadni P, Łapienis G, Dawidowski M, Kleps J, Górska S, Pisklak DM, Turło J.

Carbohydr Polym. 2018 Oct 15;198:407-417. doi: 10.1016/j.carbpol.2018.06.057. Epub 2018 Jun 15.

PMID:
30093016
4.

Structural basis for ADP-dependent glucokinase inhibition by 8-bromo-substituted adenosine nucleotide.

Grudnik P, Kamiński MM, Rembacz KP, Kuśka K, Madej M, Potempa J, Dawidowski M, Dubin G.

J Biol Chem. 2018 Jul 13;293(28):11088-11099. doi: 10.1074/jbc.RA117.001562. Epub 2018 May 21.

PMID:
29784881
5.

Selective Cytotoxic Activity of Se-Methyl-Seleno-L-Cysteine- and Se-Polysaccharide-Containing Extracts from Shiitake Medicinal Mushroom, Lentinus edodes (Agaricomycetes).

Klimaszewska M, Górska S, Dawidowski M, Podsadni P, Szczepanska A, Orzechowska E, Kurpios-Piec D, Grosicka-Maciag E, Rahden-Staroń I, Turło J.

Int J Med Mushrooms. 2017;19(8):709-716. doi: 10.1615/IntJMedMushrooms.2017021250.

PMID:
29199570
6.

Inhibitors of glycosomal protein import provide new leads against trypanosomiasis.

Kalel VC, Emmanouilidis L, Dawidowski M, Schliebs W, Sattler M, Popowicz GM, Erdmann R.

Microb Cell. 2017 Jul 3;4(7):229-232. doi: 10.15698/mic2017.07.581.

7.

Inhibitors of PEX14 disrupt protein import into glycosomes and kill Trypanosoma parasites.

Dawidowski M, Emmanouilidis L, Kalel VC, Tripsianes K, Schorpp K, Hadian K, Kaiser M, Mäser P, Kolonko M, Tanghe S, Rodriguez A, Schliebs W, Erdmann R, Sattler M, Popowicz GM.

Science. 2017 Mar 31;355(6332):1416-1420. doi: 10.1126/science.aal1807.

PMID:
28360328
8.

Comparison of enzymatic properties and small molecule inhibition of γ-glutamyltranspeptidases from pathogenic and commensal bacteria.

Bolz C, Bach NC, Meyer H, Müller G, Dawidowski M, Popowicz G, Sieber SA, Skerra A, Gerhard M.

Biol Chem. 2017 Mar;398(3):341-357. doi: 10.1515/hsz-2016-0198.

PMID:
27636829
9.

Biosynthesis of Se-methyl-seleno-l-cysteine in Basidiomycetes fungus Lentinula edodes (Berk.) Pegler.

Klimaszewska M, Górska S, Dawidowski M, Podsadni P, Turło J.

Springerplus. 2016 Jun 16;5(1):733. doi: 10.1186/s40064-016-2498-5. eCollection 2016.

10.

Antinociceptive activity of intraperitoneally administered novel and potent anticonvulsive compound, CY-PROLL-SS, in animal neuropathic pain models.

Bujalska-Zadrożny M, Kogut E, de Cordé A, Dawidowski M, Kleczkowska P.

Pharmacol Rep. 2016 Jun;68(3):601-7. doi: 10.1016/j.pharep.2016.01.001. Epub 2016 Jan 21.

PMID:
26977820
11.

Characterization of Disopyramide derivative ADD424042 as a non-cardiotoxic neuronal sodium channel blocker with broad-spectrum anticonvulsant activity in rodent seizure models.

Król M, Ufnal M, Szulczyk B, Podsadni P, Drapała A, Turło J, Dawidowski M.

Eur J Pharm Sci. 2016 Jan 1;81:42-51. doi: 10.1016/j.ejps.2015.10.002. Epub 2015 Oct 9.

PMID:
26441377
12.

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT(1A) activity. Part 5.

Gomółka A, Ciesielska A, Wróbel MZ, Chodkowski A, Kleps J, Dawidowski M, Siwek A, Wolak M, Stachowicz K, Sławińska A, Nowak G, Satała G, Bojarski AJ, Belka M, Ulenberg S, Bączek T, Skowronek P, Turło J, Herold F.

Eur J Med Chem. 2015 Jun 15;98:221-36. doi: 10.1016/j.ejmech.2015.05.003. Epub 2015 May 9.

PMID:
26043160
13.

Synthesis of new perhydropyrrolo[1,2-a]pyrazine derivatives and their evaluation in animal models of epilepsy.

Dawidowski M, Lewandowski W, Turło J.

Molecules. 2014 Oct 7;19(10):15955-81. doi: 10.3390/molecules191015955.

14.

Novel fluorinated pyrrolo[1,2-a]pyrazine-2,6-dione derivatives: synthesis and anticonvulsant evaluation in animal models of epilepsy.

Dawidowski M, Chońska J, Mika W, Turło J.

Bioorg Med Chem. 2014 Oct 1;22(19):5410-27. doi: 10.1016/j.bmc.2014.07.042. Epub 2014 Aug 4.

PMID:
25150088
15.

Multicomponent synthesis and anticonvulsant activity of monocyclic 2,6-diketopiperazine derivatives.

Dawidowski M, Turło J.

Med Chem Res. 2014;23:2007-2018. Epub 2013 Oct 1.

16.

Expanding the substrate scope of Ugi five-center, four-component reaction U-5C-4CR): ketones as coupling partners for secondary amino acids.

Dawidowski M, Sobczak S, Wilczek M, Kulesza A, Turło J.

Mol Divers. 2014 Feb;18(1):61-77. doi: 10.1007/s11030-013-9488-0. Epub 2013 Oct 24.

17.

Structure-activity relationships of the aromatic site in novel anticonvulsant pyrrolo[1,2-a]pyrazine derivatives.

Dawidowski M, Wilczek M, Kubica K, Skolmowski M, Turło J.

Bioorg Med Chem Lett. 2013 Nov 15;23(22):6106-10. doi: 10.1016/j.bmcl.2013.09.022. Epub 2013 Sep 17.

PMID:
24095092
18.

Enhancement of tacrolimus productivity in Streptomyces tsukubaensis by the use of novel precursors for biosynthesis.

Turło J, Gajzlerska W, Klimaszewska M, Król M, Dawidowski M, Gutkowska B.

Enzyme Microb Technol. 2012 Dec 10;51(6-7):388-95. doi: 10.1016/j.enzmictec.2012.08.008. Epub 2012 Aug 30.

PMID:
23040396
19.

Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 2: Perhydropyrido[1,2-a]pyrazines.

Dawidowski M, Herold F, Chodkowski A, Kleps J.

Eur J Med Chem. 2012 Feb;48:347-53. doi: 10.1016/j.ejmech.2011.11.032. Epub 2011 Nov 26.

PMID:
22178094
20.

Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 1: perhydropyrrole[1,2-a]pyrazines.

Dawidowski M, Herold F, Chodkowski A, Kleps J, Szulczyk P, Wilczek M.

Eur J Med Chem. 2011 Oct;46(10):4859-69. doi: 10.1016/j.ejmech.2011.07.027. Epub 2011 Jul 22.

PMID:
21862182
21.

Synthesis and biological investigation of potential atypical antipsychotics with a tropane core. Part 1.

Słowiński T, Stefanowicz J, Dawidowski M, Kleps J, Czuczwar S, Andres-Mach M, Łuszczki JJ, Nowak G, Stachowicz K, Szewczyk B, Sławińska A, Mazurek AP, Mazurek A, Pluciński F, Wolska I, Herold F.

Eur J Med Chem. 2011 Sep;46(9):4474-88. doi: 10.1016/j.ejmech.2011.07.022. Epub 2011 Jul 26.

PMID:
21816515
22.

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT(1A) activity. part 3.

Herold F, Chodkowski A, Izbicki Ł, Turło J, Dawidowski M, Kleps J, Nowak G, Stachowicz K, Dybała M, Siwek A, Mazurek AP, Mazurek A, Pluciński F.

Eur J Med Chem. 2011 Jan;46(1):142-9. doi: 10.1016/j.ejmech.2010.10.026. Epub 2010 Oct 29.

PMID:
21093118
23.

Relationship between selenium accumulation and mycelial cell composition in Lentinula edodes (Berk.) cultures.

Turlo J, Gutkowska B, Herold F, Dawidowski M, Słowiński T, Zobel A.

J Toxicol Environ Health A. 2010;73(17-18):1211-9. doi: 10.1080/15287394.2010.492005.

PMID:
20706946
24.

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity: part 2.

Herold F, Izbicki Ł, Chodkowski A, Dawidowski M, Król M, Kleps J, Turło J, Wolska I, Nowak G, Stachowicz K, Dybała M, Siwek A, Nowak M, Pieniazek E, Jarończyk M, Sylte I, Mazurek AP.

Eur J Med Chem. 2009 Nov;44(11):4702-15. doi: 10.1016/j.ejmech.2009.07.007. Epub 2009 Jul 16.

PMID:
19665823

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