Format
Sort by
Items per page

Send to

Choose Destination

Search results

Items: 15

1.

The discovery of potent blockers of the canonical transient receptor channels, TRPC3 and TRPC6, based on an anilino-thiazole pharmacophore.

Washburn DG, Holt DA, Dodson J, McAtee JJ, Terrell LR, Barton L, Manns S, Waszkiewicz A, Pritchard C, Gillie DJ, Morrow DM, Davenport EA, Lozinskaya IM, Guss J, Basilla JB, Negron LK, Klein M, Willette RN, Fries RE, Jensen TC, Xu X, Schnackenberg CG, Marino JP Jr.

Bioorg Med Chem Lett. 2013 Sep 1;23(17):4979-84. doi: 10.1016/j.bmcl.2013.06.047. Epub 2013 Jun 26.

PMID:
23886683
2.

An orally active TRPV4 channel blocker prevents and resolves pulmonary edema induced by heart failure.

Thorneloe KS, Cheung M, Bao W, Alsaid H, Lenhard S, Jian MY, Costell M, Maniscalco-Hauk K, Krawiec JA, Olzinski A, Gordon E, Lozinskaya I, Elefante L, Qin P, Matasic DS, James C, Tunstead J, Donovan B, Kallal L, Waszkiewicz A, Vaidya K, Davenport EA, Larkin J, Burgert M, Casillas LN, Marquis RW, Ye G, Eidam HS, Goodman KB, Toomey JR, Roethke TJ, Jucker BM, Schnackenberg CG, Townsley MI, Lepore JJ, Willette RN.

Sci Transl Med. 2012 Nov 7;4(159):159ra148. doi: 10.1126/scitranslmed.3004276.

3.

The development of a high-content screening binding assay for the smoothened receptor.

Bee WT, Xie W, Truong M, Will M, Turunen B, Zuercher WJ, McMillan L, Li H, Hornberger KR, Davenport EA, Ames RS, Kallal LA.

J Biomol Screen. 2012 Aug;17(7):900-11. doi: 10.1177/1087057112447872. Epub 2012 May 29.

PMID:
22644265
4.

Benzofuran-substituted urea derivatives as novel P2Y(1) receptor antagonists.

Thalji RK, Aiyar N, Davenport EA, Erhardt JA, Kallal LA, Morrow DM, Senadhi S, Burns-Kurtis CL, Marino JP Jr.

Bioorg Med Chem Lett. 2010 Jul 15;20(14):4104-7. doi: 10.1016/j.bmcl.2010.05.072. Epub 2010 Jun 9.

PMID:
20542694
5.

Development of a high-throughput cell-based assay for superoxide production in HL-60 cells.

Seitz PM, Cooper R, Gatto GJ Jr, Ramon F, Sweitzer TD, Johns DG, Davenport EA, Ames RS, Kallal LA.

J Biomol Screen. 2010 Apr;15(4):388-97. doi: 10.1177/1087057109359687. Epub 2010 Mar 12.

PMID:
20228280
6.

BacMam: versatile gene delivery technology for GPCR assays.

Davenport EA, Nuthulaganti P, Ames RS.

Methods Mol Biol. 2009;552:199-211. doi: 10.1007/978-1-60327-317-6_14.

PMID:
19513651
7.

Evidence for allosteric interactions of antagonist binding to the smoothened receptor.

Rominger CM, Bee WL, Copeland RA, Davenport EA, Gilmartin A, Gontarek R, Hornberger KR, Kallal LA, Lai Z, Lawrie K, Lu Q, McMillan L, Truong M, Tummino PJ, Turunen B, Will M, Zuercher WJ, Rominger DH.

J Pharmacol Exp Ther. 2009 Jun;329(3):995-1005. doi: 10.1124/jpet.109.152090. Epub 2009 Mar 20. Erratum in: J Pharmacol Exp Ther. 2010 Feb;332(2):690.

PMID:
19304771
8.

Tetrahydro-4-quinolinamines identified as novel P2Y(1) receptor antagonists.

Morales-Ramos AI, Mecom JS, Kiesow TJ, Graybill TL, Brown GD, Aiyar NV, Davenport EA, Kallal LA, Knapp-Reed BA, Li P, Londregan AT, Morrow DM, Senadhi S, Thalji RK, Zhao S, Burns-Kurtis CL, Marino JP Jr.

Bioorg Med Chem Lett. 2008 Dec 1;18(23):6222-6. doi: 10.1016/j.bmcl.2008.09.102. Epub 2008 Oct 2.

PMID:
18926700
9.

AMTB, a TRPM8 channel blocker: evidence in rats for activity in overactive bladder and painful bladder syndrome.

Lashinger ES, Steiginga MS, Hieble JP, Leon LA, Gardner SD, Nagilla R, Davenport EA, Hoffman BE, Laping NJ, Su X.

Am J Physiol Renal Physiol. 2008 Sep;295(3):F803-10. doi: 10.1152/ajprenal.90269.2008. Epub 2008 Jun 18.

10.

Type I collagen gel modulates extracellular matrix synthesis and deposition by tracheal epithelial cells.

Davenport EA, Nettesheim P.

Exp Cell Res. 1996 Feb 25;223(1):155-62.

PMID:
8635488
11.

Regulation of mucociliary differentiation of rat tracheal epithelial cells by type I collagen gel substratum.

Davenport EA, Nettesheim P.

Am J Respir Cell Mol Biol. 1996 Jan;14(1):19-26.

PMID:
8534482
12.

Basal levels of max are sufficient for the cotransformation of C3H10T1/2 cells by ras and myc.

Davenport EA, Taparowsky EJ.

Exp Cell Res. 1992 Oct;202(2):532-40.

PMID:
1397104
13.
14.

Cooperation of oncogenes in the multistep transformation of established fibroblasts in culture.

Davenport EA, Drobes BL, Menke SL, Vaidya TB, Taparowsky EJ.

Anticancer Res. 1988 Sep-Oct;8(5A):959-69.

PMID:
2845855
15.

[Effect of antihistamines in the evolution of experimental glomerulonephritis].

DAVENPORT EA, SAFIAN J.

Folha Med. 1951 Apr 25;32(8):58-60. Undetermined Language. No abstract available.

PMID:
14849649

Supplemental Content

Loading ...
Support Center