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Items: 28

1.

Mass spectral databases for metabolomics: How to build a consistently annotated mass spectral database from pure reference compounds analyzed under electrospray ionization conditions?

Damont A, Olivier MF, Warnet A, Lyan B, Pujos-Guillot E, Jamin EL, Debrauwer L, Bernillon S, Junot C, Tabet JC, Fenaille F.

J Mass Spectrom. 2019 May 13. doi: 10.1002/jms.4372. [Epub ahead of print]

PMID:
31083780
2.

Experimental evidence that electrospray-produced sodiated lysophosphatidyl ester structures exist essentially as protonated salts.

Colsch B, Damont A, Junot C, Fenaille F, Tabet JC.

Eur J Mass Spectrom (Chichester). 2019 Jun;25(3):333-338. doi: 10.1177/1469066719838924. Epub 2019 Mar 25.

PMID:
30909743
3.

Identification of new molecular targets for PET imaging of the microglial anti-inflammatory activation state.

Villa A, Klein B, Janssen B, Pedragosa J, Pepe G, Zinnhardt B, Vugts DJ, Gelosa P, Sironi L, Beaino W, Damont A, Dollé F, Jego B, Winkeler A, Ory D, Solin O, Vercouillie J, Funke U, Laner-Plamberger S, Blomster LV, Christophersen P, Vegeto E, Aigner L, Jacobs A, Planas AM, Maggi A, Windhorst AD.

Theranostics. 2018 Oct 27;8(19):5400-5418. doi: 10.7150/thno.25572. eCollection 2018.

4.

[18F]F-DPA for the detection of activated microglia in a mouse model of Alzheimer's disease.

Keller T, López-Picón FR, Krzyczmonik A, Forsback S, Kirjavainen AK, Takkinen JS, Alzghool O, Rajander J, Teperi S, Cacheux F, Damont A, Dollé F, Rinne JO, Solin O, Haaparanta-Solin M.

Nucl Med Biol. 2018 Dec;67:1-9. doi: 10.1016/j.nucmedbio.2018.09.001. Epub 2018 Sep 26.

5.

From Structure-Activity Relationships on Thiazole Derivatives to the In Vivo Evaluation of a New Radiotracer for Cannabinoid Subtype 2 PET Imaging.

Caillé F, Cacheux F, Peyronneau MA, Jego B, Jaumain E, Pottier G, Ullmer C, Grether U, Winkeler A, Dollé F, Damont A, Kuhnast B.

Mol Pharm. 2017 Nov 6;14(11):4064-4078. doi: 10.1021/acs.molpharmaceut.7b00746. Epub 2017 Oct 18.

PMID:
28968497
6.

Avidin/Biotin Bioinspired Platform for Dual In Vivo 18F-PET/NIRF Molecular Imaging.

Damont A, Boisgard R, Dollé F, Hollocou M, Kuhnast B.

Bioconjug Chem. 2017 Oct 18;28(10):2524-2529. doi: 10.1021/acs.bioconjchem.7b00536. Epub 2017 Sep 26.

PMID:
28931274
7.

Neuroprotective effect of the alpha 7 nicotinic receptor agonist PHA 543613 in an in vivo excitotoxic adult rat model.

Foucault-Fruchard L, Doméné A, Page G, Windsor M, Emond P, Rodrigues N, Dollé F, Damont A, Buron F, Routier S, Chalon S, Antier D.

Neuroscience. 2017 Jul 25;356:52-63. doi: 10.1016/j.neuroscience.2017.05.019. Epub 2017 May 18.

PMID:
28527955
8.

Radiosynthesis and Preclinical Evaluation of [18F]F-DPA, A Novel Pyrazolo[1,5a]pyrimidine Acetamide TSPO Radioligand, in Healthy Sprague Dawley Rats.

Keller T, Krzyczmonik A, Forsback S, Picón FRL, Kirjavainen AK, Takkinen J, Rajander J, Cacheux F, Damont A, Dollé F, Rinne JO, Haaparanta-Solin M, Solin O.

Mol Imaging Biol. 2017 Oct;19(5):736-745. doi: 10.1007/s11307-016-1040-z.

9.

Synthesis and in vitro characterization of novel fluorinated derivatives of the translocator protein 18 kDa ligand CfO-DPA-714.

Cacheux F, Médran-Navarrete V, Dollé F, Marguet F, Puech F, Damont A.

Eur J Med Chem. 2017 Jan 5;125:346-359. doi: 10.1016/j.ejmech.2016.09.025. Epub 2016 Sep 9.

PMID:
27688189
10.

Imaging the impact of cyclosporin A and dipyridamole on P-glycoprotein (ABCB1) function at the blood-brain barrier: A [(11)C]-N-desmethyl-loperamide PET study in nonhuman primates.

Damont A, Goutal S, Auvity S, Valette H, Kuhnast B, Saba W, Tournier N.

Eur J Pharm Sci. 2016 Aug 25;91:98-104. doi: 10.1016/j.ejps.2016.06.005. Epub 2016 Jun 7.

PMID:
27283486
11.

Novel Pyrazolo[1,5-a]pyrimidines as Translocator Protein 18 kDa (TSPO) Ligands: Synthesis, in Vitro Biological Evaluation, [(18)F]-Labeling, and in Vivo Neuroinflammation PET Images.

Damont A, Médran-Navarrete V, Cacheux F, Kuhnast B, Pottier G, Bernards N, Marguet F, Puech F, Boisgard R, Dollé F.

J Med Chem. 2015 Sep 24;58(18):7449-64. doi: 10.1021/acs.jmedchem.5b00932. Epub 2015 Sep 3.

PMID:
26280386
12.

Synthesis and in vitro characterization of novel fluorinated derivatives of the TSPO 18 kDa ligand SSR180575.

Damont A, Marguet F, Puech F, Dollé F.

Eur J Med Chem. 2015 Aug 28;101:736-45. doi: 10.1016/j.ejmech.2015.07.033. Epub 2015 Jul 17.

PMID:
26218651
13.

Efficient tritiation of the translocator protein (18 kDa) selective ligand DPA-714.

Damont A, Garcia-Argote S, Buisson DA, Rousseau B, Dollé F.

J Labelled Comp Radiopharm. 2015 Jan;58(1):1-6. doi: 10.1002/jlcr.3252.

PMID:
25616229
14.

[18F]DPA-C5yne, a novel fluorine-18-labelled analogue of DPA-714: radiosynthesis and preliminary evaluation as a radiotracer for imaging neuroinflammation with PET.

Médran-Navarrete V, Bernards N, Kuhnast B, Damont A, Pottier G, Peyronneau MA, Kassiou M, Marguet F, Puech F, Boisgard R, Dollé F.

J Labelled Comp Radiopharm. 2014 May 30;57(6):410-8. doi: 10.1002/jlcr.3199. Epub 2014 Apr 24.

PMID:
24764161
15.

Preparation and evaluation of novel pyrazolo[1,5-a]pyrimidine acetamides, closely related to DPA-714, as potent ligands for imaging the TSPO 18kDa with PET.

Médran-Navarrete V, Damont A, Peyronneau MA, Kuhnast B, Bernards N, Pottier G, Marguet F, Puech F, Boisgard R, Dollé F.

Bioorg Med Chem Lett. 2014 Mar 15;24(6):1550-6. doi: 10.1016/j.bmcl.2014.01.080. Epub 2014 Feb 7.

PMID:
24560538
16.

The potential of carbon-11 and fluorine-18 chemistry: illustration through the development of positron emission tomography radioligands targeting the translocator protein 18 kDa.

Damont A, Roeda D, Dollé F.

J Labelled Comp Radiopharm. 2013 Mar-Apr;56(3-4):96-104. doi: 10.1002/jlcr.2992. Review.

PMID:
24285315
17.

Effects of selected OATP and/or ABC transporter inhibitors on the brain and whole-body distribution of glyburide.

Tournier N, Saba W, Cisternino S, Peyronneau MA, Damont A, Goutal S, Dubois A, Dollé F, Scherrmann JM, Valette H, Kuhnast B, Bottlaender M.

AAPS J. 2013 Oct;15(4):1082-90. doi: 10.1208/s12248-013-9514-2. Epub 2013 Aug 2.

18.

Synthesis and characterization of an MRI Gd-based probe designed to target the translocator protein.

Cerutti E, Damont A, Dollé F, Baroni S, Aime S.

Magn Reson Chem. 2013 Feb;51(2):116-22. doi: 10.1002/mrc.3919. Epub 2013 Jan 10.

PMID:
23303709
19.

Metabolism and quantification of [(18)F]DPA-714, a new TSPO positron emission tomography radioligand.

Peyronneau MA, Saba W, Goutal S, Damont A, Dollé F, Kassiou M, Bottlaender M, Valette H.

Drug Metab Dispos. 2013 Jan;41(1):122-31. doi: 10.1124/dmd.112.046342. Epub 2012 Oct 12.

PMID:
23065531
20.

Current paradigm of the 18-kDa translocator protein (TSPO) as a molecular target for PET imaging in neuroinflammation and neurodegenerative diseases.

Ching AS, Kuhnast B, Damont A, Roeda D, Tavitian B, Dollé F.

Insights Imaging. 2012 Feb;3(1):111-9. doi: 10.1007/s13244-011-0128-x. Epub 2011 Oct 16.

21.

[18F]DPA-714, [18F]PBR111 and [18F]FEDAA1106-selective radioligands for imaging TSPO 18 kDa with PET: automated radiosynthesis on a TRACERLAb FX-FN synthesizer and quality controls.

Kuhnast B, Damont A, Hinnen F, Catarina T, Demphel S, Le Helleix S, Coulon C, Goutal S, Gervais P, Dollé F.

Appl Radiat Isot. 2012 Mar;70(3):489-97. doi: 10.1016/j.apradiso.2011.10.015. Epub 2011 Nov 11.

PMID:
22104496
22.

Synthesis and testing of a p-H2 hyperpolarized 13C probe based on the pyrazolo[1,5-a]pyrimidineacetamide DPA-713, an MRI vector to target the peripheral benzodiazepine receptors.

Cerutti E, Viale A, Damont A, Dollé F, Aime S.

Magn Reson Chem. 2011 Dec;49(12):795-800. doi: 10.1002/mrc.2839. Epub 2011 Nov 17.

PMID:
22095873
23.

Synthesis of 6-[¹⁸F]fluoro-PBR28, a novel radiotracer for imaging the TSPO 18 kDa with PET.

Damont A, Boisgard R, Kuhnast B, Lemée F, Raggiri G, Scarf AM, Da Pozzo E, Selleri S, Martini C, Tavitian B, Kassiou M, Dollé F.

Bioorg Med Chem Lett. 2011 Aug 15;21(16):4819-22. doi: 10.1016/j.bmcl.2011.06.048. Epub 2011 Jun 17.

PMID:
21741237
24.

Pyrazolo[1,5-a]pyrimidine acetamides: 4-Phenyl alkyl ether derivatives as potent ligands for the 18 kDa translocator protein (TSPO).

Reynolds A, Hanani R, Hibbs D, Damont A, Da Pozzo E, Selleri S, Dollé F, Martini C, Kassiou M.

Bioorg Med Chem Lett. 2010 Oct 1;20(19):5799-802. doi: 10.1016/j.bmcl.2010.07.135. Epub 2010 Aug 4.

PMID:
20727749
25.

Evaluation of the PBR/TSPO radioligand [(18)F]DPA-714 in a rat model of focal cerebral ischemia.

Martín A, Boisgard R, Thézé B, Van Camp N, Kuhnast B, Damont A, Kassiou M, Dollé F, Tavitian B.

J Cereb Blood Flow Metab. 2010 Jan;30(1):230-41. doi: 10.1038/jcbfm.2009.205. Epub 2009 Sep 30.

26.

18F-ZW-104: a new radioligand for imaging neuronal nicotinic acetylcholine receptors--in vitro binding properties and PET studies in baboons.

Valette H, Xiao Y, Peyronneau MA, Damont A, Kozikowski AP, Wei ZL, Kassiou M, Kellar KJ, Dollé F, Bottlaender M.

J Nucl Med. 2009 Aug;50(8):1349-55. doi: 10.2967/jnumed.108.061374.

27.

Comparative evaluation of the translocator protein radioligands 11C-DPA-713, 18F-DPA-714, and 11C-PK11195 in a rat model of acute neuroinflammation.

Chauveau F, Van Camp N, Dollé F, Kuhnast B, Hinnen F, Damont A, Boutin H, James M, Kassiou M, Tavitian B.

J Nucl Med. 2009 Mar;50(3):468-76. doi: 10.2967/jnumed.108.058669. Epub 2009 Feb 17.

28.

Synthesis of 1'-C-fluoromethyladenosine.

Damont A, Dukhan D, Gosselin G, Peyronnet J, Storer R.

Nucleosides Nucleotides Nucleic Acids. 2007;26(10-12):1431-4.

PMID:
18066799

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