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Items: 12

1.

Parallel medicinal chemistry approaches to selective HDAC1/HDAC2 inhibitor (SHI-1:2) optimization.

Kattar SD, Surdi LM, Zabierek A, Methot JL, Middleton RE, Hughes B, Szewczak AA, Dahlberg WK, Kral AM, Ozerova N, Fleming JC, Wang H, Secrist P, Harsch A, Hamill JE, Cruz JC, Kenific CM, Chenard M, Miller TA, Berk SC, Tempest P.

Bioorg Med Chem Lett. 2009 Feb 15;19(4):1168-72. doi: 10.1016/j.bmcl.2008.12.083. Epub 2008 Dec 25.

PMID:
19138845
2.

Versatile solid-phase synthesis of trisubstituted 1H-pyrido[2,3-d]pyrimidin-4-ones and related heterocycles.

Schell P, Richards MP, Hanson K, Berk SC, Makara GM.

J Comb Chem. 2005 Jan-Feb;7(1):96-8.

PMID:
15638487
3.

Combinatorial synthesis of substituted biaryls and heterocyclic arylamines.

Ma Y, Margarida L, Brookes J, Makara GM, Berk SC.

J Comb Chem. 2004 May-Jun;6(3):426-30.

PMID:
15132604
4.

Recent advances in chemical library synthesis methodology.

Flynn DL, Berk SC, Makara GM.

Curr Opin Drug Discov Devel. 2002 Jul;5(4):580-93. Review.

PMID:
12197316
5.
6.

Combinatorial synthesis of CCR5 antagonists.

Willoughby CA, Berk SC, Rosauer KG, Degrado S, Chapman KT, Gould SL, Springer MS, Malkowitz L, Schleif WA, Hazuda D, Miller M, Kessler J, Danzeisen R, Holmes K, Lineberger J, Carella A, Carver G, Emini EA.

Bioorg Med Chem Lett. 2001 Dec 17;11(24):3137-41.

PMID:
11720860
7.

Titanocene-Catalyzed Reduction of Lactones to Lactols.

Verdaguer X, Hansen MC, Berk SC, Buchwald SL.

J Org Chem. 1997 Nov 28;62(24):8522-8528.

PMID:
11671995
8.

A combinatorial approach toward the discovery of non-peptide, subtype-selective somatostatin receptor ligands.

Berk SC, Rohrer SP, Degrado SJ, Birzin ET, Mosley RT, Hutchins SM, Pasternak A, Schaeffer JM, Underwood DJ, Chapman KT.

J Comb Chem. 1999 Sep-Oct;1(5):388-96.

PMID:
10748735
9.

Development of somatostatin receptor subtype selective agonists through combinatorial chemistry.

Rohrer SP, Berk SC.

Curr Opin Drug Discov Devel. 1999 Jul;2(4):293-303.

PMID:
19649957
10.

Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry.

Rohrer SP, Birzin ET, Mosley RT, Berk SC, Hutchins SM, Shen DM, Xiong Y, Hayes EC, Parmar RM, Foor F, Mitra SW, Degrado SJ, Shu M, Klopp JM, Cai SJ, Blake A, Chan WW, Pasternak A, Yang L, Patchett AA, Smith RG, Chapman KT, Schaeffer JM.

Science. 1998 Oct 23;282(5389):737-40. Erratum in: Science 1998 Nov 27;282(5394):1646.

11.

Synthesis and biological activities of potent peptidomimetics selective for somatostatin receptor subtype 2.

Yang L, Berk SC, Rohrer SP, Mosley RT, Guo L, Underwood DJ, Arison BH, Birzin ET, Hayes EC, Mitra SW, Parmar RM, Cheng K, Wu TJ, Butler BS, Foor F, Pasternak A, Pan Y, Silva M, Freidinger RM, Smith RG, Chapman K, Schaeffer JM, Patchett AA.

Proc Natl Acad Sci U S A. 1998 Sep 1;95(18):10836-41.

12.

A Practical Titanium-Catalyzed Synthesis of Bicyclic Cyclopentenones and Allylic Amines.

Hicks FA, Berk SC, Buchwald SL.

J Org Chem. 1996 Apr 19;61(8):2713-2718.

PMID:
11667103

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