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Items: 1 to 50 of 88

1.

Cu(I)- and Pd(0)-Catalyzed Arylation of Oxadiamines with Fluorinated Halogenobenzenes: Comparison of Efficiency.

Lyakhovich MS, Averin AD, Grigorova OK, Roznyatovsky VA, Maloshitskaya OA, Beletskaya IP.

Molecules. 2020 Feb 28;25(5). pii: E1084. doi: 10.3390/molecules25051084.

2.

Tuning the Luminescent Properties of Ruthenium(II) Amino-1,10-Phenanthroline Complexes by Varying the Position of the Amino Group on the Heterocycle.

Abel AS, Zenkov IS, Averin AD, Cheprakov AV, Bessmertnykh-Lemeune AG, Orlinson BS, Beletskaya IP.

Chempluschem. 2019 May;84(5):498-503. doi: 10.1002/cplu.201900206.

PMID:
31943904
3.

Trifluoroacetaldehyde N-Tosylhydrazone as a Precursor of Trifluorodiazoethane in Reactions of Insertion into the Heteroatom-Hydrogen Bond.

Ostrovskii VS, Beletskaya IP, Titanyuk ID.

Org Lett. 2019 Nov 15;21(22):9080-9083. doi: 10.1021/acs.orglett.9b03471. Epub 2019 Nov 1.

PMID:
31674792
4.

Metal-catalyzed regiodivergent organic reactions.

Nájera C, Beletskaya IP, Yus M.

Chem Soc Rev. 2019 Aug 12;48(16):4515-4618. doi: 10.1039/c8cs00872h. Review.

PMID:
31282495
5.

An alternative approach to study the enzymatic specificities of the CfrBI restriction-modification system.

Zakharova MV, Beletskaya IV, Ibryashkina EM, Solonin AS.

Heliyon. 2019 Jun 8;5(6):e01846. doi: 10.1016/j.heliyon.2019.e01846. eCollection 2019 Jun.

6.

6-Polyamino-substituted quinolines: synthesis and multiple metal (CuII, HgII and ZnII) monitoring in aqueous media.

Abel AS, Averin AD, Cheprakov AV, Roznyatovsky VA, Denat F, Bessmertnykh-Lemeune A, Beletskaya IP.

Org Biomol Chem. 2019 Apr 24;17(17):4243-4260. doi: 10.1039/c9ob00259f.

PMID:
30860543
7.

Towards the 150th Anniversary of the Markovnikov Rule.

Beletskaya IP, Nenajdenko VG.

Angew Chem Int Ed Engl. 2019 Apr 1;58(15):4778-4789. doi: 10.1002/anie.201810035. Epub 2019 Mar 1. Review.

PMID:
30537023
8.

Annulation-Induced Cascade Transformation of 5-Iodo-1,2,3-triazoles to 2-(1-Aminoalkyl)benzoxazoles.

Kotovshchikov YN, Latyshev GV, Navasardyan MA, Erzunov DA, Beletskaya IP, Lukashev NV.

Org Lett. 2018 Aug 3;20(15):4467-4470. doi: 10.1021/acs.orglett.8b01755. Epub 2018 Jul 24.

PMID:
30040429
9.

Stereodivergent Catalysis.

Beletskaya IP, Nájera C, Yus M.

Chem Rev. 2018 May 23;118(10):5080-5200. doi: 10.1021/acs.chemrev.7b00561. Epub 2018 Apr 20.

PMID:
29676895
10.

Direct catalytic arylation of heteroarenes with meso-bromophenyl-substituted porphyrins.

Kiselev AN, Grigorova OK, Averin AD, Syrbu SA, Koifman OI, Beletskaya IP.

Beilstein J Org Chem. 2017 Aug 3;13:1524-1532. doi: 10.3762/bjoc.13.152. eCollection 2017.

11.

Pd- and Cu-catalyzed approaches in the syntheses of new cholane aminoanthraquinone pincer-like ligands.

Lukashev NV, Grabovyi GA, Erzunov DA, Kazantsev AV, Latyshev GV, Averin AD, Beletskaya IP.

Beilstein J Org Chem. 2017 Mar 20;13:564-570. doi: 10.3762/bjoc.13.55. eCollection 2017.

12.

Functional characterization of CFI-402257, a potent and selective Mps1/TTK kinase inhibitor, for the treatment of cancer.

Mason JM, Wei X, Fletcher GC, Kiarash R, Brokx R, Hodgson R, Beletskaya I, Bray MR, Mak TW.

Proc Natl Acad Sci U S A. 2017 Mar 21;114(12):3127-3132. doi: 10.1073/pnas.1700234114. Epub 2017 Mar 7.

13.

Base mediated 1,3-dipolar cycloaddition of α-substituted vinyl phosphonates with diazo compounds for synthesis of 3-pyrazolylphosphonates and 5-pyrazolcarboxylates.

Goulioukina NS, Makukhin NN, Shinkarev ED, Grishin YK, Roznyatovsky VA, Beletskaya IP.

Org Biomol Chem. 2016 Oct 25;14(42):10000-10010.

PMID:
27722648
14.

Design and optimization of (3-aryl-1H-indazol-6-yl)spiro[cyclopropane-1,3'-indolin]-2'-ones as potent PLK4 inhibitors with oral antitumor efficacy.

Li SW, Liu Y, Sampson PB, Patel NK, Forrest BT, Edwards L, Laufer R, Feher M, Ban F, Awrey DE, Hodgson R, Beletskaya I, Mao G, Mason JM, Wei X, Luo X, Kiarash R, Green E, Mak TW, Pan G, Pauls HW.

Bioorg Med Chem Lett. 2016 Oct 1;26(19):4625-4630. doi: 10.1016/j.bmcl.2016.08.063. Epub 2016 Aug 23.

PMID:
27592744
15.

Discovery of Pyrazolo[1,5-a]pyrimidine TTK Inhibitors: CFI-402257 is a Potent, Selective, Bioavailable Anticancer Agent.

Liu Y, Laufer R, Patel NK, Ng G, Sampson PB, Li SW, Lang Y, Feher M, Brokx R, Beletskaya I, Hodgson R, Plotnikova O, Awrey DE, Qiu W, Chirgadze NY, Mason JM, Wei X, Lin DC, Che Y, Kiarash R, Fletcher GC, Mak TW, Bray MR, Pauls HW.

ACS Med Chem Lett. 2016 May 6;7(7):671-5. doi: 10.1021/acsmedchemlett.5b00485. eCollection 2016 Jul 14.

16.

Discovery of 4-(4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)benzamides as novel, highly potent and selective, orally bioavailable inhibitors of Tyrosine Threonine Kinase, TTK.

Laufer R, Li SW, Liu Y, Ng G, Lang Y, Feher M, Brokx R, Beletskaya I, Hodgson R, Mao G, Plotnikova O, Awrey DE, Mason JM, Wei X, Lin DC, Che Y, Kiarash R, Madeira B, Fletcher GC, Mak TW, Bray MR, Pauls HW.

Bioorg Med Chem Lett. 2016 Aug 1;26(15):3562-6. doi: 10.1016/j.bmcl.2016.06.021. Epub 2016 Jun 9.

PMID:
27335255
17.

Excitonic Coupling and Femtosecond Relaxation of Zinc Porphyrin Oligomers Linked with Triazole Bridge: Dynamics and Modeling.

Bukreev A, Mikhailov K, Shelaev I, Gostev F, Polevaya Y, Tyurin V, Beletskaya I, Umansky S, Nadtochenko V.

J Phys Chem A. 2016 Mar 31;120(12):1961-70. doi: 10.1021/acs.jpca.5b11025. Epub 2016 Mar 17.

PMID:
26935579
18.

Is It Easy to Be a Woman in Science?

Beletskaya IP.

Chemistry. 2016 Mar 7;22(11):3531-2. doi: 10.1002/chem.201505051. Epub 2016 Feb 16.

PMID:
26880132
19.

Carbonylmetallates--A Special Family of Nucleophiles in Aromatic and Vinylic Substitution Reactions.

Sazonov PK, Beletskaya IP.

Chemistry. 2016 Mar 7;22(11):3644-53. doi: 10.1002/chem.201504423. Epub 2016 Jan 25. Review.

PMID:
26808811
20.

Cu(I)-catalyzed N,N'-diarylation of natural diamines and polyamines with aryl iodides.

Panchenko SP, Averin AD, Anokhin MV, Maloshitskaya OA, Beletskaya IP.

Beilstein J Org Chem. 2015 Nov 24;11:2297-305. doi: 10.3762/bjoc.11.250. eCollection 2015.

21.

Ditopic Macrocyclic Receptors with a 4,7-Diamino-1,10-phenanthroline Fragment for Multimodal Detection of Toxic Metal Ions.

Abel AS, Mitrofanov AY, Rousselin Y, Denat F, Bessmertnykh-Lemeune A, Averin AD, Beletskaya IP.

Chempluschem. 2016 Jan;81(1):35-39. doi: 10.1002/cplu.201500390. Epub 2015 Oct 16.

PMID:
31968726
22.

Phosphonate derivatives of tetraazamacrocycles as new inhibitors of protein tyrosine phosphatases.

Kobzar OL, Shevchuk MV, Lyashenko AN, Tanchuk VY, Romanenko VD, Kobelev SM, Averin AD, Beletskaya IP, Vovk AI, Kukhar VP.

Org Biomol Chem. 2015 Jul 21;13(27):7437-44. doi: 10.1039/c5ob00713e.

PMID:
26058329
23.

Alkynylation of steroids via Pd-free Sonogashira coupling.

Kotovshchikov YN, Latyshev GV, Lukashev NV, Beletskaya IP.

Org Biomol Chem. 2015 May 21;13(19):5542-55. doi: 10.1039/c5ob00559k.

PMID:
25880697
24.

The Discovery of Orally Bioavailable Tyrosine Threonine Kinase (TTK) Inhibitors: 3-(4-(heterocyclyl)phenyl)-1H-indazole-5-carboxamides as Anticancer Agents.

Liu Y, Lang Y, Patel NK, Ng G, Laufer R, Li SW, Edwards L, Forrest B, Sampson PB, Feher M, Ban F, Awrey DE, Beletskaya I, Mao G, Hodgson R, Plotnikova O, Qiu W, Chirgadze NY, Mason JM, Wei X, Lin DC, Che Y, Kiarash R, Madeira B, Fletcher GC, Mak TW, Bray MR, Pauls HW.

J Med Chem. 2015 Apr 23;58(8):3366-92. doi: 10.1021/jm501740a. Epub 2015 Apr 3.

PMID:
25763473
25.

The discovery of Polo-like kinase 4 inhibitors: identification of (1R,2S).2-(3-((E).4-(((cis).2,6-dimethylmorpholino)methyl)styryl). 1H.indazol-6-yl)-5'-methoxyspiro[cyclopropane-1,3'-indolin]-2'-one (CFI-400945) as a potent, orally active antitumor agent.

Sampson PB, Liu Y, Forrest B, Cumming G, Li SW, Patel NK, Edwards L, Laufer R, Feher M, Ban F, Awrey DE, Mao G, Plotnikova O, Hodgson R, Beletskaya I, Mason JM, Luo X, Nadeem V, Wei X, Kiarash R, Madeira B, Huang P, Mak TW, Pan G, Pauls HW.

J Med Chem. 2015 Jan 8;58(1):147-69.

PMID:
25723005
26.

Synthesis and biological evaluation of furanoallocolchicinoids.

Voitovich YV, Shegravina ES, Sitnikov NS, Faerman VI, Fokin VV, Schmalz HG, Combes S, Allegro D, Barbier P, Beletskaya IP, Svirshchevskaya EV, Fedorov AY.

J Med Chem. 2015 Jan 22;58(2):692-704. doi: 10.1021/jm501678w. Epub 2014 Dec 24.

PMID:
25496412
27.

Exclusive selectivity in the one-pot formation of C-C and C-Se bonds involving Ni-catalyzed alkyne hydroselenation: optimization of the synthetic procedure and a mechanistic study.

Orlov NV, Chistyakov IV, Khemchyan LL, Ananikov VP, Beletskaya IP, Starikova ZA.

J Org Chem. 2014 Dec 19;79(24):12111-21. doi: 10.1021/jo501953f. Epub 2014 Oct 23.

PMID:
25288369
28.

Insights into the binding of PARP inhibitors to the catalytic domain of human tankyrase-2.

Qiu W, Lam R, Voytyuk O, Romanov V, Gordon R, Gebremeskel S, Vodsedalek J, Thompson C, Beletskaya I, Battaile KP, Pai EF, Rottapel R, Chirgadze NY.

Acta Crystallogr D Biol Crystallogr. 2014 Oct;70(Pt 10):2740-53. doi: 10.1107/S1399004714017660. Epub 2014 Sep 27.

29.

A halogenophilic pathway in the reactions of transition metal carbonyl anions with [(η⁶-iodobenzene)Cr(CO)₃].

Sazonov PK, Ivushkin VA, Khrustalev VN, Kolotyrkina NG, Beletskaya IP.

Dalton Trans. 2014 Sep 21;43(35):13392-8. doi: 10.1039/c4dt01363h.

PMID:
25072592
30.

Discovery of inhibitors of the mitotic kinase TTK based on N-(3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-acetamides and carboxamides.

Laufer R, Ng G, Liu Y, Patel NK, Edwards LG, Lang Y, Li SW, Feher M, Awrey DE, Leung G, Beletskaya I, Plotnikova O, Mason JM, Hodgson R, Wei X, Mao G, Luo X, Huang P, Green E, Kiarash R, Lin DC, Harris-Brandts M, Ban F, Nadeem V, Mak TW, Pan GJ, Qiu W, Chirgadze NY, Pauls HW.

Bioorg Med Chem. 2014 Sep 1;22(17):4968-97. doi: 10.1016/j.bmc.2014.06.027. Epub 2014 Jun 23.

PMID:
25043312
31.

Synthesis of novel 1,2,3-triazolyl derivatives of pregnane, androstane and D-homoandrostane. Tandem "click" reaction/Cu-catalyzed D-homo rearrangement.

Kotovshchikov YN, Latyshev GV, Lukashev NV, Beletskaya IP.

Org Biomol Chem. 2014 Jun 14;12(22):3707-20. doi: 10.1039/c4ob00404c. Epub 2014 Apr 30.

PMID:
24781658
32.

Pd-catalyzed amination in the synthesis of a new family of macropolycyclic compounds comprising diazacrown ether moieties.

Yakushev AA, Chernichenko NM, Anokhin MV, Averin AD, Buryak AK, Denat F, Beletskaya IP.

Molecules. 2014 Jan 15;19(1):940-65. doi: 10.3390/molecules19010940.

33.

Palladium-catalyzed amination of meso-(bromophenyl)porphyrins with diamines and azamacrocycles.

Mikhalitsyna EA, Tyurin VS, Khrustalev VN, Lonin IS, Beletskaya IP.

Dalton Trans. 2014 Mar 7;43(9):3563-75. doi: 10.1039/c3dt52685b.

PMID:
24399206
34.
35.

Dualism of Ion-Pairing Effects in Nucleophilic Vinylic Substitution with Transition-Metal Carbonyl Anions.

Sazonov PK, Beletskaya IP.

Chempluschem. 2013 Sep;78(9):1190-1194. doi: 10.1002/cplu.201300171. Epub 2013 Aug 19.

PMID:
31986713
37.

The discovery of PLK4 inhibitors: (E)-3-((1H-Indazol-6-yl)methylene)indolin-2-ones as novel antiproliferative agents.

Laufer R, Forrest B, Li SW, Liu Y, Sampson P, Edwards L, Lang Y, Awrey DE, Mao G, Plotnikova O, Leung G, Hodgson R, Beletskaya I, Mason JM, Luo X, Wei X, Yao Y, Feher M, Ban F, Kiarash R, Green E, Mak TW, Pan G, Pauls HW.

J Med Chem. 2013 Aug 8;56(15):6069-87. doi: 10.1021/jm400380m. Epub 2013 Jul 26.

PMID:
23829549
38.

Opioid receptor selectivity profile change via isosterism for 14-O-substituted naltrexone derivatives.

Zhang Y, Elbegdorj O, Yuan Y, Beletskaya IO, Selley DE.

Bioorg Med Chem Lett. 2013 Jul 1;23(13):3719-22. doi: 10.1016/j.bmcl.2013.05.027. Epub 2013 May 16.

39.

Palladium-catalyzed amination of dichloroquinolines with adamantane-containing amines.

Abel AS, Averin AD, Maloshitskaya OA, Savelyev EN, Orlinson BS, Novakov IA, Beletskaya IP.

Molecules. 2013 Feb 6;18(2):2096-109. doi: 10.3390/molecules18022096.

40.

Radical-chain oxidative addition mechanism for the reaction of an [Re(CO)5]- anion with α-bromostilbene.

Sazonov PK, Ptushkin DS, Khrustalev VN, Kolotyrkina NG, Beletskaya IP.

Dalton Trans. 2013 Mar 28;42(12):4223-32. doi: 10.1039/c2dt32552g.

PMID:
23292281
41.

Design, synthesis, and biological evaluation of 17-cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-[(4'-pyridyl)carboxamido]morphinan derivatives as peripheral selective μ opioid receptor Agents.

Yuan Y, Elbegdorj O, Chen J, Akubathini SK, Zhang F, Stevens DL, Beletskaya IO, Scoggins KL, Zhang Z, Gerk PM, Selley DE, Akbarali HI, Dewey WL, Zhang Y.

J Med Chem. 2012 Nov 26;55(22):10118-29. doi: 10.1021/jm301247n. Epub 2012 Nov 9.

42.

Synthesis, characterization and cation-induced dimerization of new aza-crown ether-appended metalloporphyrins.

Mikhalitsyna EA, Tyurin VS, Zamylatskov IA, Khrustalev VN, Beletskaya IP.

Dalton Trans. 2012 Jul 7;41(25):7624-36. doi: 10.1039/c2dt30123g. Epub 2012 May 18.

PMID:
22610260
43.

Catalytic adaptive recognition of thiol (SH) and selenol (SeH) groups toward synthesis of functionalized vinyl monomers.

Ananikov VP, Orlov NV, Zalesskiy SS, Beletskaya IP, Khrustalev VN, Morokuma K, Musaev DG.

J Am Chem Soc. 2012 Apr 18;134(15):6637-49. doi: 10.1021/ja210596w. Epub 2012 Apr 4.

PMID:
22475174
44.

Catalytic hydrofunctionalization of alkynes through P-H bond addition: the unique role of orientation and properties of the phosphorus group in the insertion step.

Ananikov VP, Makarov AV, Beletskaya IP.

Chemistry. 2011 Nov 4;17(45):12623-30. doi: 10.1002/chem.201101898. Epub 2011 Oct 4.

PMID:
21971879
45.

Rational design of aminoanthraquinones for colorimetric detection of heavy metal ions in aqueous solution.

Ranyuk E, Uglov A, Meyer M, Bessmertnykh Lemeune A, Denat F, Averin A, Beletskaya I, Guilard R.

Dalton Trans. 2011 Oct 28;40(40):10491-502. doi: 10.1039/c1dt10677e. Epub 2011 Aug 9.

PMID:
21811711
46.

Structure selectivity relationship studies of 17-cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-[(4'-pyridyl)carboxamido]morphinan derivatives toward the development of the mu opioid receptor antagonists.

Yuan Y, Elbegdorj O, Chen J, Akubathini SK, Beletskaya IO, Selley DE, Zhang Y.

Bioorg Med Chem Lett. 2011 Sep 15;21(18):5625-9. doi: 10.1016/j.bmcl.2011.06.135. Epub 2011 Jul 18.

47.

Alkyne insertion into the M-P and M-H bonds (M=Pd, Ni, Pt, and Rh): a theoretical mechanistic study of the C-P and C-H bond-formation steps.

Ananikov VP, Beletskaya IP.

Chem Asian J. 2011 Jun 6;6(6):1423-30. doi: 10.1002/asia.201000840. Epub 2011 Apr 7.

PMID:
21480533
48.

Transition-metal-catalyzed C-S, C-Se, and C-Te bond formation via cross-coupling and atom-economic addition reactions.

Beletskaya IP, Ananikov VP.

Chem Rev. 2011 Mar 9;111(3):1596-636. doi: 10.1021/cr100347k. No abstract available.

PMID:
21391564
49.

Preparation of metal "nanosalts" and their application in catalysis: heterogeneous and homogeneous pathways.

Ananikov VP, Beletskaya IP.

Dalton Trans. 2011 Apr 28;40(16):4011-23. doi: 10.1039/c0dt01277g. Epub 2011 Feb 14.

PMID:
21321732
50.

1,4-Diiodo-1,3-dienes: versatile reagents in organic synthesis.

Ananikov VP, Hazipov OV, Beletskaya IP.

Chem Asian J. 2011 Feb 1;6(2):306-23. doi: 10.1002/asia.201000405. Epub 2010 Sep 17. Review.

PMID:
20853391

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