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Items: 19

1.

Pharmacological and functional characterization of novel EP and DP receptor agonists: DP1 receptor mediates penile erection in multiple species.

Brugger N, Kim NN, Araldi GL, Traish AM, Palmer SS.

J Sex Med. 2008 Feb;5(2):344-56. Epub 2007 Nov 28.

PMID:
18047485
2.

Synthesis and evaluation of a gamma-lactam as a highly selective EP2 and EP4 receptor agonist.

Xiao Y, Araldi GL, Zhao Z, Reddy A, Karra S, Brugger N, Fischer D, Palmer E, Bao B, McKenna SD.

Bioorg Med Chem Lett. 2008 Jan 15;18(2):821-4. Epub 2007 Nov 13.

PMID:
18039575
3.

Synthesis and evaluation of novel pyrazolidinone analogs of PGE2 as EP2 and EP4 receptors agonists.

Zhao Z, Araldi GL, Xiao Y, Reddy AP, Liao Y, Karra S, Brugger N, Fischer D, Palmer E.

Bioorg Med Chem Lett. 2007 Dec 1;17(23):6572-5. Epub 2007 Sep 26.

PMID:
17931866
4.

Discovery of novel prostaglandin analogs of PGE2 as potent and selective EP2 and EP4 receptor agonists.

Xiao Y, Araldi GL, Zhao Z, Brugger N, Karra S, Fischer D, Palmer E.

Bioorg Med Chem Lett. 2007 Aug 1;17(15):4323-7. Epub 2007 May 16.

PMID:
17531488
5.

Mixed cocaine agonist/antagonist properties of (+)-methyl 4beta-(4-chlorophenyl)-1-methylpiperidine-3alpha-carboxylate, a piperidine-based analog of cocaine.

Kozikowski AP, Johnson KM, Deschaux O, Bandyopadhyay BC, Araldi GL, Carmona G, Munzar P, Smith MP, Balster RL, Beardsley PM, Tella SR.

J Pharmacol Exp Ther. 2003 Apr;305(1):143-50.

PMID:
12649362
6.

Novel diketopiperazine enhances motor and cognitive recovery after traumatic brain injury in rats and shows neuroprotection in vitro and in vivo.

Faden AI, Knoblach SM, Cernak I, Fan L, Vink R, Araldi GL, Fricke ST, Roth BL, Kozikowski AP.

J Cereb Blood Flow Metab. 2003 Mar;23(3):342-54.

PMID:
12621309
7.

Non-covalent thrombin inhibitors featuring P3-heterocycles with P1-bicyclic arginine surrogates.

Cui JJ, Araldi GL, Reiner JE, Reddy KM, Kemp SJ, Ho JZ, Siev DV, Mamedova L, Gibson TS, Gaudette JA, Minami NK, Anderson SM, Bradbury AE, Nolan TG, Semple JE.

Bioorg Med Chem Lett. 2002 Oct 21;12(20):2925-30.

PMID:
12270176
8.

Non-covalent thrombin inhibitors featuring P(3)-heterocycles with P(1)-monocyclic arginine surrogates.

Reiner JE, Siev DV, Araldi GL, Cui JJ, Ho JZ, Reddy KM, Mamedova L, Vu PH, Lee KS, Minami NK, Gibson TS, Anderson SM, Bradbury AE, Nolan TG, Semple JE.

Bioorg Med Chem Lett. 2002 Apr 22;12(8):1203-8.

PMID:
11934589
9.

Neuroprotective and cognitive enhancing effects of novel small peptides.

Faden AI, Fox G, Fan L, Knoblach S, Araldi GL, Kozikowski AP.

Ann N Y Acad Sci. 1999;890:120. No abstract available.

PMID:
10668419
10.

N-phenylalkyl-substituted tropane analogs of boat conformation with high selectivity for the dopamine versus serotonin transporter.

Prakash KR, Tamiz AP, Araldi GL, Zhang M, Johnson KM, Kozikowski AP.

Bioorg Med Chem Lett. 1999 Dec 6;9(23):3325-8.

PMID:
10612593
11.

Novel TRH analog improves motor and cognitive recovery after traumatic brain injury in rodents.

Faden AI, Fox GB, Fan L, Araldi GL, Qiao L, Wang S, Kozikowski AP.

Am J Physiol. 1999 Oct;277(4):R1196-204. doi: 10.1152/ajpregu.1999.277.4.R1196.

PMID:
10516262
12.

1-amino-APDC, a partial agonist of group II metabotropic glutamate receptors with neuroprotective properties.

Kozikowski AP, Araldi GL, Tückmantel W, Pshenichkin S, Surina E, Wroblewski JT.

Bioorg Med Chem Lett. 1999 Jun 21;9(12):1721-6.

PMID:
10397508
13.

Synthesis and metabotropic glutamate receptor activity of a 2-aminobicyclo[3.2.0]heptane-2,5-dicarboxylic acid, a molecule possessing an extended glutamate conformation.

Kozikowski AP, Araldi GL, Flippen-Anderson J, George C, Pshenichkin S, Surina E, Wroblewski J.

Bioorg Med Chem Lett. 1998 Apr 21;8(8):925-30.

PMID:
9871513
15.

Chemistry and pharmacology of the piperidine-based analogues of cocaine. Identification of potent DAT inhibitors lacking the tropane skeleton.

Kozikowski AP, Araldi GL, Boja J, Meil WM, Johnson KM, Flippen-Anderson JL, George C, Saiah E.

J Med Chem. 1998 May 21;41(11):1962-9.

PMID:
9599245
16.

Synthesis and biology of the conformationally restricted ACPD analogue, 2-aminobicyclo[2.1.1]hexane-2,5-dicarboxylic acid-I, a potent mGluR agonist.

Kozikowski AP, Steensma D, Araldi GL, Tückmantel W, Wang S, Pshenichkin S, Surina E, Wroblewski JT.

J Med Chem. 1998 May 7;41(10):1641-50.

PMID:
9572889
17.

Diastereomeric separation of 1,5-benzodiazepines due to the presence of a chiral centre on the N-5 alkylic chain.

Araldi GL, Donati D, Tranquillini ME, Ursini A.

Farmaco. 1998 Jan;53(1):49-54.

PMID:
9543726
18.

Synthesis of 5-membered ring-type compounds as potential cholecystokinin receptor ligands.

Pentassuglia G, Araldi GL, Donati D, Feriani A, Oliosi B, Pasquarello A, Ursini A.

Farmaco. 1997 Oct;52(10):573-81.

PMID:
9507668
19.

Dipolar Cycloaddition Route to Diverse Analogues of Cocaine: The 6- and 7-Substituted 3-Phenyltropanes.

Kozikowski AP, Araldi GL, Ball RG.

J Org Chem. 1997 Feb 7;62(3):503-509.

PMID:
11671441

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