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Items: 19

1.

Synthesis, Characterization, Crystal Structure, and DFT Study of a New Square Planar Cu(II) Complex Containing Bulky Adamantane Ligand.

Khanfar MA, Jaber AM, AlDamen MA, Al-Qawasmeh RA.

Molecules. 2018 Mar 20;23(3). pii: E701. doi: 10.3390/molecules23030701.

2.

Design, Synthesis and Qualitative Structure Activity Relationship Evaluations of Quinoline-Based Bisarylimidazoles as Antibacterial Motifs.

Al-Qawasmeh RA, Huthail BB, Sinnokrot MO, Semreen MH, Odeh RA, Abu-Zarga MH, Tarazi H, Yousef IA, Al-Tel TH.

Med Chem. 2016;12(6):563-73.

PMID:
27188185
3.

In-silico identification of the binding mode of synthesized adamantyl derivatives inside cholinesterase enzymes.

Al-Aboudi A, Al-Qawasmeh RA, Shahwan A, Mahmood U, Khalid A, Ul-Haq Z.

Acta Pharmacol Sin. 2015 Jul;36(7):879-86. doi: 10.1038/aps.2014.173. Epub 2015 May 4.

4.

Design synthesis and antibacterial activity studies of new thiadiazoloquinolone compounds.

Al-Qawasmeh RA, Abadleh MM, Zahra JA, El-Abadelah MM, Albashiti R, Zani F, Incerti M, Vicini P.

J Enzyme Inhib Med Chem. 2014 Dec;29(6):777-85. doi: 10.3109/14756366.2013.855925. Epub 2014 Feb 10.

PMID:
24506209
5.

Tandem multicomponent reactions toward the design and synthesis of novel antibacterial and cytotoxic motifs.

Semreen MH, El-Awady R, Abu-Odeh R, Saber-Ayad M, Al-Qawasmeh RA, Chouaib S, Voelter W, Al-Tel TH.

Curr Med Chem. 2013;20(11):1445-59.

PMID:
23409711
6.

2-(4-Methyl-phen-yl)quinoline-4-carb-oxy-lic acid.

Al-Qawasmeh RA, A Khanfar M, H Abu Zarga M, A Aldamen M.

Acta Crystallogr Sect E Struct Rep Online. 2012 Oct 1;68(Pt 10):o2892. doi: 10.1107/S160053681203797X. Epub 2012 Sep 8.

7.

Ethyl 7-chloro-1-cyclo-propyl-6-fluoro-8-nitro-4-oxo-1,4-dihydro-quinoline-3-carboxyl-ate.

Al-Qawasmeh RA.

Acta Crystallogr Sect E Struct Rep Online. 2012 Aug 1;68(Pt 8):o2533. doi: 10.1107/S1600536812011373. Epub 2012 Jul 25.

8.

Design, synthesis, and qualitative structure-activity evaluations of novel β-secretase inhibitors as potential Alzheimer's drug leads.

Al-Tel TH, Semreen MH, Al-Qawasmeh RA, Schmidt MF, El-Awadi R, Ardah M, Zaarour R, Rao SN, El-Agnaf O.

J Med Chem. 2011 Dec 22;54(24):8373-85. doi: 10.1021/jm201181f. Epub 2011 Nov 16.

PMID:
22044119
9.

Design, synthesis and in vitro antimicrobial evaluation of novel Imidazo[1,2-a]pyridine and imidazo[2,1-b][1,3]benzothiazole motifs.

Al-Tel TH, Al-Qawasmeh RA, Zaarour R.

Eur J Med Chem. 2011 May;46(5):1874-81. doi: 10.1016/j.ejmech.2011.02.051. Epub 2011 Feb 26.

PMID:
21414694
10.

Post Groebke-Blackburn multicomponent protocol: synthesis of new polyfunctional imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrimidine derivatives as potential antimicrobial agents.

Al-Tel TH, Al-Qawasmeh RA.

Eur J Med Chem. 2010 Dec;45(12):5848-55. doi: 10.1016/j.ejmech.2010.09.049. Epub 2010 Sep 25.

PMID:
20934788
11.

Synthesis and inhibition properties of a series of pyranose derivatives towards a Zn-metalloproteinase from Saccharomonospora canescens.

Dolashka-Angelova P, Abdel-Jalil RJ, Al-Qawasmeh RA, Stambolieva N, Voelter W.

Carbohydr Res. 2010 Nov 2;345(16):2343-7. doi: 10.1016/j.carres.2010.07.038. Epub 2010 Jul 29.

PMID:
20801431
12.

Potent antimicrobial activity of 3-(4,5-diaryl-1H-imidazol-2-yl)-1H-indole derivatives against methicillin-resistant Staphylococcus aureus.

Al-Qawasmeh RA, Huesca M, Nedunuri V, Peralta R, Wright J, Lee Y, Young A.

Bioorg Med Chem Lett. 2010 Jun 15;20(12):3518-20. doi: 10.1016/j.bmcl.2010.04.137. Epub 2010 May 17.

PMID:
20483613
13.

Synthesis and antimicrobial activity of cholic acid hydrazone analogues.

Rasras AJ, Al-Tel TH, Al-Aboudi AF, Al-Qawasmeh RA.

Eur J Med Chem. 2010 Jun;45(6):2307-13. doi: 10.1016/j.ejmech.2010.02.006. Epub 2010 Feb 6.

PMID:
20181416
14.

Rational design and synthesis of potent dibenzazepine motifs as beta-secretase inhibitors.

Al-Tel TH, Al-Qawasmeh RA, Schmidt MF, Al-Aboudi A, Rao SN, Sabri SS, Voelter W.

J Med Chem. 2009 Oct 22;52(20):6484-8. doi: 10.1021/jm9008482.

PMID:
19788239
15.

A novel small molecule with potent anticancer activity inhibits cell growth by modulating intracellular labile zinc homeostasis.

Huesca M, Lock LS, Khine AA, Viau S, Peralta R, Cukier IH, Jin H, Al-Qawasmeh RA, Lee Y, Wright J, Young A.

Mol Cancer Ther. 2009 Sep;8(9):2586-96. doi: 10.1158/1535-7163.MCT-08-1104. Epub 2009 Sep 15.

16.
17.

11-Phenyl-[b,e]-dibenzazepine compounds: novel antitumor agents.

Al-Qawasmeh RA, Lee Y, Cao MY, Gu X, Viau S, Lightfoot J, Wright JA, Young AH.

Bioorg Med Chem Lett. 2009 Jan 1;19(1):104-7. doi: 10.1016/j.bmcl.2008.11.001. Epub 2008 Nov 6.

PMID:
19027297
18.

Triaryl methane derivatives as antiproliferative agents.

Al-Qawasmeh RA, Lee Y, Cao MY, Gu X, Vassilakos A, Wright JA, Young A.

Bioorg Med Chem Lett. 2004 Jan 19;14(2):347-50.

PMID:
14698156
19.

NC381, a novel anticancer agent, arrests the cell cycle in G0-G1 and inhibits lung tumor cell growth in vitro and in vivo.

Cao MY, Lee Y, Feng NP, Al-Qawasmeh RA, Viau S, Gu XP, Lau L, Jin H, Wang M, Vassilakos A, Wright JA, Young AH.

J Pharmacol Exp Ther. 2004 Feb;308(2):538-46. Epub 2003 Nov 10.

PMID:
14610220

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