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Items: 1 to 20 of 100

1.

Development of novel lithocholic acid derivatives as vitamin D receptor agonists.

Masuno H, Kazui Y, Tanatani A, Fujii S, Kawachi E, Ikura T, Ito N, Yamamoto K, Kagechika H.

Bioorg Med Chem. 2019 Aug 15;27(16):3674-3681. doi: 10.1016/j.bmc.2019.07.003. Epub 2019 Jul 3.

PMID:
31300316
2.

Crystal Structure of the Vitamin D Receptor Ligand-Binding Domain with Lithocholic Acids.

Ikura T, Ito N.

Vitam Horm. 2016;100:117-36. doi: 10.1016/bs.vh.2015.10.004. Epub 2015 Dec 8. Review.

PMID:
26827950
3.

Evolutionary and Functional Diversification of the Vitamin D Receptor-Lithocholic Acid Partnership.

Kollitz EM, Zhang G, Hawkins MB, Whitfield GK, Reif DM, Kullman SW.

PLoS One. 2016 Dec 12;11(12):e0168278. doi: 10.1371/journal.pone.0168278. eCollection 2016.

4.

Novel vitamin D receptor ligands having a carboxyl group as an anchor to arginine 274 in the ligand-binding domain.

Fujishima T, Tsuji G, Tanaka C, Harayama H.

J Steroid Biochem Mol Biol. 2010 Jul;121(1-2):60-2. doi: 10.1016/j.jsbmb.2010.04.020. Epub 2010 May 6.

PMID:
20435140
5.

Selective activation of vitamin D receptor by lithocholic acid acetate, a bile acid derivative.

Adachi R, Honma Y, Masuno H, Kawana K, Shimomura I, Yamada S, Makishima M.

J Lipid Res. 2005 Jan;46(1):46-57. Epub 2004 Oct 16.

6.

[Update on recent progress in vitamin D research. Vitamin D receptor and the nuclear receptor superfamily.]

Makishima M.

Clin Calcium. 2017;27(11):1533-1541. doi: CliCa171115331541. Review. Japanese.

PMID:
29074825
7.

Crystal structures of complexes of vitamin D receptor ligand-binding domain with lithocholic acid derivatives.

Masuno H, Ikura T, Morizono D, Orita I, Yamada S, Shimizu M, Ito N.

J Lipid Res. 2013 Aug;54(8):2206-13. doi: 10.1194/jlr.M038307. Epub 2013 May 30.

9.

Lithocholic Acid Is a Vitamin D Receptor Ligand That Acts Preferentially in the Ileum.

Ishizawa M, Akagi D, Makishima M.

Int J Mol Sci. 2018 Jul 6;19(7). pii: E1975. doi: 10.3390/ijms19071975.

10.

Structural determinants for vitamin D receptor response to endocrine and xenobiotic signals.

Adachi R, Shulman AI, Yamamoto K, Shimomura I, Yamada S, Mangelsdorf DJ, Makishima M.

Mol Endocrinol. 2004 Jan;18(1):43-52. Epub 2003 Oct 2.

PMID:
14525957
11.

Molecular and functional comparison of 1,25-dihydroxyvitamin D(3) and the novel vitamin D receptor ligand, lithocholic acid, in activating transcription of cytochrome P450 3A4.

Jurutka PW, Thompson PD, Whitfield GK, Eichhorst KR, Hall N, Dominguez CE, Hsieh JC, Haussler CA, Haussler MR.

J Cell Biochem. 2005 Apr 1;94(5):917-43.

PMID:
15578590
12.

Lithocholic acid derivatives act as selective vitamin D receptor modulators without inducing hypercalcemia.

Ishizawa M, Matsunawa M, Adachi R, Uno S, Ikeda K, Masuno H, Shimizu M, Iwasaki K, Yamada S, Makishima M.

J Lipid Res. 2008 Apr;49(4):763-72. doi: 10.1194/jlr.M700293-JLR200. Epub 2008 Jan 7.

13.

1alpha,25-Dihydroxyvitamin D(3)-26,23-lactam analogues function as vitamin D receptor antagonists in human and rodent cells.

Ishizuka S, Kurihara N, Hiruma Y, Miura D, Namekawa J, Tamura A, Kato-Nakamura Y, Nakano Y, Takenouchi K, Hashimoto Y, Nagasawa K, Roodman GD.

J Steroid Biochem Mol Biol. 2008 Jun;110(3-5):269-77. doi: 10.1016/j.jsbmb.2007.11.007. Epub 2008 Apr 22.

14.

Structural insights into the molecular mechanism of vitamin D receptor activation by lithocholic acid involving a new mode of ligand recognition.

Belorusova AY, Eberhardt J, Potier N, Stote RH, Dejaegere A, Rochel N.

J Med Chem. 2014 Jun 12;57(11):4710-9. doi: 10.1021/jm5002524. Epub 2014 May 21.

PMID:
24818857
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17.

A new class of vitamin D analogues that induce structural rearrangement of the ligand-binding pocket of the receptor.

Inaba Y, Yoshimoto N, Sakamaki Y, Nakabayashi M, Ikura T, Tamamura H, Ito N, Shimizu M, Yamamoto K.

J Med Chem. 2009 Mar 12;52(5):1438-49. doi: 10.1021/jm8014348.

PMID:
19193059
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