Format
Sort by
Items per page

Send to

Choose Destination

Search results

Items: 42

1.

Study of 2-aminoquinolin-4(1H)-one under Mannich and retro-Mannich reaction.

Funk P, Motyka K, Soural M, Malon M, Koshino H, Kusz J, Hlavac J.

PLoS One. 2017 May 30;12(5):e0175364. doi: 10.1371/journal.pone.0175364. eCollection 2017.

2.

RP-HPLC determination of dissociation constant using solely aqueous mobile phase.

Volná T, Motyka K, Hlaváč J.

J Pharm Biomed Anal. 2017 Feb 5;134:143-148. doi: 10.1016/j.jpba.2016.11.038. Epub 2016 Nov 27.

PMID:
27915191
3.

Solid-Phase Synthesis of ɤ-Lactone and 1,2-Oxazine Derivatives and Their Efficient Chiral Analysis.

Krupkova S, Aguete GP, Kocmanova L, Volna T, Grepl M, Novakova L, Miller MJ, Hlavac J.

PLoS One. 2016 Nov 28;11(11):e0166558. doi: 10.1371/journal.pone.0166558. eCollection 2016.

4.

Stereo- and regioselectivity of the hetero-Diels-Alder reaction of nitroso derivatives with conjugated dienes.

Brulíková L, Harrison A, Miller MJ, Hlaváč J.

Beilstein J Org Chem. 2016 Sep 1;12:1949-1980. doi: 10.3762/bjoc.12.184. eCollection 2016. Review.

5.

A solid-phase synthetic approach to pH-independent rhodamine-type fluorophores.

Brulikova L, Okorochenkova Y, Hlavac J.

Org Biomol Chem. 2016 Nov 8;14(44):10437-10443.

PMID:
27754510
6.

MYD88 and functionally related genes are associated with multiple infections in a model population of Kenyan village dogs.

Necesankova M, Vychodilova L, Albrechtova K, Kennedy LJ, Hlavac J, Sedlak K, Modry D, Janova E, Vyskocil M, Horin P.

Mol Biol Rep. 2016 Dec;43(12):1451-1463. Epub 2016 Sep 21.

PMID:
27655108
7.

Efficient Route to Deuterated Aromatics by the Deamination of Anilines.

Burglova K, Okorochenkov S, Hlavac J.

Org Lett. 2016 Jul 15;18(14):3342-5. doi: 10.1021/acs.orglett.6b01438. Epub 2016 Jul 5.

PMID:
27378277
8.

New (green) methodology for efficient hydrazine cleavage.

Kubovičová L, Bürglová K, Hlaváč J.

Org Biomol Chem. 2016 Jun 7;14(21):4824-8. doi: 10.1039/c6ob00737f. Epub 2016 May 4.

PMID:
27143442
9.

Study and application of noncatalyzed photoinduced conjugation of azides and cycloocta-1,2,3-selenadiazoles.

Jedináková P, Šebej P, Slanina T, Klán P, Hlaváč J.

Chem Commun (Camb). 2016 Apr 4;52(26):4792-5. doi: 10.1039/c6cc01789d. Epub 2016 Mar 9.

PMID:
26956058
10.

Effects of Ginger Phenylpropanoids and Quercetin on Nrf2-ARE Pathway in Human BJ Fibroblasts and HaCaT Keratinocytes.

Schadich E, Hlaváč J, Volná T, Varanasi L, Hajdúch M, Džubák P.

Biomed Res Int. 2016;2016:2173275. doi: 10.1155/2016/2173275. Epub 2016 Jan 28.

11.

7-(2-Thienyl)-7-Deazaadenosine (AB61), a New Potent Nucleoside Cytostatic with a Complex Mode of Action.

Perlíková P, Rylová G, Nauš P, Elbert T, Tloušťová E, Bourderioux A, Slavětínská LP, Motyka K, Doležal D, Znojek P, Nová A, Harvanová M, Džubák P, Šiller M, Hlaváč J, Hajdúch M, Hocek M.

Mol Cancer Ther. 2016 May;15(5):922-37. doi: 10.1158/1535-7163.MCT-14-0933. Epub 2016 Jan 27.

12.

Non-Catalyzed Click Reactions of ADIBO Derivatives with 5-Methyluridine Azides and Conformational Study of the Resulting Triazoles.

Smyslova P, Popa I, Lyčka A, Tejral G, Hlavac J.

PLoS One. 2015 Dec 16;10(12):e0144613. doi: 10.1371/journal.pone.0144613. eCollection 2015.

13.

Solid-supported hydrazone of 4-(4'-formyl-3'-methoxyphenoxy)butyric acid as a new traceless linker for solid-phase synthesis.

Okorochenkov S, Burglova K, Popa I, Hlavac J.

Org Lett. 2015 Jan 16;17(2):180-3. doi: 10.1021/ol5034223. Epub 2014 Dec 23.

PMID:
25536078
14.

Affinity-based methods in drug-target discovery.

Rylova G, Ozdian T, Varanasi L, Soural M, Hlavac J, Holub D, Dzubak P, Hajduch M.

Curr Drug Targets. 2015;16(1):60-76.

PMID:
25410410
15.

Fluorescence properties of selected benzo[c]phenanthridines.

Motyka K, Stýskala J, Cankař P, Hlaváč J.

J Fluoresc. 2014 Jul;24(4):1177-82. doi: 10.1007/s10895-014-1398-8. Epub 2014 May 6.

PMID:
24796969
16.

4-Chloro-2-fluoro-5-nitrobenzoic acid as a possible building block for solid-phase synthesis of various heterocyclic scaffolds.

Křupková S, Funk P, Soural M, Hlaváč J.

ACS Comb Sci. 2013 Jan 14;15(1):20-8. doi: 10.1021/co300109h. Epub 2013 Jan 3.

PMID:
23163899
17.

DNA interstrand cross-linking agents and their chemotherapeutic potential.

Brulikova L, Hlavac J, Hradil P.

Curr Med Chem. 2012;19(3):364-85. Review.

PMID:
22335513
18.

Overcoming instability and low solubility of new cytostatic compounds: a comparison of two approaches.

di Cagno M, Stein PC, Styskala J, Hlaváč J, Skalko-Basnet N, Bauer-Brandl A.

Eur J Pharm Biopharm. 2012 Apr;80(3):657-62. doi: 10.1016/j.ejpb.2011.11.016. Epub 2011 Nov 28.

PMID:
22142591
19.

Synthesis of various 5-alkoxymethyluracil analogues and structure-cytotoxic activity relationship study.

Brulíková L, Džubák P, Hajdúch M, Hlaváč J.

Carbohydr Res. 2011 Oct 18;346(14):2136-44. doi: 10.1016/j.carres.2011.07.026. Epub 2011 Aug 5.

PMID:
21864833
20.

Purine scaffold effect on fluorescence properties of purine-hydroxyquinolinone bisheterocycles.

Motyka K, Vaňková B, Hlaváč J, Soural M, Funk P.

J Fluoresc. 2011 Nov;21(6):2207-12. doi: 10.1007/s10895-011-0925-0. Epub 2011 Aug 9.

PMID:
21826428
21.

Synthesis, reactivity and biological activity of 5-alkoxymethyluracil analogues.

Brulikova L, Hlavac J.

Beilstein J Org Chem. 2011;7:678-98. doi: 10.3762/bjoc.7.80. Epub 2011 May 26.

22.

Occurrence of filaria in domestic dogs of Samburu pastoralists in Northern Kenya and its associations with canine distemper.

Albrechtová K, Sedlák K, Petrželková KJ, Hlaváč J, Mihalca AD, Lesingirian A, Kanyari PW, Modrý D.

Vet Parasitol. 2011 Dec 15;182(2-4):230-8. doi: 10.1016/j.vetpar.2011.05.042. Epub 2011 May 27.

PMID:
21724332
23.

Direct C-H arylation of purine on solid phase and its use for chemical libraries synthesis.

Vanková B, Krchnák V, Soural M, Hlavác J.

ACS Comb Sci. 2011 Sep 12;13(5):496-500. doi: 10.1021/co200075r. Epub 2011 Jun 30.

PMID:
21675766
24.

Liposomal solubilization of new 3-hydroxy-quinolinone derivatives with promising anticancer activity: a screening method to identify maximum incorporation capacity.

di Cagno M, Styskala J, Hlaváč J, Brandl M, Bauer-Brandl A, Skalko-Basnet N.

J Liposome Res. 2011 Dec;21(4):272-8. doi: 10.3109/08982104.2010.550265. Epub 2011 Feb 17.

PMID:
21323606
25.

2-phenylsubstituted-3-hydroxyquinolin-4(1H)-one-carboxamides: Structure-cytotoxic activity relationship study.

Soural M, Hlavác J, Funk P, Dzubák P, Hajdúch M.

ACS Comb Sci. 2011 Jan 10;13(1):39-44. doi: 10.1021/co100013t. Epub 2010 Nov 10.

PMID:
21247123
26.

Solid-phase synthesis of highly diverse purine-hydroxyquinolinone bisheterocycles.

Vanková B, Hlavác J, Soural M.

J Comb Chem. 2010 Nov 8;12(6):890-4. doi: 10.1021/cc100132z. Epub 2010 Sep 17.

PMID:
20849113
27.

Synthesis of 5-[alkoxy-(4-nitro-phenyl)-methyl]-uridines and study of their cytotoxic activity.

Brulíková L, Dzubák P, Hajdúch M, Lachnitová L, Kollareddy M, Kolár M, Bogdanová K, Hlavác J.

Eur J Med Chem. 2010 Sep;45(9):3588-94. doi: 10.1016/j.ejmech.2010.05.003. Epub 2010 May 12.

PMID:
20605656
28.

Mass spectrometry as a tool for characterization of N,N-dialkylaminoethane-2-thiols--precursors and degradation products of chemical warfare agents.

Papousková B, Bednár P, Stýskala J, Hlavác J, Barták P, Lemr K.

J Mass Spectrom. 2009 Nov;44(11):1604-12. doi: 10.1002/jms.1674.

PMID:
19802902
29.

Solid-phase synthesis of 3-hydroxy-6-nitroquinolin-4(1H)-ones with two diversity positions.

Krupková S, Soural M, Hlavác J, Hradil P.

J Comb Chem. 2009 Nov-Dec;11(6):951-5. doi: 10.1021/cc900068w.

PMID:
19778035
30.

3-Hydroxy-2-phenyl-4(1H)-quinolinones as promising biologically active compounds.

Hradil P, Hlavác J, Soural M, Hajdúch M, Kolár M, Vecerová R.

Mini Rev Med Chem. 2009 Jun;9(6):696-702. Review.

PMID:
19519495
31.

Mass spectrometric study of selected precursors and degradation products of chemical warfare agents.

Papousková B, Bednár P, Frysová I, Stýskala J, Hlavác J, Barták P, Ulrichová J, Jirkovský J, Lemr K.

J Mass Spectrom. 2007 Dec;42(12):1550-61.

PMID:
18085550
32.

Synthesis and cytotoxic activity of various 5-[alkoxy-(4-nitro-phenyl)-methyl]-uracils in their racemic form.

Spácilová L, Dzubák P, Hajdúch M, Krupková S, Hradil P, Hlavác J.

Bioorg Med Chem Lett. 2007 Dec 1;17(23):6647-50. Epub 2007 Sep 8.

PMID:
17935983
33.

Synthesis and cytotoxic activity of substituted 2-phenyl-3-hydroxy-4(1H)-quinolinones-7-carboxylic acids and their phenacyl esters.

Soural M, Hlavác J, Hradil P, Frysová I, Hajdúch M, Bertolasi V, Malon M.

Eur J Med Chem. 2006 Apr;41(4):467-74. Epub 2006 Mar 15.

PMID:
16540209
34.

Some new routes for the preparation of 3-amino-2-phenyl-4(1H)-quinolinones from anthranilamides.

Hradil P, Grepl M, Hlavác J, Soural M, Malon M, Bertolasi V.

J Org Chem. 2006 Jan 20;71(2):819-22.

PMID:
16409002
36.

Capillary electrophoresis/mass spectrometry: a promising tool for the control of some physiologically hazardous compounds. I-derivatives of 3-quinuclidinol.

Bednár P, Lemr K, Barták P, Sevcík J, Hlavác J, Stýskala J, Wiedermannová I, Stránský Z.

J Mass Spectrom. 2002 Dec;37(12):1213-8.

PMID:
12489080
37.

Simple method for determination of dietary fiber in frozen foods.

al-Hasani SM, Hlavac J, Huntsman MA.

J AOAC Int. 1993 Sep-Oct;76(5):1014-6.

PMID:
8241807
38.

Rapid determination of cholesterol in single and multicomponent prepared foods.

al-Hasani SM, Hlavac J, Carpenter MW.

J AOAC Int. 1993 Jul-Aug;76(4):902-6.

PMID:
8374334
39.

Contribution to investigations of endemic degeneration. IV. Hearing disorders and the incidence of morphological ENT anomalies in endemic degeneration.

Kremenová J, Bláha K, Hlavác J, Reisenauer R.

Rev Czech Med. 1967;13(1):30-42. No abstract available.

PMID:
6044709
40.

[CLINICAL PATHOLOGY OF THE UPPER RESPIRATORY TRACT AND LARYNX IN WELDERS].

BLAHA K, HOUSTKOVA E, HLAVAC J.

Cesk Otolaryngol. 1963 Jun;12:161-7. Czech. No abstract available.

PMID:
14043796
41.

[Rupture of hypopharynx caused by indirect injury].

HLAVAC J.

Cesk Otolaryngol. 1957 Jun;6(3):140-1. Czech. No abstract available.

PMID:
13461170
42.

[Psychogenic deafness].

MELLAN J, HLAVAC J.

Cesk Psychiatr. 1957 Mar;53(2):117-21. Czech. No abstract available.

PMID:
13447087

Supplemental Content

Loading ...
Support Center