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Items: 24

1.

Synthesis and optimization of furano[3,2-d]pyrimidines as selective spleen tyrosine kinase (Syk) inhibitors.

Hoemann M, Wilson N, Argiriadi M, Banach D, Burchat A, Calderwood D, Clapham B, Cox P, Duignan DB, Konopacki D, Somal G, Vasudevan A.

Bioorg Med Chem Lett. 2016 Nov 15;26(22):5562-5567. doi: 10.1016/j.bmcl.2016.09.077. Epub 2016 Oct 11.

PMID:
27789138
2.

Synthesis and Pharmacology of (Pyridin-2-yl)methanol Derivatives as Novel and Selective Transient Receptor Potential Vanilloid 3 Antagonists.

Gomtsyan A, Schmidt RG, Bayburt EK, Gfesser GA, Voight EA, Daanen JF, Schmidt DL, Cowart MD, Liu H, Altenbach RJ, Kort ME, Clapham B, Cox PB, Shrestha A, Henry R, Whittern DN, Reilly RM, Puttfarcken PS, Brederson JD, Song P, Li B, Huang SM, McDonald HA, Neelands TR, McGaraughty SP, Gauvin DM, Joshi SK, Banfor PN, Segreti JA, Shebley M, Faltynek CR, Dart MJ, Kym PR.

J Med Chem. 2016 May 26;59(10):4926-47. doi: 10.1021/acs.jmedchem.6b00287. Epub 2016 May 2.

PMID:
27077528
3.

Size-dependent phase transformation of catalytically active nanoparticles captured in situ.

Fischer N, Clapham B, Feltes T, van Steen E, Claeys M.

Angew Chem Int Ed Engl. 2014 Jan 27;53(5):1342-5. doi: 10.1002/anie.201306899. Epub 2014 Jan 21.

PMID:
24449054
4.

Construction and validation of an automated flow hydrogenation instrument for application in high-throughput organic chemistry.

Clapham B, Wilson NS, Michmerhuizen MJ, Blanchard DP, Dingle DM, Nemcek TA, Pan JY, Sauer DR.

J Comb Chem. 2008 Jan-Feb;10(1):88-93. Epub 2007 Dec 21.

PMID:
18095655
5.

Antibody interference with N-acyl homoserine lactone-mediated bacterial quorum sensing.

Kaufmann GF, Sartorio R, Lee SH, Mee JM, Altobell LJ 3rd, Kujawa DP, Jeffries E, Clapham B, Meijler MM, Janda KD.

J Am Chem Soc. 2006 Mar 8;128(9):2802-3.

6.

Revisiting quorum sensing: Discovery of additional chemical and biological functions for 3-oxo-N-acylhomoserine lactones.

Kaufmann GF, Sartorio R, Lee SH, Rogers CJ, Meijler MM, Moss JA, Clapham B, Brogan AP, Dickerson TJ, Janda KD.

Proc Natl Acad Sci U S A. 2005 Jan 11;102(2):309-14. Epub 2004 Dec 27.

7.

Application of diazocarbonyls in the synthesis of chemical libraries.

Clapham B.

Curr Opin Drug Discov Devel. 2004 Nov;7(6):813-22.

PMID:
15595442
8.

N-H insertion reactions of primary ureas: the synthesis of highly substituted imidazolones and imidazoles from diazocarbonyls.

Lee SH, Yoshida K, Matsushita H, Clapham B, Koch G, Zimmermann J, Janda KD.

J Org Chem. 2004 Dec 10;69(25):8829-35.

PMID:
15575764
9.

N-h insertion reactions of Boc-amino acid amides: solution- and solid-phase synthesis of pyrazinones and pyrazines.

Matsushita H, Lee SH, Yoshida K, Clapham B, Koch G, Zimmermann J, Janda KD.

Org Lett. 2004 Nov 25;6(24):4627-9.

PMID:
15548092
10.

Smart cleavage reactions: the synthesis of an array of ureas from polymer-bound carbamates.

Lee SH, Matsushita H, Koch G, Zimmermann J, Clapham B, Janda KD.

J Comb Chem. 2004 Sep-Oct;6(5):822-7.

PMID:
15360219
11.
12.

Solid-phase rhodium carbenoid N-H insertion reactions: the synthesis of a diverse array of indoles.

Lee SH, Clapham B, Koch G, Zimmermann J, Janda KD.

J Comb Chem. 2003 Mar-Apr;5(2):188-96.

PMID:
12625710
13.

Scintillation-based potassium signalling using 2,5-diphenyloxazole-tagged aza-18-crown-6.

Clapham B, Sutherland AJ.

Chem Commun (Camb). 2003 Jan 7;(1):84-5.

PMID:
12610977
14.

Rhodium carbenoid N-H insertion reactions of primary ureas: solution and solid-phase synthesis of imidazolones.

Lee SH, Clapham B, Koch G, Zimmermann J, Janda KD.

Org Lett. 2003 Feb 20;5(4):511-4.

PMID:
12583756
15.
16.

Preparation of soluble and insoluble polymer supported IBX reagents.

Reed NN, Delgado M, Hereford K, Clapham B, Janda KD.

Bioorg Med Chem Lett. 2002 Aug 5;12(15):2047-9.

PMID:
12113839
17.

Preparation of new microgel polymers and their application as supports in organic synthesis.

Spanka C, Clapham B, Janda KD.

J Org Chem. 2002 May 3;67(9):3045-50.

PMID:
11975565
18.

Stille coupling reactions of 4-substituted-2,5-diphenyloxazoles.

Clapham B, Sutherland AJ.

J Org Chem. 2001 Dec 28;66(26):9033-7. No abstract available.

PMID:
11749641
19.

A sequential application of kinetic resolution and polymer-supported scavenging for the isolation of chiral secondary alcohols.

Córdova A, Tremblay MR, Clapham B, Janda KD.

J Org Chem. 2001 Aug 10;66(16):5645-8. No abstract available.

PMID:
11485501
20.

Solid-phase rhodium carbenoid reactions: an N-H insertion route to a diverse series of oxazoles.

Clapham B, Spanka C, Janda KD.

Org Lett. 2001 Jul 12;3(14):2173-6.

PMID:
11440572
21.
22.

Recent developments and applications of polymer-supported reagents in synthetic organic chemistry.

Brümmer O, Clapham B, Janda KD.

Curr Opin Drug Discov Devel. 2000 Jul;3(4):462-73.

PMID:
19649877
23.

AN INTERESTING CASE OF HYPOGLYCEMIA.

CLAPHAM B.

Med Leg J. 1965;33:72-3. No abstract available.

PMID:
14302177
24.

Vitamins in Experimental Hyperthyroidism.

Korenchevsky V, Hall K, Clapham B.

Br Med J. 1943 Feb 27;1(4286):245-7. No abstract available.

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