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Items: 1 to 20 of 35

1.

Evaluation of [(11)C]metergoline as a PET radiotracer for 5HTR in nonhuman primates.

Hooker JM, Kim SW, Reibel AT, Alexoff D, Xu Y, Shea C.

Bioorg Med Chem. 2010 Nov 15;18(22):7739-45. doi: 10.1016/j.bmc.2010.04.039. Epub 2010 Apr 20.

2.

Synthesis and evaluation of 1-[2-(4-[(11)C]methoxyphenyl)phenyl]piperazine for imaging of the serotonin 5-HT7 receptor in the rat brain.

Shimoda Y, Yui J, Xie L, Fujinaga M, Yamasaki T, Ogawa M, Nengaki N, Kumata K, Hatori A, Kawamura K, Zhang MR.

Bioorg Med Chem. 2013 Sep 1;21(17):5316-22. doi: 10.1016/j.bmc.2013.06.020. Epub 2013 Jun 17.

PMID:
23830697
3.

Synthesis and evaluation of [¹¹C]Cimbi-806 as a potential PET ligand for 5-HT₇ receptor imaging.

Herth MM, Hansen HD, Ettrup A, Dyssegaard A, Lehel S, Kristensen J, Knudsen GM.

Bioorg Med Chem. 2012 Jul 15;20(14):4574-81. doi: 10.1016/j.bmc.2012.05.005. Epub 2012 May 18.

PMID:
22682922
4.

Synthesis and in vivo evaluation of [O-methyl-11C] N-[3,5-dichloro-2-(methoxy)phenyl]-4-(methoxy)-3-(1-piperazinyl)benzenesulfonamide as an imaging probe for 5-HT6 receptors.

Liu F, Majo VJ, Prabhakaran J, Milak MS, John Mann J, Parsey RV, Kumar JS.

Bioorg Med Chem. 2011 Sep 1;19(17):5255-9. doi: 10.1016/j.bmc.2011.06.090. Epub 2011 Jul 19.

PMID:
21821420
5.
6.

Development of new carbon-11 labelled radiotracers for imaging GABAA- and GABAB-benzodiazepine receptors.

Moran MD, Wilson AA, Elmore CS, Parkes J, Ng A, Sadovski O, Graff A, Daskalakis ZJ, Houle S, Chapdelaine MJ, Vasdev N.

Bioorg Med Chem. 2012 Jul 15;20(14):4482-8. doi: 10.1016/j.bmc.2012.05.046. Epub 2012 May 24.

PMID:
22717238
7.

Brain uptake and distribution of the dopamine D3 /D2 receptor partial agonist [11 C]cariprazine: an in vivo positron emission tomography study in nonhuman primates.

Tóth M, Varrone A, Steiger C, Laszlovszky I, Horváth A, Kiss B, Gyertyán I, Adham N, Halldin C, Gulyás B.

Synapse. 2013 May;67(5):258-64. doi: 10.1002/syn.21631. Epub 2013 Feb 8.

PMID:
23238770
8.

Current status of positron emission tomography radiotracers for serotonin receptors in humans.

Zimmer L, Le Bars D.

J Labelled Comp Radiopharm. 2013 Mar-Apr;56(3-4):105-13. doi: 10.1002/jlcr.3001. Review.

PMID:
24285316
9.

[3H]Metergoline: a new ligand of serotonin receptors in the rat brain.

Hamon M, Mallat M, Herbet A, Nelson DL, Audinot M, Pichat L, Glowinski J.

J Neurochem. 1981 Feb;36(2):613-26.

PMID:
7463079
10.

Syntheses, radiolabelings, and in vitro evaluations of fluorinated PET radioligands of 5-HT6 serotoninergic receptors.

Colomb J, Becker G, Fieux S, Zimmer L, Billard T.

J Med Chem. 2014 May 8;57(9):3884-90. doi: 10.1021/jm500372e. Epub 2014 Apr 29.

PMID:
24754711
11.

Synthesis and Preclinical Evaluation of Three Novel Fluorine-18 Labeled Radiopharmaceuticals for P-Glycoprotein PET Imaging at the Blood-Brain Barrier.

Savolainen H, Cantore M, Colabufo NA, Elsinga PH, Windhorst AD, Luurtsema G.

Mol Pharm. 2015 Jul 6;12(7):2265-75. doi: 10.1021/mp5008103. Epub 2015 Jun 4.

PMID:
26043236
12.

Synthesis, in vitro characterization, and radiolabeling of reboxetine analogs as potential PET radioligands for imaging the norepinephrine transporter.

Zeng F, Jarkas N, Stehouwer JS, Voll RJ, Owens MJ, Kilts CD, Nemeroff CB, Goodman MM.

Bioorg Med Chem. 2008 Jan 15;16(2):783-93. Epub 2007 Oct 13.

PMID:
17983754
13.

Characterization of radioactive metabolites of 5-HT2A receptor PET ligand [18F]altanserin in human and rodent.

Tan PZ, Baldwin RM, Van Dyck CH, Al-Tikriti M, Roth B, Khan N, Charney DS, Innis RB.

Nucl Med Biol. 1999 Aug;26(6):601-8.

PMID:
10587097
14.

Synthesis and positron emission tomography studies of carbon-11-labeled imatinib (Gleevec).

Kil KE, Ding YS, Lin KS, Alexoff D, Kim SW, Shea C, Xu Y, Muench L, Fowler JS.

Nucl Med Biol. 2007 Feb;34(2):153-63.

15.

Radiosynthesis and biodistribution of a histamine H3 receptor antagonist 4-[3-(4-piperidin-1-yl-but-1-ynyl)-[11C]benzyl]-morpholine: evaluation of a potential PET ligand.

Airaksinen AJ, Jablonowski JA, van der Mey M, Barbier AJ, Klok RP, Verbeek J, Schuit R, Herscheid JD, Leysen JE, Carruthers NI, Lammertsma AA, Windhorst AD.

Nucl Med Biol. 2006 Aug;33(6):801-10.

PMID:
16934699
17.

Looking for a 5-HT7 radiotracer for positron emission tomography.

Andriès J, Lemoine L, Mouchel-Blaisot A, Tang S, Verdurand M, Le Bars D, Zimmer L, Billard T.

Bioorg Med Chem Lett. 2010 Jun 15;20(12):3730-3. doi: 10.1016/j.bmcl.2010.04.076. Epub 2010 Apr 24.

PMID:
20471259
18.

Positron emission tomography radiochemistry.

Mason NS, Mathis CA.

Neuroimaging Clin N Am. 2003 Nov;13(4):671-87. Review.

PMID:
15024954
19.

Evaluation of 3-Ethyl-3-(phenylpiperazinylbutyl)oxindoles as PET Ligands for the Serotonin 5-HT₇ Receptor: Synthesis, Pharmacology, Radiolabeling, and in Vivo Brain Imaging in Pigs.

Herth MM, Andersen VL, Hansen HD, Stroth N, Volk B, Lehel S, Dyssegaard A, Ettrup A, Svenningsson P, Knudsen GM, Kristensen JL.

J Med Chem. 2015 Apr 23;58(8):3631-6. doi: 10.1021/acs.jmedchem.5b00095. Epub 2015 Apr 13.

PMID:
25825999
20.

[11C]AZ10419369: a selective 5-HT1B receptor radioligand suitable for positron emission tomography (PET). Characterization in the primate brain.

Pierson ME, Andersson J, Nyberg S, McCarthy DJ, Finnema SJ, Varnäs K, Takano A, Karlsson P, Gulyás B, Medd AM, Lee CM, Powell ME, Heys JR, Potts W, Seneca N, Mrzljak L, Farde L, Halldin C.

Neuroimage. 2008 Jul 1;41(3):1075-85. doi: 10.1016/j.neuroimage.2008.02.063. Epub 2008 Mar 14.

PMID:
18434202

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