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Items: 1 to 20 of 70

1.

Iminochromene inhibitors of dynamins I and II GTPase activity and endocytosis.

Hill TA, Mariana A, Gordon CP, Odell LR, Robertson MJ, McGeachie AB, Chau N, Daniel JA, Gorgani NN, Robinson PJ, McCluskey A.

J Med Chem. 2010 May 27;53(10):4094-102. doi: 10.1021/jm100119c.

PMID:
20426422
2.

The pthaladyns: GTP competitive inhibitors of dynamin I and II GTPase derived from virtual screening.

Odell LR, Howan D, Gordon CP, Robertson MJ, Chau N, Mariana A, Whiting AE, Abagyan R, Daniel JA, Gorgani NN, Robinson PJ, McCluskey A.

J Med Chem. 2010 Jul 22;53(14):5267-80. doi: 10.1021/jm100442u.

PMID:
20575553
3.

Myristyl trimethyl ammonium bromide and octadecyl trimethyl ammonium bromide are surface-active small molecule dynamin inhibitors that block endocytosis mediated by dynamin I or dynamin II.

Quan A, McGeachie AB, Keating DJ, van Dam EM, Rusak J, Chau N, Malladi CS, Chen C, McCluskey A, Cousin MA, Robinson PJ.

Mol Pharmacol. 2007 Dec;72(6):1425-39.

4.

Inhibition of dynamin mediated endocytosis by the dynoles--synthesis and functional activity of a family of indoles.

Hill TA, Gordon CP, McGeachie AB, Venn-Brown B, Odell LR, Chau N, Quan A, Mariana A, Sakoff JA, Chircop M, Robinson PJ, McCluskey A.

J Med Chem. 2009 Jun 25;52(12):3762-73. doi: 10.1021/jm900036m.

PMID:
19459681
5.

Suppression of dynamin GTPase activity by sertraline leads to inhibition of dynamin-dependent endocytosis.

Takahashi K, Miyoshi H, Otomo M, Osada K, Yamaguchi N, Nakashima H.

Biochem Biophys Res Commun. 2010 Jan 1;391(1):382-7. doi: 10.1016/j.bbrc.2009.11.067.

PMID:
19913505
6.

Development of second-generation indole-based dynamin GTPase inhibitors.

Gordon CP, Venn-Brown B, Robertson MJ, Young KA, Chau N, Mariana A, Whiting A, Chircop M, Robinson PJ, McCluskey A.

J Med Chem. 2013 Jan 10;56(1):46-59. doi: 10.1021/jm300844m.

PMID:
23167654
7.

Some selective serotonin reuptake inhibitors inhibit dynamin I guanosine triphosphatase (GTPase).

Otomo M, Takahashi K, Miyoshi H, Osada K, Nakashima H, Yamaguchi N.

Biol Pharm Bull. 2008 Aug;31(8):1489-95.

8.

Calcineurin inhibition of dynamin I GTPase activity coupled to nerve terminal depolarization.

Liu JP, Sim AT, Robinson PJ.

Science. 1994 Aug 12;265(5174):970-3.

PMID:
8052858
9.

Small molecule inhibitors of dynamin I GTPase activity: development of dimeric tyrphostins.

Hill T, Odell LR, Edwards JK, Graham ME, McGeachie AB, Rusak J, Quan A, Abagyan R, Scott JL, Robinson PJ, McCluskey A.

J Med Chem. 2005 Dec 1;48(24):7781-8.

PMID:
16302817
10.

Azido and diazarinyl analogues of bis-tyrphostin as asymmetrical inhibitors of dynamin GTPase.

Odell LR, Chau N, Mariana A, Graham ME, Robinson PJ, McCluskey A.

ChemMedChem. 2009 Jul;4(7):1182-8. doi: 10.1002/cmdc.200900054.

PMID:
19437476
11.

Building a better dynasore: the dyngo compounds potently inhibit dynamin and endocytosis.

McCluskey A, Daniel JA, Hadzic G, Chau N, Clayton EL, Mariana A, Whiting A, Gorgani NN, Lloyd J, Quan A, Moshkanbaryans L, Krishnan S, Perera S, Chircop M, von Kleist L, McGeachie AB, Howes MT, Parton RG, Campbell M, Sakoff JA, Wang X, Sun JY, Robertson MJ, Deane FM, Nguyen TH, Meunier FA, Cousin MA, Robinson PJ.

Traffic. 2013 Dec;14(12):1272-89. doi: 10.1111/tra.12119.

12.

Increased GTP-binding to dynamin II does not stimulate receptor-mediated endocytosis.

Jeong MJ, Yoo J, Lee SS, Lee KI, Cho A, Kwon BM, Moon MJ, Park YM, Han MY.

Biochem Biophys Res Commun. 2001 Apr 27;283(1):136-42.

PMID:
11322780
13.
14.

The calcineurin-dynamin 1 complex as a calcium sensor for synaptic vesicle endocytosis.

Lai MM, Hong JJ, Ruggiero AM, Burnett PE, Slepnev VI, De Camilli P, Snyder SH.

J Biol Chem. 1999 Sep 10;274(37):25963-6.

15.
16.

Synthesis of potent chemical inhibitors of dynamin GTPase.

Lee S, Jung KY, Park J, Cho JH, Kim YC, Chang S.

Bioorg Med Chem Lett. 2010 Aug 15;20(16):4858-64. doi: 10.1016/j.bmcl.2010.06.092.

PMID:
20621477
17.
18.

Dynamin, endocytosis and intracellular signalling (review).

McClure SJ, Robinson PJ.

Mol Membr Biol. 1996 Oct-Dec;13(4):189-215. Review.

PMID:
9116759
19.
20.

Sorting nexin 9 interacts with dynamin 1 and N-WASP and coordinates synaptic vesicle endocytosis.

Shin N, Lee S, Ahn N, Kim SA, Ahn SG, YongPark Z, Chang S.

J Biol Chem. 2007 Sep 28;282(39):28939-50.

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