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Items: 1 to 20 of 1510

1.

The anxioselective agent 7-(2-chloropyridin-4-yl)pyrazolo-[1,5-a]-pyrimidin-3-yl](pyridin-2-yl)methanone (DOV 51892) is more efficacious than diazepam at enhancing GABA-gated currents at alpha1 subunit-containing GABAA receptors.

Popik P, Kostakis E, Krawczyk M, Nowak G, Szewczyk B, Krieter P, Chen Z, Russek SJ, Gibbs TT, Farb DH, Skolnick P, Lippa AS, Basile AS.

J Pharmacol Exp Ther. 2006 Dec;319(3):1244-52. Epub 2006 Sep 13.

2.

GABA(A) receptor alpha-1 subunit deletion alters receptor subtype assembly, pharmacological and behavioral responses to benzodiazepines and zolpidem.

Kralic JE, O'Buckley TK, Khisti RT, Hodge CW, Homanics GE, Morrow AL.

Neuropharmacology. 2002 Sep;43(4):685-94.

PMID:
12367614
3.

Diazepam enhancement of GABA-gated currents in binary and ternary GABAA receptors: relationship to benzodiazepine binding site density.

Granja R, Gunnersen D, Wong G, Valeyev A, Skolnick P.

J Mol Neurosci. 1997 Dec;9(3):187-95.

PMID:
9481620
4.

Functional comparison of the role of gamma subunits in recombinant human gamma-aminobutyric acidA/benzodiazepine receptors.

Wafford KA, Bain CJ, Whiting PJ, Kemp JA.

Mol Pharmacol. 1993 Aug;44(2):437-42.

PMID:
8102787
5.

Pharmacological properties of GABAA receptors containing gamma1 subunits.

Khom S, Baburin I, Timin EN, Hohaus A, Sieghart W, Hering S.

Mol Pharmacol. 2006 Feb;69(2):640-9. Epub 2005 Nov 4.

6.

SL651498: an anxioselective compound with functional selectivity for alpha2- and alpha3-containing gamma-aminobutyric acid(A) (GABA(A)) receptors.

Griebel G, Perrault G, Simiand J, Cohen C, Granger P, Decobert M, Françon D, Avenet P, Depoortere H, Tan S, Oblin A, Schoemaker H, Evanno Y, Sevrin M, George P, Scatton B.

J Pharmacol Exp Ther. 2001 Aug;298(2):753-68.

7.

Barbiturate interactions at the human GABAA receptor: dependence on receptor subunit combination.

Thompson SA, Whiting PJ, Wafford KA.

Br J Pharmacol. 1996 Feb;117(3):521-527.

8.
9.

RP 59037 and RP 60503: anxiolytic cyclopyrrolone derivatives with low sedative potential. interaction with the gamma-aminobutyric acidA/benzodiazepine receptor complex and behavioral effects in the rodent.

Doble A, Canton T, Dreisler S, Piot O, Boireau A, Stutzmann JM, Bardone MC, Rataud J, Roux M, Roussel G, et al.

J Pharmacol Exp Ther. 1993 Sep;266(3):1213-26.

PMID:
8103792
11.

Pharmacology of the human gamma-aminobutyric acidA receptor alpha 4 subunit expressed in Xenopus laevis oocytes.

Whittemore ER, Yang W, Drewe JA, Woodward RM.

Mol Pharmacol. 1996 Nov;50(5):1364-75.

PMID:
8913369
12.

3-Hydroxy-2'-methoxy-6-methylflavone: a potent anxiolytic with a unique selectivity profile at GABA(A) receptor subtypes.

Karim N, Gavande N, Wellendorph P, Johnston GA, Hanrahan JR, Chebib M.

Biochem Pharmacol. 2011 Dec 15;82(12):1971-83. doi: 10.1016/j.bcp.2011.09.002. Epub 2011 Sep 8.

PMID:
21924247
13.

Imidazenil: a new partial positive allosteric modulator of gamma-aminobutyric acid (GABA) action at GABAA receptors.

Giusti P, Ducić I, Puia G, Arban R, Walser A, Guidotti A, Costa E.

J Pharmacol Exp Ther. 1993 Aug;266(2):1018-28.

PMID:
8394902
14.

New evidence that the pharmacological effects of benzodiazepine receptor ligands can be associated with activities at different BZ (omega) receptor subtypes.

Griebel G, Perrault G, Letang V, Granger P, Avenet P, Schoemaker H, Sanger DJ.

Psychopharmacology (Berl). 1999 Sep;146(2):205-13.

PMID:
10525757
17.

Flavan-3-ol derivatives are positive modulators of GABA(A) receptors with higher efficacy for the alpha(2) subtype and anxiolytic action in mice.

Fernandez SP, Mewett KN, Hanrahan JR, Chebib M, Johnston GA.

Neuropharmacology. 2008 Oct;55(5):900-7. doi: 10.1016/j.neuropharm.2008.06.069. Epub 2008 Jul 9.

PMID:
18657554
18.

Properties of recombinant gamma-aminobutyric acid A receptor isoforms containing the alpha 5 subunit subtype.

Burgard EC, Tietz EI, Neelands TR, Macdonald RL.

Mol Pharmacol. 1996 Jul;50(1):119-27.

PMID:
8700104
19.

Molecular and neurochemical evaluation of the effects of etizolam on GABAA receptors under normal and stress conditions.

Sanna E, Pau D, Tuveri F, Massa F, Maciocco E, Acquas C, Floris C, Fontana SN, Maira G, Biggio G.

Arzneimittelforschung. 1999 Feb;49(2):88-95.

PMID:
10083975
20.

Anxiolytic-like effects of sinapic acid in mice.

Yoon BH, Jung JW, Lee JJ, Cho YW, Jang CG, Jin C, Oh TH, Ryu JH.

Life Sci. 2007 Jun 27;81(3):234-40. Epub 2007 May 21.

PMID:
17570441

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