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Items: 1 to 20 of 91

1.

Identification of an inhibitor-binding site to HIV-1 integrase with affinity acetylation and mass spectrometry.

Shkriabai N, Patil SS, Hess S, Budihas SR, Craigie R, Burke TR Jr, Le Grice SF, Kvaratskhelia M.

Proc Natl Acad Sci U S A. 2004 May 4;101(18):6894-9. Epub 2004 Apr 26.

2.

Arylisothiocyanate-containing esters of caffeic acid designed as affinity ligands for HIV-1 integrase.

Zhang X, Neamati N, Lee YK, Orr A, Brown RD, Whitaker N, Pommier Y, Burke TR Jr.

Bioorg Med Chem. 2001 Jul;9(7):1649-57.

PMID:
11425564
3.
4.

Binding aspects of baicalein to HIV-1 integrase.

Ahn HC, Lee SY, Kim JW, Son WS, Shin CG, Lee BJ.

Mol Cells. 2001 Aug 31;12(1):127-30.

5.

Mapping the epitope of an inhibitory monoclonal antibody to the C-terminal DNA-binding domain of HIV-1 integrase.

Yi J, Cheng H, Andrake MD, Dunbrack RL Jr, Roder H, Skalka AM.

J Biol Chem. 2002 Apr 5;277(14):12164-74. Epub 2002 Jan 22.

6.

Triketoacid inhibitors of HIV-integrase: a new chemotype useful for probing the integrase pharmacophore.

Walker MA, Johnson T, Ma Z, Banville J, Remillard R, Kim O, Zhang Y, Staab A, Wong H, Torri A, Samanta H, Lin Z, Deminie C, Terry B, Krystal M, Meanwell N.

Bioorg Med Chem Lett. 2006 Jun 1;16(11):2920-4. Epub 2006 Mar 20.

PMID:
16546383
7.

Characterization and structural analysis of HIV-1 integrase conservation.

Ceccherini-Silberstein F, Malet I, D'Arrigo R, Antinori A, Marcelin AG, Perno CF.

AIDS Rev. 2009 Jan-Mar;11(1):17-29. Review.

PMID:
19290031
8.

Hyrtiosal, from the marine sponge Hyrtios erectus, inhibits HIV-1 integrase binding to viral DNA by a new inhibitor binding site.

Du L, Shen L, Yu Z, Chen J, Guo Y, Tang Y, Shen X, Jiang H.

ChemMedChem. 2008 Jan;3(1):173-80.

PMID:
17943714
9.

Mass spectrometric analysis of the HIV-1 integrase-pyridoxal 5'-phosphate complex reveals a new binding site for a nucleotide inhibitor.

Williams KL, Zhang Y, Shkriabai N, Karki RG, Nicklaus MC, Kotrikadze N, Hess S, Le Grice SF, Craigie R, Pathak VK, Kvaratskhelia M.

J Biol Chem. 2005 Mar 4;280(9):7949-55. Epub 2004 Dec 22.

10.

Study on the inhibitory mechanism and binding mode of the hydroxycoumarin compound NSC158393 to HIV-1 integrase by molecular modeling.

Liu M, Cong XJ, Li P, Tan JJ, Chen WZ, Wang CX.

Biopolymers. 2009 Sep;91(9):700-9. doi: 10.1002/bip.21211.

PMID:
19382173
11.

Dissecting Tn5 transposition using HIV-1 integrase diketoacid inhibitors.

Czyz A, Stillmock KA, Hazuda DJ, Reznikoff WS.

Biochemistry. 2007 Sep 25;46(38):10776-89. Epub 2007 Aug 29.

PMID:
17725323
12.

Modeling, analysis, and validation of a novel HIV integrase structure provide insights into the binding modes of potent integrase inhibitors.

Chen X, Tsiang M, Yu F, Hung M, Jones GS, Zeynalzadegan A, Qi X, Jin H, Kim CU, Swaminathan S, Chen JM.

J Mol Biol. 2008 Jul 11;380(3):504-19. doi: 10.1016/j.jmb.2008.04.054. Epub 2008 May 1.

PMID:
18565342
13.

Symmetrical 1-pyrrolidineacetamide showing anti-HIV activity through a new binding site on HIV-1 integrase.

Du L, Zhao YX, Yang LM, Zheng YT, Tang Y, Shen X, Jiang HL.

Acta Pharmacol Sin. 2008 Oct;29(10):1261-7. doi: 10.1111/j.1745-7254.2008.00863.x.

14.
15.

An allosteric mechanism for inhibiting HIV-1 integrase with a small molecule.

Kessl JJ, Eidahl JO, Shkriabai N, Zhao Z, McKee CJ, Hess S, Burke TR Jr, Kvaratskhelia M.

Mol Pharmacol. 2009 Oct;76(4):824-32. doi: 10.1124/mol.109.058883. Epub 2009 Jul 28.

16.

Sequence-based design and discovery of peptide inhibitors of HIV-1 integrase: insight into the binding mode of the enzyme.

Li HY, Zawahir Z, Song LD, Long YQ, Neamati N.

J Med Chem. 2006 Jul 27;49(15):4477-86.

PMID:
16854053
17.

Correlation between shiftide activity and HIV-1 integrase inhibition by a peptide selected from a combinatorial library.

Armon-Omer A, Levin A, Hayouka Z, Butz K, Hoppe-Seyler F, Loya S, Hizi A, Friedler A, Loyter A.

J Mol Biol. 2008 Feb 29;376(4):971-82. doi: 10.1016/j.jmb.2007.11.095. Epub 2007 Dec 5.

PMID:
18201721
18.

Identification of cellular factors binding to acetylated HIV-1 integrase.

Allouch A, Cereseto A.

Amino Acids. 2011 Nov;41(5):1137-45. doi: 10.1007/s00726-009-0444-3. Epub 2009 Dec 18.

PMID:
20016921
19.

A structural study of model peptides derived from HIV-1 integrase central domain.

Maroun RG, Zargarian L, Stocklin R, Troalen F, Jankowski CK, Fermandjian S.

Rapid Commun Mass Spectrom. 2005;19(18):2539-48.

PMID:
16106350
20.

Discovery of a small-molecule HIV-1 integrase inhibitor-binding site.

Al-Mawsawi LQ, Fikkert V, Dayam R, Witvrouw M, Burke TR Jr, Borchers CH, Neamati N.

Proc Natl Acad Sci U S A. 2006 Jun 27;103(26):10080-5. Epub 2006 Jun 19.

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