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2012 2
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2020 4
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Page 1
Identification of Inhibitors of the Schistosoma mansoni VKR2 Kinase Domain.
Mathavan I, Liu LJ, Robinson SW, El-Sakkary N, Elatico AJJ, Gomez D, Nellas R, Owens RJ, Zuercher W, Navratilova I, Caffrey CR, Beis K. Mathavan I, et al. Among authors: el sakkary n. ACS Med Chem Lett. 2022 Oct 5;13(11):1715-1722. doi: 10.1021/acsmedchemlett.2c00248. eCollection 2022 Nov 10. ACS Med Chem Lett. 2022. PMID: 36385939 Free PMC article.
Lead Optimization of 3,5-Disubstituted-7-Azaindoles for the Treatment of Human African Trypanosomiasis.
Klug DM, Mavrogiannaki EM, Forbes KC, Silva L, Diaz-Gonzalez R, Pérez-Moreno G, Ceballos-Pérez G, Garcia-Hernández R, Bosch-Navarrete C, Cordón-Obras C, Gómez-Liñán C, Saura A, Momper JD, Martinez-Martinez MS, Manzano P, Syed A, El-Sakkary N, Caffrey CR, Gamarro F, Ruiz-Perez LM, Gonzalez Pacanowska D, Ferrins L, Navarro M, Pollastri MP. Klug DM, et al. Among authors: el sakkary n. J Med Chem. 2021 Jul 8;64(13):9404-9430. doi: 10.1021/acs.jmedchem.1c00674. Epub 2021 Jun 22. J Med Chem. 2021. PMID: 34156862 Free PMC article.
Structure-Bioactivity Relationships of Lapatinib Derived Analogs against Schistosoma mansoni.
Buskes MJ, Clements M, Bachovchin KA, Jalani HB, Leonard A, Bag S, Klug DM, Singh B, Campbell RF, Sciotti RJ, El-Sakkary N, Caffrey CR, Pollastri MP, Ferrins L. Buskes MJ, et al. Among authors: el sakkary n. ACS Med Chem Lett. 2020 Jan 10;11(3):258-265. doi: 10.1021/acsmedchemlett.9b00455. eCollection 2020 Mar 12. ACS Med Chem Lett. 2020. PMID: 32184954 Free PMC article.
Biomechanical interactions of Schistosoma mansoni eggs with vascular endothelial cells facilitate egg extravasation.
Yeh YT, Skinner DE, Criado-Hidalgo E, Chen NS, Garcia-De Herreros A, El-Sakkary N, Liu L, Zhang S, Kandasamy A, Chien S, Lasheras JC, Del Álamo JC, Caffrey CR. Yeh YT, et al. Among authors: el sakkary n. PLoS Pathog. 2022 Mar 22;18(3):e1010309. doi: 10.1371/journal.ppat.1010309. eCollection 2022 Mar. PLoS Pathog. 2022. PMID: 35316298 Free PMC article.
Development of subunit selective proteasome substrates for Schistosoma species.
Jiang Z, Silva EB, Liu C, Fajtová P, Liu LJ, El-Sakkary N, Skinner DE, Syed A, Wang SC, Caffrey CR, O'Donoghue AJ. Jiang Z, et al. Among authors: el sakkary n. bioRxiv [Preprint]. 2024 Feb 14:2024.02.13.580161. doi: 10.1101/2024.02.13.580161. bioRxiv. 2024. PMID: 38405969 Free PMC article. Preprint.
The Proteasome as a Drug Target in the Metazoan Pathogen, Schistosoma mansoni.
Bibo-Verdugo B, Wang SC, Almaliti J, Ta AP, Jiang Z, Wong DA, Lietz CB, Suzuki BM, El-Sakkary N, Hook V, Salvesen GS, Gerwick WH, Caffrey CR, O'Donoghue AJ. Bibo-Verdugo B, et al. Among authors: el sakkary n. ACS Infect Dis. 2019 Oct 11;5(10):1802-1812. doi: 10.1021/acsinfecdis.9b00237. Epub 2019 Aug 12. ACS Infect Dis. 2019. PMID: 31355632 Free PMC article.
EF24, a schistosomicidal curcumin analog: Insights from its synthesis and phenotypic, biochemical and cytotoxic activities.
Badoco FR, Paula LAL, Orenha RP, Mendes TMF, Squarisi IS, El-Sakkary N, Loiola MC, Katz N, Tavares DC, Sairre MI, Parreira RLT, Janku Cabral F, Alegretti SM, Caffrey CR, Magalhães LG. Badoco FR, et al. Among authors: el sakkary n. Chem Biol Interact. 2022 Dec 1;368:110191. doi: 10.1016/j.cbi.2022.110191. Epub 2022 Sep 28. Chem Biol Interact. 2022. PMID: 36181831 Free article.
17 results