Akahoshi F[Author] - Search Results

Year	Number of Results
1991	1
1994	1
1996	1
1998	3
2001	3
2003	1
2005	1
2006	2
2007	2
2012	2
2013	2
2016	1
2018	1
2024	0

1

[Pharmacological and clinical profile of a novel DPP-4 inhibitor teneligliptin hydrobromide hydrate (TENELIA(®)].

Goda M, Akahoshi F, Ishii S, Terata R, Hayashi Y. Goda M, et al. Among authors: akahoshi f. Nihon Yakurigaku Zasshi. 2013 Sep;142(3):134-43. doi: 10.1254/fpj.142.134. Nihon Yakurigaku Zasshi. 2013. PMID: 24025495 Review. Japanese. No abstract available.

2

Nonpeptidic chymase inhibitors: design and structure-activity relationships of pyrimidinone derivatives based on the predicted binding mode of a peptidic inhibitor.

Akahoshi F. Akahoshi F. Curr Pharm Des. 2003;9(15):1191-9. doi: 10.2174/1381612033454964. Curr Pharm Des. 2003. PMID: 12769746 Review.

3

Discovery of Novel Pyrazole-Based Selective Aldosterone Synthase (CYP11B2) Inhibitors: A New Template to Coordinate the Heme-Iron Motif of CYP11B2.

Sakakibara R, Sasaki W, Onda Y, Yamaguchi M, Ushirogochi H, Hiraga Y, Sato K, Nishio M, Egi Y, Takedomi K, Shimizu H, Ohbora T, Akahoshi F. Sakakibara R, et al. Among authors: akahoshi f. J Med Chem. 2018 Jul 12;61(13):5594-5608. doi: 10.1021/acs.jmedchem.8b00328. Epub 2018 Jun 22. J Med Chem. 2018. PMID: 29878770

4

Fused bicyclic heteroarylpiperazine-substituted L-prolylthiazolidines as highly potent DPP-4 inhibitors lacking the electrophilic nitrile group.

Yoshida T, Akahoshi F, Sakashita H, Sonda S, Takeuchi M, Tanaka Y, Nabeno M, Kishida H, Miyaguchi I, Hayashi Y. Yoshida T, et al. Among authors: akahoshi f. Bioorg Med Chem. 2012 Aug 15;20(16):5033-41. doi: 10.1016/j.bmc.2012.06.033. Epub 2012 Jul 5. Bioorg Med Chem. 2012. PMID: 22824762

5

Synthesis and pharmacological activity of triazolo[1,5-a]triazine derivatives inhibiting eosinophilia.

Akahoshi F, Takeda S, Okada T, Kajii M, Nishimura H, Sugiura M, Inoue Y, Fukaya C, Naito Y, Imagawa T, Nakamura N. Akahoshi F, et al. J Med Chem. 1998 Jul 30;41(16):2985-93. doi: 10.1021/jm970759u. J Med Chem. 1998. PMID: 9685237

6

Synthesis and pharmacological activity of triazole derivatives inhibiting eosinophilia.

Naito Y, Akahoshi F, Takeda S, Okada T, Kajii M, Nishimura H, Sugiura M, Fukaya C, Kagitani Y. Naito Y, et al. Among authors: akahoshi f. J Med Chem. 1996 Jul 19;39(15):3019-29. doi: 10.1021/jm9507993. J Med Chem. 1996. PMID: 8709136

7

Tissue distribution of teneligliptin in rats and comparisons with data reported for other dipeptidyl peptidase-4 inhibitors.

Nakamaru Y, Akahoshi F, Iijima H, Hisanaga N, Kume T. Nakamaru Y, et al. Among authors: akahoshi f. Biopharm Drug Dispos. 2016 Apr;37(3):142-155. doi: 10.1002/bdd.2003. Epub 2016 Jan 8. Biopharm Drug Dispos. 2016. PMID: 26749565 Free PMC article.

8

1-((S)-gamma-substituted prolyl)-(S)-2-cyanopyrrolidine as a novel series of highly potent DPP-IV inhibitors.

Sakashita H, Kitajima H, Nakamura M, Akahoshi F, Hayashi Y. Sakashita H, et al. Among authors: akahoshi f. Bioorg Med Chem Lett. 2005 May 16;15(10):2441-5. doi: 10.1016/j.bmcl.2005.03.077. Bioorg Med Chem Lett. 2005. PMID: 15863294

9

A comparative study of the binding modes of recently launched dipeptidyl peptidase IV inhibitors in the active site.

Nabeno M, Akahoshi F, Kishida H, Miyaguchi I, Tanaka Y, Ishii S, Kadowaki T. Nabeno M, et al. Among authors: akahoshi f. Biochem Biophys Res Commun. 2013 May 3;434(2):191-6. doi: 10.1016/j.bbrc.2013.03.010. Epub 2013 Mar 15. Biochem Biophys Res Commun. 2013. PMID: 23501107

10

Discovery and preclinical profile of teneligliptin (3-[(2S,4S)-4-[4-(3-methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]pyrrolidin-2-ylcarbonyl]thiazolidine): a highly potent, selective, long-lasting and orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes.

Yoshida T, Akahoshi F, Sakashita H, Kitajima H, Nakamura M, Sonda S, Takeuchi M, Tanaka Y, Ueda N, Sekiguchi S, Ishige T, Shima K, Nabeno M, Abe Y, Anabuki J, Soejima A, Yoshida K, Takashina Y, Ishii S, Kiuchi S, Fukuda S, Tsutsumiuchi R, Kosaka K, Murozono T, Nakamaru Y, Utsumi H, Masutomi N, Kishida H, Miyaguchi I, Hayashi Y. Yoshida T, et al. Among authors: akahoshi f. Bioorg Med Chem. 2012 Oct 1;20(19):5705-19. doi: 10.1016/j.bmc.2012.08.012. Epub 2012 Aug 17. Bioorg Med Chem. 2012. PMID: 22959556

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