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Items: 1 to 20 of 93

1.

Selenols: a new class of carbonic anhydrase inhibitors.

Angeli A, Tanini D, Nocentini A, Capperucci A, Ferraroni M, Gratteri P, Supuran CT.

Chem Commun (Camb). 2019 Jan 10;55(5):648-651. doi: 10.1039/c8cc08562e.

PMID:
30560259
2.

Synthesis of 1,2,4-triazole-5-on derivatives and determination of carbonic anhydrase II isoenzyme inhibition effects.

Akin S, Ayaloglu H, Gultekin E, Colak A, Bekircan O, Akatin MY.

Bioorg Chem. 2018 Oct 23;83:170-179. doi: 10.1016/j.bioorg.2018.10.042. [Epub ahead of print]

PMID:
30380445
3.

Carbonic anhydrase inhibitory potential of 1,2,4-triazole-3-thione derivatives of flurbiprofen, ibuprofen and 4-tert-butylbenzoic hydrazide : Design, synthesis, characterization, biochemical evaluation, molecular docking and dynamic simulation studies.

Abbas S, Zaib S, Ur Rahman S, Ali S, Hameed S, Tahir MN, Munawar KS, Shaheen F, Abbas SM, Iqbal J.

Med Chem. 2018 Oct 12. doi: 10.2174/1573406414666181012165156. [Epub ahead of print]

PMID:
30324884
4.

Synthesis, carbonic anhydrase inhibitory activity and antioxidant activity of some 1,3-oxazine derivatives.

Qamar R, Saeed A, Saeed M, Ashraf Z, Abbas Q, Hassan M, Albericio F.

Drug Dev Res. 2018 Nov;79(7):352-361. doi: 10.1002/ddr.21464. Epub 2018 Oct 10.

PMID:
30302774
5.

Mechanistic investigation of sulfonamide ligands as human carbonic anhydrase II inhibitors.

Alaei L, Khodarahmi R, Sheikh-Hasani V, Sheibani N, Moosavi-Movahedi AA.

Int J Biol Macromol. 2018 Dec;120(Pt A):1198-1207. doi: 10.1016/j.ijbiomac.2018.08.186. Epub 2018 Aug 31.

PMID:
30176324
6.

Development of a Fingerprint-Based Scoring Function for the Prediction of the Binding Mode of Carbonic Anhydrase II Inhibitors.

Poli G, Jha V, Martinelli A, Supuran CT, Tuccinardi T.

Int J Mol Sci. 2018 Jun 23;19(7). pii: E1851. doi: 10.3390/ijms19071851.

7.

4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors.

Salerno S, Barresi E, Amendola G, Berrino E, Milite C, Marini AM, Da Settimo F, Novellino E, Supuran CT, Cosconati S, Taliani S.

J Med Chem. 2018 Jul 12;61(13):5765-5770. doi: 10.1021/acs.jmedchem.8b00670. Epub 2018 Jun 27.

PMID:
29912561
8.

Extending the scope of amantadine drug by incorporation of phenolic azo Schiff bases as potent selective inhibitors of carbonic anhydrase II, drug-likeness and binding analysis.

Channar PA, Saeed A, Shahzad D, Larik FA, Hassan M, Raza H, Abbas Q, Seo SY.

Chem Biol Drug Des. 2018 Sep;92(3):1692-1698. doi: 10.1111/cbdd.13335. Epub 2018 Jun 26.

PMID:
29770563
9.

Implication of sulfonylurea derivatives as prospective inhibitors of human carbonic anhydrase II.

Idrees D, Hadianawala M, Mahapatra AD, Datta B, Roy S, Ahamad S, Khan P, Imtaiyaz Hassan M.

Int J Biol Macromol. 2018 Aug;115:961-969. doi: 10.1016/j.ijbiomac.2018.04.131. Epub 2018 Apr 26.

PMID:
29704602
10.

2-Benzylpiperazine: A new scaffold for potent human carbonic anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents.

Chiaramonte N, Bua S, Ferraroni M, Nocentini A, Bonardi A, Bartolucci G, Durante M, Lucarini L, Chiapponi D, Dei S, Manetti D, Teodori E, Gratteri P, Masini E, Supuran CT, Romanelli MN.

Eur J Med Chem. 2018 May 10;151:363-375. doi: 10.1016/j.ejmech.2018.04.002. Epub 2018 Apr 3.

PMID:
29635168
11.

Synthesis and Molecular Docking Studies of (E)-4-(Substituted-benzylideneamino)-2H-Chromen-2-one Derivatives: Entry to New Carbonic Anhydrase Class Of Inhibitors.

Fattah TA, Saeed A, Channar PA, Larik FA, Hassan M, Raza H, Abbas Q, Seo SY.

Drug Res (Stuttg). 2018 Jul;68(7):378-386. doi: 10.1055/s-0043-123998. Epub 2018 Feb 12.

PMID:
29433141
12.

Synthesis, biological evaluation and computational studies of novel iminothiazolidinone benzenesulfonamides as potent carbonic anhydrase II and IX inhibitors.

Mahmood SU, Saeed A, Bua S, Nocentini A, Gratteri P, Supuran CT.

Bioorg Chem. 2018 Apr;77:381-386. doi: 10.1016/j.bioorg.2018.01.031. Epub 2018 Jan 31.

PMID:
29421714
13.

Novel sulfonamide incorporating piperazine, aminoalcohol and 1,3,5-triazine structural motifs with carbonic anhydrase I, II and IX inhibitory action.

Havránková E, Csöllei J, Vullo D, Garaj V, Pazdera P, Supuran CT.

Bioorg Chem. 2018 Apr;77:25-37. doi: 10.1016/j.bioorg.2017.12.034. Epub 2018 Jan 3.

PMID:
29324250
14.

Ranking Power of the SQM/COSMO Scoring Function on Carbonic Anhydrase II-Inhibitor Complexes.

Pecina A, Brynda J, Vrzal L, Gnanasekaran R, Hořejší M, Eyrilmez SM, Řezáč J, Lepšík M, Řezáčová P, Hobza P, Majer P, Veverka V, Fanfrlík J.

Chemphyschem. 2018 Apr 5;19(7):873-879. doi: 10.1002/cphc.201701104. Epub 2018 Feb 19.

PMID:
29316128
15.

Design, synthesis and biological evaluation of novel pyridine-thiazolidinone derivatives as anticancer agents: Targeting human carbonic anhydrase IX.

Ansari MF, Idrees D, Hassan MI, Ahmad K, Avecilla F, Azam A.

Eur J Med Chem. 2018 Jan 20;144:544-556. doi: 10.1016/j.ejmech.2017.12.049. Epub 2017 Dec 15.

PMID:
29289880
16.

Sulfonamides containing curcumin scaffold: Synthesis, characterization, carbonic anhydrase inhibition and molecular docking studies.

Ahmed M, Qadir MA, Hameed A, Arshad MN, Asiri AM, Muddassar M.

Bioorg Chem. 2018 Feb;76:218-227. doi: 10.1016/j.bioorg.2017.11.015. Epub 2017 Nov 20.

PMID:
29190478
17.

Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms.

Krasavin M, Shetnev A, Sharonova T, Baykov S, Tuccinardi T, Kalinin S, Angeli A, Supuran CT.

Bioorg Chem. 2018 Feb;76:88-97. doi: 10.1016/j.bioorg.2017.10.005. Epub 2017 Oct 16.

PMID:
29153590
18.

Synthesis and Carbonic Anhydrase Inhibition of Tetrabromo Chalcone Derivatives.

Kocyigit UM, Budak Y, Eligüzel F, Taslimi P, Kılıç D, Gulçin İ, Ceylan M.

Arch Pharm (Weinheim). 2017 Dec;350(12). doi: 10.1002/ardp.201700198. Epub 2017 Nov 14.

PMID:
29134667
19.

The synthesis of novel sulfamides derived from β-benzylphenethylamines as acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase enzymes inhibitors.

Akıncıoğlu A, Kocaman E, Akıncıoğlu H, Salmas RE, Durdagi S, Gülçin İ, Supuran CT, Göksu S.

Bioorg Chem. 2017 Oct;74:238-250. doi: 10.1016/j.bioorg.2017.08.012. Epub 2017 Aug 23.

PMID:
28866249
20.

Identification of a New Zinc Binding Chemotype by Fragment Screening.

Chrysanthopoulos PK, Mujumdar P, Woods LA, Dolezal O, Ren B, Peat TS, Poulsen SA.

J Med Chem. 2017 Sep 14;60(17):7333-7349. doi: 10.1021/acs.jmedchem.7b00606. Epub 2017 Sep 1.

PMID:
28817930

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