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Items: 1 to 20 of 52

1.

Direct and Chemoselective Electrophilic Monofluoromethylation of Heteroatoms (O-, S-, N-, P-, Se-) with Fluoroiodomethane.

Senatore R, Malik M, Spreitzer M, Holzer W, Pace V.

Org Lett. 2020 Jan 31. doi: 10.1021/acs.orglett.9b04654. [Epub ahead of print]

PMID:
32004004
2.

Highly chemoselective difluoromethylative homologation of iso(thio)cyanates: expeditious access to unprecedented α,α-difluoro(thio)amides.

Miele M, D'Orsi R, Sridharan V, Holzer W, Pace V.

Chem Commun (Camb). 2019 Oct 24;55(86):12960-12963. doi: 10.1039/c9cc06929a.

PMID:
31602439
3.

Direct and Chemoselective Synthesis of Tertiary Difluoroketones via Weinreb Amide Homologation with a CHF2-Carbene Equivalent.

Miele M, Citarella A, Micale N, Holzer W, Pace V.

Org Lett. 2019 Oct 18;21(20):8261-8265. doi: 10.1021/acs.orglett.9b03024. Epub 2019 Oct 10.

PMID:
31599599
4.

A Combination of Pharmacophore and Docking-based Virtual Screening to Discover new Tyrosinase Inhibitors.

Vittorio S, Seidel T, Germanò MP, Gitto R, Ielo L, Garon A, Rapisarda A, Pace V, Langer T, De Luca L.

Mol Inform. 2019 Sep 11. doi: 10.1002/minf.201900054. [Epub ahead of print]

PMID:
31508903
5.

Direct Access to 9-Chloro-1H-benzo[b]furo[3,4-e]azepin-1-ones via Palladium(II)-Catalyzed Intramolecular syn-Oxypalladation/Olefin Insertion/sp2-C-H Bond Activation Cascade.

Karuppasamy M, Vachan BS, Vinoth P, Muthukrishnan I, Nagarajan S, Ielo L, Pace V, Banik S, Maheswari CU, Sridharan V.

Org Lett. 2019 Aug 2;21(15):5784-5788. doi: 10.1021/acs.orglett.9b01482. Epub 2019 Jul 16.

PMID:
31310552
6.

Palladium-Catalyzed Regioselective Syn-Chloropalladation-Olefin Insertion-Oxidative Chlorination Cascade: Synthesis of Dichlorinated Tetrahydroquinolines.

Vinoth P, Karuppasamy M, Vachan BS, Muthukrishnan I, Maheswari CU, Nagarajan S, Pace V, Roller A, Bhuvanesh N, Sridharan V.

Org Lett. 2019 May 3;21(9):3465-3469. doi: 10.1021/acs.orglett.9b01295. Epub 2019 Apr 19.

PMID:
31001984
7.

17O NMR and 15N NMR chemical shifts of sterically-hindered amides: ground-state destabilization in amide electrophilicity.

Pace V, Holzer W, Ielo L, Shi S, Meng G, Hanna M, Szostak R, Szostak M.

Chem Commun (Camb). 2019 Apr 9;55(30):4423-4426. doi: 10.1039/c9cc01402k.

PMID:
30916689
8.

Sustainable Asymmetric Organolithium Chemistry: Enantio- and Chemoselective Acylations through Recycling of Solvent, Sparteine, and Weinreb "Amine".

Monticelli S, Holzer W, Langer T, Roller A, Olofsson B, Pace V.

ChemSusChem. 2019 Mar 21;12(6):1147-1154. doi: 10.1002/cssc.201802815. Epub 2019 Feb 13.

9.

Modular and Chemoselective Strategy for the Direct Access to α-Fluoroepoxides and Aziridines via the Addition of Fluoroiodomethyllithium to Carbonyl-Like Compounds.

Monticelli S, Colella M, Pillari V, Tota A, Langer T, Holzer W, Degennaro L, Luisi R, Pace V.

Org Lett. 2019 Jan 18;21(2):584-588. doi: 10.1021/acs.orglett.8b04001. Epub 2019 Jan 2.

PMID:
30600682
10.

Telescoped, Divergent, Chemoselective C1 and C1-C1 Homologation of Imine Surrogates: Access to Quaternary Chloro- and Halomethyl-Trifluoromethyl Aziridines.

Ielo L, Touqeer S, Roller A, Langer T, Holzer W, Pace V.

Angew Chem Int Ed Engl. 2019 Feb 18;58(8):2479-2484. doi: 10.1002/anie.201812525. Epub 2019 Jan 24.

11.

Chemoselective reduction of isothiocyanates to thioformamides mediated by the Schwartz reagent.

de la Vega-Hernández K, Senatore R, Miele M, Urban E, Holzer W, Pace V.

Org Biomol Chem. 2019 Feb 13;17(7):1970-1978. doi: 10.1039/c8ob02312c.

PMID:
30362485
12.

Design, Synthesis, and Pharmacological Evaluation of Novel β2/3 Subunit-Selective γ-Aminobutyric Acid Type A (GABAA) Receptor Modulators.

Stadler M, Monticelli S, Seidel T, Luger D, Salzer I, Boehm S, Holzer W, Schwarzer C, Urban E, Khom S, Langer T, Pace V, Hering S.

J Med Chem. 2019 Jan 10;62(1):317-341. doi: 10.1021/acs.jmedchem.8b00859. Epub 2018 Oct 23.

PMID:
30289721
13.

Cyclopentyl Methyl Ether: An Elective Ecofriendly Ethereal Solvent in Classical and Modern Organic Chemistry.

Azzena U, Carraro M, Pisano L, Monticelli S, Bartolotta R, Pace V.

ChemSusChem. 2019 Jan 10;12(1):40-70. doi: 10.1002/cssc.201801768. Epub 2018 Nov 20. Review.

14.

Identification of dual Sigma1 receptor modulators/acetylcholinesterase inhibitors with antioxidant and neurotrophic properties, as neuroprotective agents.

Rui M, Rossino G, Coniglio S, Monteleone S, Scuteri A, Malacrida A, Rossi D, Catenacci L, Sorrenti M, Paolillo M, Curti D, Venturini L, Schepmann D, Wünsch B, Liedl KR, Cavaletti G, Pace V, Urban E, Collina S.

Eur J Med Chem. 2018 Oct 5;158:353-370. doi: 10.1016/j.ejmech.2018.09.010. Epub 2018 Sep 8.

PMID:
30223122
15.

Easy as one, two, three.

Castoldi L, Pace V.

Nat Chem. 2018 Nov;10(11):1081-1082. doi: 10.1038/s41557-018-0139-z. No abstract available.

PMID:
30202102
16.

Homologation of halostannanes with carbenoids: a convenient and straightforward one-step access to α-functionalized organotin reagents.

Touqeer S, Castoldi L, Langer T, Holzer W, Pace V.

Chem Commun (Camb). 2018 Sep 6;54(72):10112-10115. doi: 10.1039/c8cc04786c.

PMID:
30124702
17.

A practical guide for using lithium halocarbenoids in homologation reactions.

Monticelli S, Rui M, Castoldi L, Missere G, Pace V.

Monatsh Chem. 2018;149(7):1285-1291. doi: 10.1007/s00706-018-2232-9. Epub 2018 Jun 11.

18.

An unusual thionyl chloride-promoted C-C bond formation to obtain 4,4'-bipyrazolones.

Eller GA, Vilkauskaitė G, Šačkus A, Martynaitis V, Mamuye AD, Pace V, Holzer W.

Beilstein J Org Chem. 2018 Jun 4;14:1287-1292. doi: 10.3762/bjoc.14.110. eCollection 2018.

19.

Homologation chemistry with nucleophilic α-substituted organometallic reagents: chemocontrol, new concepts and (solved) challenges.

Castoldi L, Monticelli S, Senatore R, Ielo L, Pace V.

Chem Commun (Camb). 2018 Jun 19;54(50):6692-6704. doi: 10.1039/c8cc02499e.

PMID:
29850663
20.

Expeditious and Chemoselective Synthesis of α-Aryl and α-Alkyl Selenomethylketones via Homologation Chemistry.

Senatore R, Castoldi L, Ielo L, Holzer W, Pace V.

Org Lett. 2018 May 4;20(9):2685-2688. doi: 10.1021/acs.orglett.8b00896. Epub 2018 Apr 17.

PMID:
29664309

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