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Items: 15


Anti-Inflammatory and Antioxidant Properties of Dehydrated Potato-Derived Bioactive Compounds in Intestinal Cells.

Basilicata MG, Pepe G, Rapa SF, Merciai F, Ostacolo C, Manfra M, Di Sarno V, Autore G, De Vita D, Marzocco S, Campiglia P.

Int J Mol Sci. 2019 Dec 3;20(23). pii: E6087. doi: 10.3390/ijms20236087.


Synthesis and Pharmacological Characterization of Conformationally Restricted Retigabine Analogues as Novel Neuronal Kv7 Channel Activators.

Ostacolo C, Miceli F, Di Sarno V, Nappi P, Iraci N, Soldovieri MV, Ciaglia T, Ambrosino P, Vestuto V, Lauritano A, Musella S, Pepe G, Basilicata MG, Manfra M, Perinelli DR, Novellino E, Bertamino A, Gomez-Monterrey IM, Campiglia P, Taglialatela M.

J Med Chem. 2020 Jan 9;63(1):163-185. doi: 10.1021/acs.jmedchem.9b00796. Epub 2019 Dec 24.


β-Lactoglobulin Heptapeptide Reduces Oxidative Stress in Intestinal Epithelial Cells and Angiotensin II-Induced Vasoconstriction on Mouse Mesenteric Arteries by Induction of Nuclear Factor Erythroid 2-Related Factor 2 (Nrf2) Translocation.

Pepe G, Basilicata MG, Carrizzo A, Adesso S, Ostacolo C, Sala M, Sommella E, Ruocco M, Cascioferro S, Ambrosio M, Pisanti S, Di Sarno V, Bertamino A, Marzocco S, Vecchione C, Campiglia P.

Oxid Med Cell Longev. 2019 Nov 12;2019:1616239. doi: 10.1155/2019/1616239. eCollection 2019.


Towards a new application of amaranth seed oil as an agent against Candida albicans.

De Vita D, Messore A, Toniolo C, Frezza C, Scipione L, Bertea CM, Micera M, Di Sarno V, Madia VN, Pindinello I, Roscilli P, Botto A, Simonetti G, Orekhova A, Manfredini S, Costi R, Di Santo R.

Nat Prod Res. 2019 Dec 4:1-6. doi: 10.1080/14786419.2019.1696335. [Epub ahead of print]


An Efficient Approach to Aromatic Aminomethylation Using Dichloromethane as Methylene Source.

Ostacolo C, Di Sarno V, Musella S, Ciaglia T, Vestuto V, Pepe G, Merciai F, Campiglia P, Gomez Monterrey IM, Bertamino A.

Front Chem. 2019 Aug 13;7:568. doi: 10.3389/fchem.2019.00568. eCollection 2019.


2,6-Disubstituted imidazo[2,1-b][1,3,4]thiadiazole derivatives as potent staphylococcal biofilm inhibitors.

Cascioferro S, Parrino B, Petri GL, Cusimano MG, Schillaci D, Di Sarno V, Musella S, Giovannetti E, Cirrincione G, Diana P.

Eur J Med Chem. 2019 Apr 1;167:200-210. doi: 10.1016/j.ejmech.2019.02.007. Epub 2019 Feb 10.


Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach.

Ostacolo C, Di Sarno V, Lauro G, Pepe G, Musella S, Ciaglia T, Vestuto V, Autore G, Bifulco G, Marzocco S, Campiglia P, Gomez-Monterrey IM, Bertamino A.

Eur J Med Chem. 2019 Apr 1;167:61-75. doi: 10.1016/j.ejmech.2019.01.066. Epub 2019 Feb 6.


New 1,2,4-Oxadiazole Nortopsentin Derivatives with Cytotoxic Activity.

Cascioferro S, Attanzio A, Di Sarno V, Musella S, Tesoriere L, Cirrincione G, Diana P, Parrino B.

Mar Drugs. 2019 Jan 8;17(1). pii: E35. doi: 10.3390/md17010035.


Polyphenolic Extract from Tarocco (Citrus sinensis L. Osbeck) Clone "Lempso" Exerts Anti-Inflammatory and Antioxidant Effects via NF-kB and Nrf-2 Activation in Murine Macrophages.

Pepe G, Sommella E, Cianciarulo D, Ostacolo C, Manfra M, Di Sarno V, Musella S, Russo M, Messore A, Parrino B, Bertamino A, Autore G, Marzocco S, Campiglia P.

Nutrients. 2018 Dec 11;10(12). pii: E1961. doi: 10.3390/nu10121961.


Identification of a Potent Tryptophan-Based TRPM8 Antagonist With in Vivo Analgesic Activity.

Bertamino A, Iraci N, Ostacolo C, Ambrosino P, Musella S, Di Sarno V, Ciaglia T, Pepe G, Sala M, Soldovieri MV, Mosca I, Gonzalez-Rodriguez S, Fernandez-Carvajal A, Ferrer-Montiel A, Novellino E, Taglialatela M, Campiglia P, Gomez-Monterrey I.

J Med Chem. 2018 Jul 26;61(14):6140-6152. doi: 10.1021/acs.jmedchem.8b00545. Epub 2018 Jul 10.


Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds.

Bertamino A, Lauro G, Ostacolo C, Di Sarno V, Musella S, Ciaglia T, Campiglia P, Bifulco G, Gomez-Monterrey IM.

J Org Chem. 2017 Dec 1;82(23):12014-12027. doi: 10.1021/acs.joc.7b01656. Epub 2017 Nov 14.


Identification of an indol-based derivative as potent and selective varicella zoster virus (VZV) inhibitor.

Musella S, di Sarno V, Ciaglia T, Sala M, Spensiero A, Scala MC, Ostacolo C, Andrei G, Balzarini J, Snoeck R, Novellino E, Campiglia P, Bertamino A, Gomez-Monterrey IM.

Eur J Med Chem. 2016 Nov 29;124:773-781. doi: 10.1016/j.ejmech.2016.09.014. Epub 2016 Sep 7.


Tryptamine-Based Derivatives as Transient Receptor Potential Melastatin Type 8 (TRPM8) Channel Modulators.

Bertamino A, Ostacolo C, Ambrosino P, Musella S, Di Sarno V, Ciaglia T, Soldovieri MV, Iraci N, Fernandez Carvajal A, de la Torre-Martinez R, Ferrer-Montiel A, Gonzalez Muniz R, Novellino E, Taglialatela M, Campiglia P, Gomez-Monterrey I.

J Med Chem. 2016 Mar 10;59(5):2179-91. doi: 10.1021/acs.jmedchem.5b01914. Epub 2016 Feb 17.


Dihydrithieno[2,3-b]naphto-4,9-dione analogues as anticancer agents: Synthesis and in cell pharmacological studies.

Bertamino A, Musella S, Di Sarno V, Ostacolo C, Manfra M, Vanacore D, Stiuso P, Novellino E, Campiglia P, Gomez-Monterrey IM.

Eur J Med Chem. 2015 Sep 18;102:106-14. doi: 10.1016/j.ejmech.2015.07.044. Epub 2015 Jul 26.


Synthesis, in vitro, and in cell studies of a new series of [indoline-3,2'-thiazolidine]-based p53 modulators.

Bertamino A, Soprano M, Musella S, Rusciano MR, Sala M, Vernieri E, Di Sarno V, Limatola A, Carotenuto A, Cosconati S, Grieco P, Novellino E, Illario M, Campiglia P, Gomez-Monterrey I.

J Med Chem. 2013 Jul 11;56(13):5407-21. doi: 10.1021/jm400311n. Epub 2013 Jun 26.


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