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Items: 1 to 20 of 68

1.

Neuromedin U and Structural Analogs: an Overview of Their Structure, Function and Selectivity.

De Prins A, Van Eeckhaut A, Smolders I, Tourwé D, Ballet S.

Curr Med Chem. 2019 Sep 16. doi: 10.2174/0929867326666190916143028. [Epub ahead of print]

PMID:
31526341
2.

Primary hepatocytes and their cultures for the testing of drug-induced liver injury.

Vilas-Boas V, Cooreman A, Gijbels E, Van Campenhout R, Gustafson E, Ballet S, Annaert P, Cogliati B, Vinken M.

Adv Pharmacol. 2019;85:1-30. doi: 10.1016/bs.apha.2018.08.001. Epub 2018 Sep 1.

PMID:
31307583
3.

The 1,3-diyne linker as a rigid "i,i+7" staple for α-helix stabilization: Stereochemistry at work.

Verlinden S, Geudens N, Van Holsbeeck K, Mannes M, Martins JC, Verniest G, Ballet S.

J Pept Sci. 2019 Jul;25(7):e3194. doi: 10.1002/psc.3194. Epub 2019 Jun 18.

PMID:
31215108
4.

Trifluoromethylated Proline Surrogates as Part of "Pro-Pro" Turn-Inducing Templates.

Gadais C, Van Holsbeeck K, Moors SLC, Buyst D, Fehér K, Van Hecke K, Tourwé D, Brigaud T, Martin C, De Proft F, Pytkowicz J, Martins JC, Chaume G, Ballet S.

Chembiochem. 2019 May 6. doi: 10.1002/cbic.201900294. [Epub ahead of print]

PMID:
31062451
5.

Solid-Phase Azopeptide Diels-Alder Chemistry for Aza-pipecolyl Residue Synthesis To Study Peptide Conformation.

Chingle R, Mulumba M, Chung NN, Nguyen TM, Ong H, Ballet S, Schiller PW, Lubell WD.

J Org Chem. 2019 May 17;84(10):6006-6016. doi: 10.1021/acs.joc.8b03283. Epub 2019 Apr 26.

PMID:
30957495
6.

Biodegradable Amphipathic Peptide Hydrogels as Extended-Release System for Opioid Peptides.

Martin C, Dumitrascuta M, Mannes M, Lantero A, Bucher D, Walker K, Van Wanseele Y, Oyen E, Hernot S, Van Eeckhaut A, Madder A, Hoogenboom R, Spetea M, Ballet S.

J Med Chem. 2018 Nov 8;61(21):9784-9789. doi: 10.1021/acs.jmedchem.8b01282. Epub 2018 Oct 26.

PMID:
30351003
7.

Connexin and Pannexin (Hemi)Channels: Emerging Targets in the Treatment of Liver Disease.

Cooreman A, Van Campenhout R, Ballet S, Annaert P, Van Den Bossche B, Colle I, Cogliati B, Vinken M.

Hepatology. 2019 Mar;69(3):1317-1323. doi: 10.1002/hep.30306. Epub 2019 Feb 23. Review.

PMID:
30300925
8.

Radiometal-labeled anti-VCAM-1 nanobodies as molecular tracers for atherosclerosis - impact of radiochemistry on pharmacokinetics.

Bala G, Crauwels M, Blykers A, Remory I, Marschall ALJ, Dübel S, Dumas L, Broisat A, Martin C, Ballet S, Cosyns B, Caveliers V, Devoogdt N, Xavier C, Hernot S.

Biol Chem. 2019 Feb 25;400(3):323-332. doi: 10.1515/hsz-2018-0330.

PMID:
30240352
9.

The Neurokinins: Peptidomimetic Ligand Design and Therapeutic Applications.

Gadais C, Ballet S.

Curr Med Chem. 2018 Sep 12. doi: 10.2174/0929867325666180913095918. [Epub ahead of print]

PMID:
30209994
10.

Site-Specific Radioactive Labeling of Nanobodies.

Crauwels M, Massa S, Martin C, Betti C, Ballet S, Devoogdt N, Xavier C, Muyldermans S.

Methods Mol Biol. 2018;1827:505-540. doi: 10.1007/978-1-4939-8648-4_26.

PMID:
30196514
11.

Corrigendum to "Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings" [Bioorg. Med. Chem. Lett. 28(13) (2018) 2320-2323].

Willemse T, Eiselt E, Hollanders K, Schepens W, van Vlijmen HWT, Chung NN, Blais V, Holleran B, Longpré JM, Schiller PW, Maes BUW, Sarret P, Gendron L, Ballet S.

Bioorg Med Chem Lett. 2018 Nov 1;28(20):3418. doi: 10.1016/j.bmcl.2018.08.023. Epub 2018 Sep 5. No abstract available.

PMID:
30195888
12.

Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings.

Willemse T, Eiselt E, Hollanders K, Schepens W, van Vlijmen HWT, Chung NN, Blais V, Holleran B, Longpré JM, Schiller PW, Maes BUW, Sarret P, Gendron L, Ballet S.

Bioorg Med Chem Lett. 2018 Jul 15;28(13):2320-2323. doi: 10.1016/j.bmcl.2018.05.015. Epub 2018 May 12. Erratum in: Bioorg Med Chem Lett. 2018 Nov 1;28(20):3418.

13.

Synthesis and in Vitro Evaluation of Stabilized and Selective Neuromedin U-1 Receptor Agonists.

De Prins A, Martin C, Van Wanseele Y, Tömböly C, Tourwé D, Caveliers V, Holst B, Van Eeckhaut A, Rosenkilde MM, Smolders I, Ballet S.

ACS Med Chem Lett. 2018 Apr 23;9(5):496-501. doi: 10.1021/acsmedchemlett.8b00105. eCollection 2018 May 10.

14.

A bifunctional-biased mu-opioid agonist-neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects.

Drieu la Rochelle A, Guillemyn K, Dumitrascuta M, Martin C, Utard V, Quillet R, Schneider S, Daubeuf F, Willemse T, Mampuys P, Maes BUW, Frossard N, Bihel F, Spetea M, Simonin F, Ballet S.

Pain. 2018 Sep;159(9):1705-1718. doi: 10.1097/j.pain.0000000000001262.

PMID:
29708942
15.

Bromotryptophans and their incorporation in cyclic and bicyclic privileged peptides.

García-Pindado J, Willemse T, Goss R, Maes BUW, Giralt E, Ballet S, Teixidó M.

Biopolymers. 2018 Aug;109(10):e23112. doi: 10.1002/bip.23112. Epub 2018 Mar 12.

16.

Nanobody-Enabled Reverse Pharmacology on G-Protein-Coupled Receptors.

Pardon E, Betti C, Laeremans T, Chevillard F, Guillemyn K, Kolb P, Ballet S, Steyaert J.

Angew Chem Int Ed Engl. 2018 May 4;57(19):5292-5295. doi: 10.1002/anie.201712581. Epub 2018 Mar 30.

PMID:
29469969
17.

Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain-Barrier-Permeating Compounds.

Van der Poorten O, Legrand B, Vezenkov LL, García-Pindado J, Bettache N, Knuhtsen A, Pedersen DS, Sánchez-Navarro M, Martinez J, Teixidó M, Garcia M, Tourwé D, Amblard M, Ballet S.

Chembiochem. 2018 Apr 4;19(7):696-705. doi: 10.1002/cbic.201700678. Epub 2018 Feb 28.

PMID:
29377388
18.

Binding-Site Compatible Fragment Growing Applied to the Design of β2-Adrenergic Receptor Ligands.

Chevillard F, Rimmer H, Betti C, Pardon E, Ballet S, van Hilten N, Steyaert J, Diederich WE, Kolb P.

J Med Chem. 2018 Feb 8;61(3):1118-1129. doi: 10.1021/acs.jmedchem.7b01558. Epub 2018 Jan 24.

PMID:
29364664
19.

Development of potent and proteolytically stable human neuromedin U receptor agonists.

De Prins A, Martin C, Van Wanseele Y, Skov LJ, Tömböly C, Tourwé D, Caveliers V, Van Eeckhaut A, Holst B, Rosenkilde MM, Smolders I, Ballet S.

Eur J Med Chem. 2018 Jan 20;144:887-897. doi: 10.1016/j.ejmech.2017.12.035. Epub 2017 Dec 14.

PMID:
29329072
20.

χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds.

Van der Poorten O, Van Den Hauwe R, Eiselt E, Betti C, Guillemyn K, Chung NN, Hallé F, Bihel F, Schiller PW, Tourwé D, Sarret P, Gendron L, Ballet S.

ACS Med Chem Lett. 2017 Oct 4;8(11):1177-1182. doi: 10.1021/acsmedchemlett.7b00347. eCollection 2017 Nov 9.

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