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Items: 1 to 20 of 85

1.

New insights into the opening of the occluded ligand-binding pocket of Sigma1 receptor: binding of a novel bivalent RC-33 derivative.

Rossino G, Orellana I, Caballero J, Schepmann D, Wünsch B, Rui M, Rossi D, Gonzalez-Avendaño M, Collina S, Vergara-Jaque A.

J Chem Inf Model. 2019 Dec 6. doi: 10.1021/acs.jcim.9b00649. [Epub ahead of print]

PMID:
31809025
2.

Technological Competence Is a Pre-condition for Effective Implementation of Virtual Reality Head Mounted Displays in Human Neuroscience: A Technological Review and Meta-Analysis.

Kourtesis P, Collina S, Doumas LAA, MacPherson SE.

Front Hum Neurosci. 2019 Oct 2;13:342. doi: 10.3389/fnhum.2019.00342. eCollection 2019.

3.

Scope and Limitations of Boron Fluorescent Complexes from Stable Nitrile Oxides in ABPP Assays.

Moiola M, Crespi S, Memeo M, Collina S, Overkleeft H, Florea B, Quadrelli P.

ACS Omega. 2019 Apr 29;4(4):7766-7774. doi: 10.1021/acsomega.9b00672. eCollection 2019 Apr 30.

4.

Docking, Interaction Fingerprint, and Three-Dimensional Quantitative Structure-Activity Relationship (3D-QSAR) of Sigma1 Receptor Ligands, Analogs of the Neuroprotective Agent RC-33.

Velázquez-Libera JL, Rossino G, Navarro-Retamal C, Collina S, Caballero J.

Front Chem. 2019 Jul 11;7:496. doi: 10.3389/fchem.2019.00496. eCollection 2019.

5.

Anti-Multiple Myeloma Potential of Secondary Metabolites from Hibiscus sabdariffa.

Malacrida A, Cavalloro V, Martino E, Cassetti A, Nicolini G, Rigolio R, Cavaletti G, Mannucci B, Vasile F, Giacomo MD, Collina S, Miloso M.

Molecules. 2019 Jul 9;24(13). pii: E2500. doi: 10.3390/molecules24132500.

6.

Discovery of new potent dual sigma receptor/GluN2b ligands with antioxidant property as neuroprotective agents.

Zampieri D, Fortuna S, Calabretti A, Romano M, Menegazzi R, Schepmann D, Wünsch B, Collina S, Zanon D, Mamolo MG.

Eur J Med Chem. 2019 Oct 15;180:268-282. doi: 10.1016/j.ejmech.2019.07.012. Epub 2019 Jul 8.

PMID:
31319263
7.

Artemisinin and its derivatives; ancient tradition inspiring the latest therapeutic approaches against malaria.

Martino E, Tarantino M, Bergamini M, Castelluccio V, Coricello A, Falcicchio M, Lorusso E, Collina S.

Future Med Chem. 2019 Jun;11(12):1443-1459. doi: 10.4155/fmc-2018-0337. Epub 2019 Jul 12.

PMID:
31298579
8.

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5.

Mangoni AA, Eynde JJV, Jampilek J, Hadjipavlou-Litina D, Liu H, Reynisson J, Sousa ME, Gomes PAC, Prokai-Tatrai K, Tuccinardi T, Sabatier JM, Luque FJ, Rautio J, Karaman R, Vasconcelos MH, Gemma S, Galdiero S, Hulme C, Collina S, Gütschow M, Kokotos G, Siciliano C, Capasso R, Agrofoglio LA, Ragno R, Muñoz-Torrero D.

Molecules. 2019 Jun 30;24(13). pii: E2415. doi: 10.3390/molecules24132415.

9.

Anti-tumor Efficacy Assessment of the Sigma Receptor Pan Modulator RC-106. A Promising Therapeutic Tool for Pancreatic Cancer.

Tesei A, Cortesi M, Pignatta S, Arienti C, Dondio GM, Bigogno C, Malacrida A, Miloso M, Meregalli C, Chiorazzi A, Carozzi V, Cavaletti G, Rui M, Marra A, Rossi D, Collina S.

Front Pharmacol. 2019 May 14;10:490. doi: 10.3389/fphar.2019.00490. eCollection 2019.

10.

Novel Compounds Targeting the RNA-Binding Protein HuR. Structure-Based Design, Synthesis, and Interaction Studies.

Della Volpe S, Nasti R, Queirolo M, Unver MY, Jumde VK, Dömling A, Vasile F, Potenza D, Ambrosio FA, Costa G, Alcaro S, Zucal C, Provenzani A, Di Giacomo M, Rossi D, Hirsch AKH, Collina S.

ACS Med Chem Lett. 2019 Jan 21;10(4):615-620. doi: 10.1021/acsmedchemlett.8b00600. eCollection 2019 Apr 11.

PMID:
30996806
11.

DHFR Inhibitors: Reading the Past for Discovering Novel Anticancer Agents.

Raimondi MV, Randazzo O, La Franca M, Barone G, Vignoni E, Rossi D, Collina S.

Molecules. 2019 Mar 22;24(6). pii: E1140. doi: 10.3390/molecules24061140. Review.

12.

Development of a Mucoadhesive and an in Situ Gelling Formulation Based on κ-Carrageenan for Application on Oral Mucosa and Esophagus Walls. II. Loading of a Bioactive Hydroalcoholic Extract.

Vigani B, Rossi S, Gentile M, Sandri G, Bonferoni MC, Cavalloro V, Martino E, Collina S, Ferrari F.

Mar Drugs. 2019 Mar 5;17(3). pii: E153. doi: 10.3390/md17030153.

13.

DPD-Inspired Discovery of Novel LsrK Kinase Inhibitors: An Opportunity To Fight Antimicrobial Resistance.

Stotani S, Gatta V, Medarametla P, Padmanaban M, Karawajczyk A, Giordanetto F, Tammela P, Laitinen T, Poso A, Tzalis D, Collina S.

J Med Chem. 2019 Mar 14;62(5):2720-2737. doi: 10.1021/acs.jmedchem.9b00025. Epub 2019 Mar 4.

PMID:
30786203
14.

Pyrrolomycins as antimicrobial agents. Microwave-assisted organic synthesis and insights into their antimicrobial mechanism of action.

Raimondi MV, Listro R, Cusimano MG, La Franca M, Faddetta T, Gallo G, Schillaci D, Collina S, Leonchiks A, Barone G.

Bioorg Med Chem. 2019 Mar 1;27(5):721-728. doi: 10.1016/j.bmc.2019.01.010. Epub 2019 Jan 16.

PMID:
30711310
15.

The use of a microwave-assisted solvent extraction coupled with HPLC-UV/PAD to assess the quality of Marrubium vulgare L. (white horehound) herbal raw material.

Martino E, Della Volpe S, Cavalloro V, Amri B, Kaab LBB, Marrubini G, Rossi D, Collina S.

Phytochem Anal. 2019 Jul;30(4):377-384. doi: 10.1002/pca.2820. Epub 2019 Jan 27.

PMID:
30687967
16.

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes⁻4.

Mangoni AA, Guillou C, Vanden Eynde JJ, Hulme C, Jampilek J, Li W, Prokai-Tatrai K, Rautio J, Collina S, Tuccinardi T, Sousa ME, Sabatier JM, Galdiero S, Karaman R, Kokotos G, Torri G, Luque FJ, Vasconcelos MH, Hadjipavlou-Litina D, Siciliano C, Gütschow M, Ragno R, Gomes PAC, Agrofoglio LA, Muñoz-Torrero D.

Molecules. 2018 Dec 31;24(1). pii: E130. doi: 10.3390/molecules24010130.

17.

A Versatile Strategy for the Synthesis of 4,5-Dihydroxy-2,3-Pentanedione (DPD) and Related Compounds as Potential Modulators of Bacterial Quorum Sensing.

Stotani S, Gatta V, Medda F, Padmanaban M, Karawajczyk A, Tammela P, Giordanetto F, Tzalis D, Collina S.

Molecules. 2018 Oct 6;23(10). pii: E2545. doi: 10.3390/molecules23102545.

18.

Identification of dual Sigma1 receptor modulators/acetylcholinesterase inhibitors with antioxidant and neurotrophic properties, as neuroprotective agents.

Rui M, Rossino G, Coniglio S, Monteleone S, Scuteri A, Malacrida A, Rossi D, Catenacci L, Sorrenti M, Paolillo M, Curti D, Venturini L, Schepmann D, Wünsch B, Liedl KR, Cavaletti G, Pace V, Urban E, Collina S.

Eur J Med Chem. 2018 Oct 5;158:353-370. doi: 10.1016/j.ejmech.2018.09.010. Epub 2018 Sep 8.

PMID:
30223122
19.

Exploration of ligand binding modes towards the identification of compounds targeting HuR: a combined STD-NMR and Molecular Modelling approach.

Vasile F, Della Volpe S, Ambrosio FA, Costa G, Unver MY, Zucal C, Rossi D, Martino E, Provenzani A, Hirsch AKH, Alcaro S, Potenza D, Collina S.

Sci Rep. 2018 Sep 13;8(1):13780. doi: 10.1038/s41598-018-32084-z.

20.

Vinca alkaloids and analogues as anti-cancer agents: Looking back, peering ahead.

Martino E, Casamassima G, Castiglione S, Cellupica E, Pantalone S, Papagni F, Rui M, Siciliano AM, Collina S.

Bioorg Med Chem Lett. 2018 Sep 15;28(17):2816-2826. doi: 10.1016/j.bmcl.2018.06.044. Epub 2018 Jun 25. Review.

PMID:
30122223

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