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Items: 1 to 20 of 107

1.

1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors.

D'Ascenzio M, Secci D, Carradori S, Zara S, Guglielmi P, Cirilli R, Pierini M, Poli G, Tuccinardi T, Angeli A, Supuran CT.

J Med Chem. 2020 Feb 4. doi: 10.1021/acs.jmedchem.9b01434. [Epub ahead of print]

PMID:
31972093
2.

Temperature and eluent composition effects on enantiomer separation of carvedilol by high-performance liquid chromatography on immobilized amylose-based chiral stationary phases.

Panella C, Ferretti R, Casulli A, Cirilli R.

J Pharm Anal. 2019 Oct;9(5):324-331. doi: 10.1016/j.jpha.2019.04.002. Epub 2019 Apr 4.

3.

The Benzimidazole-Based Anthelmintic Parbendazole: A Repurposed Drug Candidate That Synergizes with Gemcitabine in Pancreatic Cancer.

Florio R, Veschi S, di Giacomo V, Pagotto S, Carradori S, Verginelli F, Cirilli R, Casulli A, Grassadonia A, Tinari N, Cataldi A, Amoroso R, Cama A, De Lellis L.

Cancers (Basel). 2019 Dec 17;11(12). pii: E2042. doi: 10.3390/cancers11122042.

4.

High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase.

Carradori S, Secci D, Guglielmi P, Pierini M, Cirilli R.

J Chromatogr A. 2020 Jan 11;1610:460572. doi: 10.1016/j.chroma.2019.460572. Epub 2019 Sep 27.

PMID:
31606155
5.

Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold.

Rotondi G, Guglielmi P, Carradori S, Secci D, De Monte C, De Filippis B, Maccallini C, Amoroso R, Cirilli R, Akdemir A, Angeli A, Supuran CT.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):1400-1413. doi: 10.1080/14756366.2019.1651315.

6.

TetraPh-Tol-BITIOPO: a new atropisomeric 3,3'-bithiophene based phosphine oxide as an organocatalyst in Lewis base-catalyzed Lewis acid mediated reactions.

Mirco AV, Maurizio B, Sergio R, Tiziana B, Roberto C, Marco P.

Org Biomol Chem. 2019 Aug 28;17(32):7474-7481. doi: 10.1039/c9ob01297d. Epub 2019 Jul 30.

PMID:
31361281
7.

HPLC Enantioseparations with Polysaccharide-Based Chiral Stationary Phases in HILIC Conditions.

Cirilli R.

Methods Mol Biol. 2019;1985:127-146. doi: 10.1007/978-1-4939-9438-0_7.

PMID:
31069732
8.

Highlighting spin selectivity properties of chiral electrode surfaces from redox potential modulation of an achiral probe under an applied magnetic field.

Benincori T, Arnaboldi S, Magni M, Grecchi S, Cirilli R, Fontanesi C, Mussini PR.

Chem Sci. 2019 Jan 4;10(9):2750-2757. doi: 10.1039/c8sc04126a. eCollection 2019 Mar 7.

9.

Highly enantioselective "inherently chiral" electroactive materials based on a 2,2'-biindole atropisomeric scaffold.

Arnaboldi S, Benincori T, Penoni A, Vaghi L, Cirilli R, Abbate S, Longhi G, Mazzeo G, Grecchi S, Panigati M, Mussini PR.

Chem Sci. 2019 Jan 5;10(9):2708-2717. doi: 10.1039/c8sc04862b. eCollection 2019 Mar 7.

10.

Design, Synthesis, Docking Studies and Monoamine Oxidase Inhibition of a Small Library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazoles.

Guglielmi P, Carradori S, Poli G, Secci D, Cirilli R, Rotondi G, Chimenti P, Petzer A, Petzer JP.

Molecules. 2019 Jan 29;24(3). pii: E484. doi: 10.3390/molecules24030484.

11.

Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1 H-pyrrolyl)(phenyl)methyl-1 H-imidazole Derivatives as Antiprotozoal Agents.

Saccoliti F, Madia VN, Tudino V, De Leo A, Pescatori L, Messore A, De Vita D, Scipione L, Brun R, Kaiser M, Mäser P, Calvet CM, Jennings GK, Podust LM, Pepe G, Cirilli R, Faggi C, Di Marco A, Battista MR, Summa V, Costi R, Di Santo R.

J Med Chem. 2019 Feb 14;62(3):1330-1347. doi: 10.1021/acs.jmedchem.8b01464. Epub 2019 Jan 23.

PMID:
30615444
12.

Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells.

Stazi G, Battistelli C, Piano V, Mazzone R, Marrocco B, Marchese S, Louie SM, Zwergel C, Antonini L, Patsilinakos A, Ragno R, Viviano M, Sbardella G, Ciogli A, Fabrizi G, Cirilli R, Strippoli R, Marchetti A, Tripodi M, Nomura DK, Mattevi A, Mai A, Valente S.

Eur J Med Chem. 2019 Feb 1;163:722-735. doi: 10.1016/j.ejmech.2018.11.050. Epub 2018 Nov 28.

PMID:
30576903
13.

Effect of α-Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3 H)-ones.

Nawrozkij MB, Forgione M, Yablokov AS, Lucidi A, Tomaselli D, Patsilinakos A, Panella C, Hailu GS, Kirillov IA, Badia R, Riveira-Muñoz E, Crespan E, Armijos Rivera JI, Cirilli R, Ragno R, Esté JA, Maga G, Mai A, Rotili D.

J Med Chem. 2019 Jan 24;62(2):604-621. doi: 10.1021/acs.jmedchem.8b01238. Epub 2018 Dec 20.

PMID:
30525601
14.

A chromatographic study on the retention behavior of the amylose tris(3-chloro-5-methylphenylcarbamate) chiral stationary phase under aqueous conditions.

Cirilli R, Carradori S, Casulli A, Pierini M.

J Sep Sci. 2018 Nov;41(21):4014-4021. doi: 10.1002/jssc.201800696. Epub 2018 Oct 1.

PMID:
30194899
15.

Structure-Based Drug Design of Potent Pyrazole Derivatives against Rhinovirus Replication.

Da Costa L, Scheers E, Coluccia A, Casulli A, Roche M, Di Giorgio C, Neyts J, Terme T, Cirilli R, La Regina G, Silvestri R, Mirabelli C, Vanelle P.

J Med Chem. 2018 Sep 27;61(18):8402-8416. doi: 10.1021/acs.jmedchem.8b00931. Epub 2018 Sep 7.

PMID:
30153009
16.

Unusual retention behavior of omeprazole and its chiral impurities B and E on the amylose tris (3-chloro-5-methylphenylcarbamate) chiral stationary phase in polar organic mode.

Ferretti R, Zanitti L, Casulli A, Cirilli R.

J Pharm Anal. 2018 Aug;8(4):234-239. doi: 10.1016/j.jpha.2018.04.001. Epub 2018 Apr 20.

17.

Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors.

Talapatra SK, Tham CL, Guglielmi P, Cirilli R, Chandrasekaran B, Karpoormath R, Carradori S, Kozielski F.

Eur J Med Chem. 2018 Aug 5;156:641-651. doi: 10.1016/j.ejmech.2018.07.006. Epub 2018 Jul 4.

PMID:
30031975
18.

Searching for Models Exhibiting High Circularly Polarized Luminescence: Electroactive Inherently Chiral Oligothiophenes.

Benincori T, Appoloni G, Mussini PR, Arnaboldi S, Cirilli R, Quartapelle Procopio E, Panigati M, Abbate S, Mazzeo G, Longhi G.

Chemistry. 2018 Aug 1;24(43):11082-11093. doi: 10.1002/chem.201801158. Epub 2018 Jul 2.

PMID:
29719070
19.

Progress in the pharmacological treatment of human cystic and alveolar echinococcosis: Compounds and therapeutic targets.

Siles-Lucas M, Casulli A, Cirilli R, Carmena D.

PLoS Negl Trop Dis. 2018 Apr 20;12(4):e0006422. doi: 10.1371/journal.pntd.0006422. eCollection 2018 Apr.

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