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Items: 1 to 20 of 178

1.

Chalcones and Five-Membered Heterocyclic Isosteres Bind to Alpha Synuclein Fibrils in Vitro.

Hsieh CJ, Xu K, Lee I, Graham TJA, Tu Z, Dhavale D, Kotzbauer P, Mach RH.

ACS Omega. 2018 Apr 30;3(4):4486-4493. doi: 10.1021/acsomega.7b01897. Epub 2018 Apr 24.

2.

Altering Nitrogen Heterocycles of AZD2461 Affords High Affinity Poly(ADP-ribose) Polymerase-1 Inhibitors with Decreased P-Glycoprotein Interactions.

Reilly SW, Puentes LN, Hsieh CJ, Makvandi M, Mach RH.

ACS Omega. 2018 Aug 31;3(8):9997-10001. doi: 10.1021/acsomega.8b00896. Epub 2018 Aug 28.

3.

Analogues of Arylamide Phenylpiperazine Ligands To Investigate the Factors Influencing D3 Dopamine Receptor Bitropic Binding and Receptor Subtype Selectivity.

Hayatshahi HS, Xu K, Griffin SA, Taylor M, Mach RH, Liu J, Luedtke RR.

ACS Chem Neurosci. 2018 Jul 30. doi: 10.1021/acschemneuro.8b00142. [Epub ahead of print]

PMID:
30010318
4.

Examination of Diazaspiro Cores as Piperazine Bioisosteres in the Olaparib Framework Shows Reduced DNA Damage and Cytotoxicity.

Reilly SW, Puentes LN, Wilson K, Hsieh CJ, Weng CC, Makvandi M, Mach RH.

J Med Chem. 2018 Jun 28;61(12):5367-5379. doi: 10.1021/acs.jmedchem.8b00576. Epub 2018 Jun 14.

PMID:
29856625
5.

Dopamine D3 receptor partial agonist LS-3-134 attenuates cocaine-motivated behaviors.

Powell GL, Bonadonna JP, Vannan A, Xu K, Mach RH, Luedtke RR, Neisewander JL.

Pharmacol Biochem Behav. 2018 Aug;171:46-53. doi: 10.1016/j.pbb.2018.05.015. Epub 2018 May 25.

PMID:
29807065
6.

Alpha Synuclein Fibrils Contain Multiple Binding Sites for Small Molecules.

Hsieh CJ, Ferrie JJ, Xu K, Lee I, Graham TJA, Tu Z, Yu J, Dhavale D, Kotzbauer P, Petersson EJ, Mach RH.

ACS Chem Neurosci. 2018 May 16. doi: 10.1021/acschemneuro.8b00177. [Epub ahead of print]

PMID:
29750499
7.

Letter to the Editor: International Consensus Radiochemistry Nomenclature Guidelines.

Coenen HH, Gee AD, Adam M, Antoni G, Cutler CS, Fujibayashi Y, Jeong JM, Mach RH, Mindt TL, Pike VW, Windhorst AD.

Curr Radiopharm. 2018;11(1):73-75. doi: 10.2174/187447101101180404111248. No abstract available.

PMID:
29624156
8.

Rapid Cu-Catalyzed [211At]Astatination and [125I]Iodination of Boronic Esters at Room Temperature.

Reilly SW, Makvandi M, Xu K, Mach RH.

Org Lett. 2018 Apr 6;20(7):1752-1755. doi: 10.1021/acs.orglett.8b00232. Epub 2018 Mar 21.

PMID:
29561158
9.

International Consensus Radiochemistry Nomenclature Guidelines.

Coenen HH, Gee AD, Adam M, Antoni G, Cutler CS, Fujibayashi Y, Jeong JM, Mach RH, Mindt TL, Pike VW, Windhorst AD.

Nuklearmedizin. 2018 Feb;57(1):40-41. doi: 10.1055/s-0038-1636563. Epub 2018 Feb 21. No abstract available.

PMID:
29536500
10.

Open letter to journal editors on: international consensus radiochemistry nomenclature guidelines.

Coenen HH, Gee AD, Adam M, Antoni G, Cutler CS, Fujibayashi Y, Jeong JM, Mach RH, Mindt TL, Pike VW, Windhorst AD.

Am J Nucl Med Mol Imaging. 2018 Feb 5;8(1):70-72. eCollection 2018. No abstract available.

11.

Selectivity of probes for PET imaging of dopamine D3 receptors.

Doot RK, Dubroff JG, Labban KJ, Mach RH.

Neurosci Lett. 2018 Mar 5. pii: S0304-3940(18)30175-7. doi: 10.1016/j.neulet.2018.03.006. [Epub ahead of print] Review.

PMID:
29518538
12.

PET Imaging of Microglial Activation-Beyond Targeting TSPO.

Janssen B, Vugts DJ, Windhorst AD, Mach RH.

Molecules. 2018 Mar 8;23(3). pii: E607. doi: 10.3390/molecules23030607. Review.

13.

A PET imaging agent for evaluating PARP-1 expression in ovarian cancer.

Makvandi M, Pantel A, Schwartz L, Schubert E, Xu K, Hsieh CJ, Hou C, Kim H, Weng CC, Winters H, Doot R, Farwell MD, Pryma DA, Greenberg RA, Mankoff DA, Simpkins F, Mach RH, Lin LL.

J Clin Invest. 2018 May 1;128(5):2116-2126. doi: 10.1172/JCI97992. Epub 2018 Apr 16.

14.

Design, synthesis, and in vitro evaluation of quinolinyl analogues for α-synuclein aggregation.

Yue X, Dhavale DD, Li J, Luo Z, Liu J, Yang H, Mach RH, Kotzbauer PT, Tu Z.

Bioorg Med Chem Lett. 2018 Apr 1;28(6):1011-1019. doi: 10.1016/j.bmcl.2018.02.031. Epub 2018 Feb 16.

PMID:
29482941
15.

Synthesis and pharmacological evaluation of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives as sigma-2 receptor ligands.

Sun YT, Wang GF, Yang YQ, Jin F, Wang Y, Xie XY, Mach RH, Huang YS.

Eur J Med Chem. 2018 Mar 10;147:227-237. doi: 10.1016/j.ejmech.2017.11.016. Epub 2017 Nov 9.

PMID:
29438891
16.

Open letter to journal editors on: International Consensus Radiochemistry Nomenclature Guidelines.

Coenen HH, Gee AD, Adam M, Antoni G, Cutler CS, Fujibayashi Y, Jeong JM, Mach RH, Mindt TL, Pike VW, Windhorst AD.

Nucl Med Commun. 2018 Mar;39(3):193-195. doi: 10.1097/MNM.0000000000000799. No abstract available.

PMID:
29438216
17.

Open letter to journal editors on: International Consensus Radiochemistry Nomenclature Guidelines.

Coenen HH, Gee AD, Adam M, Antoni G, Cutler CS, Fujibayashi Y, Jeong JM, Mach RH, Mindt TL, Pike VW, Windhorst AD.

Ann Nucl Med. 2018 Apr;32(3):236-238. doi: 10.1007/s12149-018-1238-z. Epub 2018 Feb 8. No abstract available.

18.

Open letter to journal editors on: International consensus radiochemistry nomenclature guidelines.

Coenen HH, Gee AD, Adam M, Antoni G, Cutler CS, Fujibayashi Y, Jeong JM, Mach RH, Mindt TL, Pike VW, Windhorst AD.

J Labelled Comp Radiopharm. 2018 Apr;61(4):402-404. doi: 10.1002/jlcr.3604. No abstract available.

PMID:
29331022
19.

Copper Loading of Preformed Nanoparticles for PET-Imaging Applications.

Lu HD, Wang LZ, Wilson BK, McManus SA, Jumai'an J, Padakanti PK, Alavi A, Mach RH, Prud'homme RK.

ACS Appl Mater Interfaces. 2018 Jan 31;10(4):3191-3199. doi: 10.1021/acsami.7b07242. Epub 2018 Jan 17.

PMID:
29272577
20.

Inflammation and DNA damage: Probing pathways to cancer and neurodegeneration.

Makvandi M, Sellmyer MA, Mach RH.

Drug Discov Today Technol. 2017 Nov;25:37-43. doi: 10.1016/j.ddtec.2017.11.001. Epub 2017 Nov 22. Review.

PMID:
29233266

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