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Items: 1 to 20 of 36

1.

New N-(2-phenyl-4-oxo-1,3-thiazolidin-3-yl)-1,2-benzothiazole-3-carboxamides and acetamides as antimicrobial agents.

Incerti M, Vicini P, Geronikaki A, Eleftheriou P, Tsagkadouras A, Zoumpoulakis P, Fotakis C, Ćirić A, Glamočlija J, Soković M.

Medchemcomm. 2017 Nov 3;8(11):2142-2154. doi: 10.1039/c7md00334j. eCollection 2017 Nov 1.

2.

4-Thiazolidinone Derivatives as MMP Inhibitors in Tissue Damage: Synthesis, Biological Evaluation and Docking Studies.

Incerti M, Crascì L, Vicini P, Aki E, Yalcin I, Ertan-Bolelli T, Cardile V, Graziano ACE, Panico A.

Molecules. 2018 Feb 14;23(2). pii: E415. doi: 10.3390/molecules23020415.

3.

Metadynamics for Perspective Drug Design: Computationally Driven Synthesis of New Protein-Protein Interaction Inhibitors Targeting the EphA2 Receptor.

Incerti M, Russo S, Callegari D, Pala D, Giorgio C, Zanotti I, Barocelli E, Vicini P, Vacondio F, Rivara S, Castelli R, Tognolini M, Lodola A.

J Med Chem. 2017 Jan 26;60(2):787-796. doi: 10.1021/acs.jmedchem.6b01642. Epub 2017 Jan 5.

PMID:
28005388
4.

Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return.

Russo S, Callegari D, Incerti M, Pala D, Giorgio C, Brunetti J, Bracci L, Vicini P, Barocelli E, Capoferri L, Rivara S, Tognolini M, Mor M, Lodola A.

Chemistry. 2016 Jun 6;22(24):8048-52. doi: 10.1002/chem.201600993. Epub 2016 May 3.

PMID:
27139720
5.

2-Benzisothiazolylimino-5-benzylidene-4-thiazolidinones as protective agents against cartilage destruction.

Crascì L, Vicini P, Incerti M, Cardile V, Avondo S, Panico A.

Bioorg Med Chem. 2015 Apr 1;23(7):1551-6. doi: 10.1016/j.bmc.2015.02.002. Epub 2015 Feb 11.

PMID:
25725607
6.

A new efficient route to 7-aryl-6-fluoro-8-nitroquinolones as potent antibacterial agents.

Al-Trawneh SA, El-Abadelah MM, Al-Abadleh MM, Zani F, Incerti M, Vicini P.

Eur J Med Chem. 2014 Oct 30;86:364-7. doi: 10.1016/j.ejmech.2014.08.065. Epub 2014 Aug 26.

PMID:
25180924
7.

Design synthesis and antibacterial activity studies of new thiadiazoloquinolone compounds.

Al-Qawasmeh RA, Abadleh MM, Zahra JA, El-Abadelah MM, Albashiti R, Zani F, Incerti M, Vicini P.

J Enzyme Inhib Med Chem. 2014 Dec;29(6):777-85. doi: 10.3109/14756366.2013.855925. Epub 2014 Feb 10.

PMID:
24506209
8.

Synthesis and structure-activity relationships of amino acid conjugates of cholanic acid as antagonists of the EphA2 receptor.

Russo S, Incerti M, Tognolini M, Castelli R, Pala D, Hassan-Mohamed I, Giorgio C, De Franco F, Gioiello A, Vicini P, Barocelli E, Rivara S, Mor M, Lodola A.

Molecules. 2013 Oct 21;18(10):13043-60. doi: 10.3390/molecules181013043.

9.

Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor.

Incerti M, Tognolini M, Russo S, Pala D, Giorgio C, Hassan-Mohamed I, Noberini R, Pasquale EB, Vicini P, Piersanti S, Rivara S, Barocelli E, Mor M, Lodola A.

J Med Chem. 2013 Apr 11;56(7):2936-47. doi: 10.1021/jm301890k. Epub 2013 Mar 22.

10.

Structure-activity relationships and mechanism of action of Eph-ephrin antagonists: interaction of cholanic acid with the EphA2 receptor.

Tognolini M, Incerti M, Hassan-Mohamed I, Giorgio C, Russo S, Bruni R, Lelli B, Bracci L, Noberini R, Pasquale EB, Barocelli E, Vicini P, Mor M, Lodola A.

ChemMedChem. 2012 Jun;7(6):1071-83. doi: 10.1002/cmdc.201200102. Epub 2012 Apr 23.

11.

Fragment-based design, docking, synthesis, biological evaluation and structure-activity relationships of 2-benzo/benzisothiazolimino-5-aryliden-4-thiazolidinones as cycloxygenase/lipoxygenase inhibitors.

Eleftheriou P, Geronikaki A, Hadjipavlou-Litina D, Vicini P, Filz O, Filimonov D, Poroikov V, Chaudhaery SS, Roy KK, Saxena AK.

Eur J Med Chem. 2012 Jan;47(1):111-24. doi: 10.1016/j.ejmech.2011.10.029. Epub 2011 Oct 25.

PMID:
22119153
12.

Structure-activity relationships of N-phenyl-N'-benzothiazol-6-ylurea synthetic derivatives: cytokinin-like activity and adventitious rooting enhancement.

Rolli E, Incerti M, Brunoni F, Vicini P, Ricci A.

Phytochemistry. 2012 Feb;74:159-65. doi: 10.1016/j.phytochem.2011.10.012. Epub 2011 Nov 22.

PMID:
22115176
13.

Benzisothiazolyliminothiazolidin-4-ones with chondroprotective properties: searching for potent and selective inhibitors of MMP-13.

Vicini P, Crascì L, Incerti M, Ronsisvalle S, Cardile V, Panico AM.

ChemMedChem. 2011 Jul 4;6(7):1199-202. doi: 10.1002/cmdc.201100223. Epub 2011 Jun 9. No abstract available.

PMID:
21661113
14.

Synthesis and biological evaluation of tetracyclic thienopyridones as antibacterial and antitumor agents.

Al-Trawneh SA, El-Abadelah MM, Zahra JA, Al-Taweel SA, Zani F, Incerti M, Cavazzoni A, Vicini P.

Bioorg Med Chem. 2011 Apr 15;19(8):2541-8. doi: 10.1016/j.bmc.2011.03.018. Epub 2011 Mar 12.

PMID:
21458275
15.

Heteroarylimino-4-thiazolidinones as inhibitors of cartilage degradation.

Panico AM, Vicini P, Geronikaki A, Incerti M, Cardile V, Crascì L, Messina R, Ronsisvalle S.

Bioorg Chem. 2011 Feb;39(1):48-52. doi: 10.1016/j.bioorg.2010.11.002. Epub 2010 Dec 5.

PMID:
21208635
16.

Synthesis and biological evaluation of tetracyclic fluoroquinolones as antibacterial and anticancer agents.

Al-Trawneh SA, Zahra JA, Kamal MR, El-Abadelah MM, Zani F, Incerti M, Cavazzoni A, Alfieri RR, Petronini PG, Vicini P.

Bioorg Med Chem. 2010 Aug 15;18(16):5873-84. doi: 10.1016/j.bmc.2010.06.098. Epub 2010 Jul 3.

PMID:
20667744
17.

4-Methyl-N-(3-oxo-2,3-dihydro-1,2-benzisothia-zol-2-yl)benzene-sulfonamide.

Rizzoli C, Vicini P, Incerti M.

Acta Crystallogr Sect E Struct Rep Online. 2009 Jan 31;65(Pt 2):o425-6. doi: 10.1107/S1600536809003201.

18.

4-Chloro-N-(4-chloro-phenyl-sulfon-yl)-N-(3-oxo-2,3-dihydro-1,2-benzisothia-zol-2-yl)benzene-sulfonamide.

Rizzoli C, Vicini P, Incerti M.

Acta Crystallogr Sect E Struct Rep Online. 2009 Jan 31;65(Pt 2):o416-7. doi: 10.1107/S1600536809003195.

19.

Complete 1H and 13C NMR spectral assignment of benzo[d]isothiazole derivatives and of an isoindole isoster.

Incerti M, Acquotti D, Vicini P.

Magn Reson Chem. 2008 Dec;46(12):1175-9. doi: 10.1002/mrc.2308.

PMID:
18853390
20.

Hybrid molecules between benzenesulfonamides and active antimicrobial benzo[d]isothiazol-3-ones.

Zani F, Incerti M, Ferretti R, Vicini P.

Eur J Med Chem. 2009 Jun;44(6):2741-7. doi: 10.1016/j.ejmech.2008.07.022. Epub 2008 Jul 25.

PMID:
18775586

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