Format
Sort by
Items per page

Send to

Choose Destination

Search results

Items: 1 to 20 of 154

1.

Synthesis of indole based acetohydrazide analogs: Their in vitro and in silico thymidine phosphorylase studies.

Taha M, Aldhamin EAJ, Almandil NB, Anouar EH, Uddin N, Alomari M, Rahim F, Adalat B, Ibrahim M, Nawaz F, Iqbal N, Alghanem B, Altolayyan A, Khan KM.

Bioorg Chem. 2020 Mar 12;98:103745. doi: 10.1016/j.bioorg.2020.103745. [Epub ahead of print]

PMID:
32200327
2.

Exploring efficacy of indole-based dual inhibitors for α-glucosidase and α-amylase enzymes: In silico, biochemical and kinetic studies.

Kawde AN, Taha M, Alansari RS, Almandil NB, Anouar EH, Uddin N, Rahim F, Chigurupati S, Nawaz M, Hayat S, Ibrahim M, Elakurthy PK, Vijayan V, Morsy M, Ibrahim H, Baig N, Khan KM.

Int J Biol Macromol. 2020 Mar 12;154:217-232. doi: 10.1016/j.ijbiomac.2020.03.090. [Epub ahead of print]

PMID:
32173438
3.

Dihydropyridines as potential α-amylase and α-glucosidase inhibitors: Synthesis, in vitro and in silico studies.

Yousuf H, Shamim S, Khan KM, Chigurupati S, Kanwal, Hameed S, Khan MN, Taha M, Arfeen M.

Bioorg Chem. 2020 Mar;96:103581. doi: 10.1016/j.bioorg.2020.103581. Epub 2020 Jan 15.

PMID:
31978686
4.

Biology-oriented drug synthesis (BIODS), in vitro urease inhibitory activity, and in silico studies on ibuprofen derivatives.

Seraj F, Kanwal, Khan KM, Khan A, Ali M, Khalil R, Ul-Haq Z, Hameed S, Taha M, Salar U, Perveen S.

Mol Divers. 2020 Jan 21. doi: 10.1007/s11030-019-10032-x. [Epub ahead of print]

PMID:
31965436
5.

Synthesis, α-glycosidase inhibitory potential and molecular docking study of benzimidazole derivatives.

Taha M, Rahim F, Zaman K, Selvaraj M, Uddin N, Farooq RK, Nawaz M, Sajid M, Nawaz F, Ibrahim M, Khan KM.

Bioorg Chem. 2020 Jan;95:103555. doi: 10.1016/j.bioorg.2019.103555. Epub 2019 Dec 26.

PMID:
31911306
6.

Synthesis and characterization of cadmium-bismuth microspheres for the catalytic and photocatalytic degradation of organic pollutants, with antibacterial, antioxidant and cytotoxicity assay.

Qureshi F, Nawaz M, Rehman S, Almofty SA, Shahzad S, Nissapatorn V, Taha M.

J Photochem Photobiol B. 2020 Jan;202:111723. doi: 10.1016/j.jphotobiol.2019.111723. Epub 2019 Nov 23.

PMID:
31785448
7.

Synthesis, in vitro α-amylase inhibitory, and radicals (DPPH & ABTS) scavenging potentials of new N-sulfonohydrazide substituted indazoles.

Rafique R, Khan KM, Arshia, Chigurupati S, Wadood A, Rehman AU, Salar U, Venugopal V, Shamim S, Taha M, Perveen S.

Bioorg Chem. 2020 Jan;94:103410. doi: 10.1016/j.bioorg.2019.103410. Epub 2019 Oct 31.

PMID:
31732193
8.

Synthesis, in vitro alpha-glucosidase inhibitory potential of benzimidazole bearing bis-Schiff bases and their molecular docking study.

Rahim F, Zaman K, Taha M, Ullah H, Ghufran M, Wadood A, Rehman W, Uddin N, Shah SAA, Sajid M, Nawaz F, Khan KM.

Bioorg Chem. 2020 Jan;94:103394. doi: 10.1016/j.bioorg.2019.103394. Epub 2019 Oct 23.

PMID:
31699396
9.

Synthesis of new isoquinoline-base-oxadiazole derivatives as potent inhibitors of thymidine phosphorylase and molecular docking study.

Zaman K, Rahim F, Taha M, Wadood A, Shah SAA, Ahmed QU, Zakaria ZA.

Sci Rep. 2019 Nov 5;9(1):16015. doi: 10.1038/s41598-019-52100-0.

10.

Synthesis of Novel Triazinoindole-Based Thiourea Hybrid: A Study on α-Glucosidase Inhibitors and Their Molecular Docking.

Taha M, Alshamrani FJ, Rahim F, Hayat S, Ullah H, Zaman K, Imran S, Khan KM, Naz F.

Molecules. 2019 Oct 23;24(21). pii: E3819. doi: 10.3390/molecules24213819.

11.

Atenolol thiourea hybrid as potent urease inhibitors: Design, biology-oriented drug synthesis, inhibitory activity screening, and molecular docking studies.

Wahid S, Jahangir S, Versiani MA, Khan KM, Salar U, Ashraf M, Farzand U, Wadood A, Kanwal, Ashfaq-Ur-Rehaman, Arshia, Taha M, Perveen S.

Bioorg Chem. 2020 Jan;94:103359. doi: 10.1016/j.bioorg.2019.103359. Epub 2019 Oct 13.

PMID:
31640931
12.

New triazinoindole bearing thiazole/oxazole analogues: Synthesis, α-amylase inhibitory potential and molecular docking study.

Rahim F, Tariq S, Taha M, Ullah H, Zaman K, Uddin I, Wadood A, Khan AA, Rehman AU, Uddin N, Zafar S, Shah SAA.

Bioorg Chem. 2019 Nov;92:103284. doi: 10.1016/j.bioorg.2019.103284. Epub 2019 Sep 17.

PMID:
31546207
13.

Synthesis of benzotriazoles derivatives and their dual potential as α-amylase and α-glucosidase inhibitors in vitro: Structure-activity relationship, molecular docking, and kinetic studies.

Hameed S, Kanwal, Seraj F, Rafique R, Chigurupati S, Wadood A, Rehman AU, Venugopal V, Salar U, Taha M, Khan KM.

Eur J Med Chem. 2019 Dec 1;183:111677. doi: 10.1016/j.ejmech.2019.111677. Epub 2019 Sep 5.

PMID:
31514061
14.

Design, synthesis, in vitro evaluation, molecular docking and ADME properties studies of hybrid bis-coumarin with thiadiazole as a new inhibitor of Urease.

Alomari M, Taha M, Imran S, Jamil W, Selvaraj M, Uddin N, Rahim F.

Bioorg Chem. 2019 Nov;92:103235. doi: 10.1016/j.bioorg.2019.103235. Epub 2019 Aug 30.

PMID:
31494327
15.

Synthesis of new indazole based dual inhibitors of α-glucosidase and α-amylase enzymes, their in vitro, in silico and kinetics studies.

Rafique R, Khan KM, Arshia, Kanwal, Chigurupati S, Wadood A, Rehman AU, Karunanidhi A, Hameed S, Taha M, Al-Rashida M.

Bioorg Chem. 2020 Jan;94:103195. doi: 10.1016/j.bioorg.2019.103195. Epub 2019 Aug 23.

PMID:
31451297
16.

Synthesis, anti-leishmanial and molecular docking study of bis-indole derivatives.

Taha M, Uddin I, Gollapalli M, Almandil NB, Rahim F, Farooq RK, Nawaz M, Ibrahim M, Alqahtani MA, Bamarouf YA, Selvaraj M.

BMC Chem. 2019 Aug 6;13(1):102. doi: 10.1186/s13065-019-0617-4. eCollection 2019 Dec.

17.

Indole bearing thiadiazole analogs: synthesis, β-glucuronidase inhibition and molecular docking study.

Almandil NB, Taha M, Gollapalli M, Rahim F, Ibrahim M, Mosaddik A, Anouar EH.

BMC Chem. 2019 Feb 4;13(1):14. doi: 10.1186/s13065-019-0522-x. eCollection 2019 Dec.

18.

Synthesis of quinoline derivatives as diabetic II inhibitors and molecular docking studies.

Taha M, Sultan S, Imran S, Rahim F, Zaman K, Wadood A, Ur Rehman A, Uddin N, Mohammed Khan K.

Bioorg Med Chem. 2019 Sep 15;27(18):4081-4088. doi: 10.1016/j.bmc.2019.07.035. Epub 2019 Jul 20.

PMID:
31378594
19.

2,5-Disubstituted thiadiazoles as potent β-glucuronidase inhibitors; Synthesis, in vitro and in silico studies.

Taha M, Barak Almandil N, Rashid U, Ali M, Ibrahim M, Gollapalli M, Mosaddik A, Mohammed Khan K.

Bioorg Chem. 2019 Oct;91:103126. doi: 10.1016/j.bioorg.2019.103126. Epub 2019 Jul 12.

PMID:
31349116
20.

Synthesis of new arylhydrazide bearing Schiff bases/thiazolidinone: α-Amylase, urease activities and their molecular docking studies.

Rahim F, Taha M, Ullah H, Wadood A, Selvaraj M, Rab A, Sajid M, Shah SAA, Uddin N, Gollapalli M.

Bioorg Chem. 2019 Oct;91:103112. doi: 10.1016/j.bioorg.2019.103112. Epub 2019 Jul 9.

PMID:
31349115

Supplemental Content

Loading ...
Support Center